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CL2012001686A1 - Analogo peptidico de oxintomodulina, en donde el aminoacido c-terminal es opcionalmente amidado; composicion farmaceutica que lo comprende y su uso en la preparacion de un medicamento para el tratamiento de diabetes no insulinodependiente u obesidad. - Google Patents

Analogo peptidico de oxintomodulina, en donde el aminoacido c-terminal es opcionalmente amidado; composicion farmaceutica que lo comprende y su uso en la preparacion de un medicamento para el tratamiento de diabetes no insulinodependiente u obesidad.

Info

Publication number
CL2012001686A1
CL2012001686A1 CL2012001686A CL2012001686A CL2012001686A1 CL 2012001686 A1 CL2012001686 A1 CL 2012001686A1 CL 2012001686 A CL2012001686 A CL 2012001686A CL 2012001686 A CL2012001686 A CL 2012001686A CL 2012001686 A1 CL2012001686 A1 CL 2012001686A1
Authority
CL
Chile
Prior art keywords
obesity
amino acid
preparation
treatment
pharmaceutical composition
Prior art date
Application number
CL2012001686A
Other languages
English (en)
Inventor
Fernandez Jorge Alsina
Wayne David Kohn
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43587001&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2012001686(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of CL2012001686A1 publication Critical patent/CL2012001686A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/605Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/26Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Zoology (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Toxicology (AREA)
  • Obesity (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)

Abstract

ANÁLOGO PEPTÍDICO DE OXIRITOMODUHINA DE SECUANCIA SEQ NO.5 QUE ESTÁ OPCIONALMENTE AMIDADO EN EL AMINOÁCIDO C-TERMINAL; COMPOSICIÓN FARMACÉUTICA QUE LO COMPRENDE Y SU USO EN LA PREPARACIÓN DE UN MEDICAMENTO PARA EL TRATAMIENTO DE DIABETES NO INSULINODEPENDIENTE U OBESIDAD.
CL2012001686A 2009-12-22 2012-06-21 Analogo peptidico de oxintomodulina, en donde el aminoacido c-terminal es opcionalmente amidado; composicion farmaceutica que lo comprende y su uso en la preparacion de un medicamento para el tratamiento de diabetes no insulinodependiente u obesidad. CL2012001686A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28888809P 2009-12-22 2009-12-22
US35257610P 2010-06-08 2010-06-08

Publications (1)

Publication Number Publication Date
CL2012001686A1 true CL2012001686A1 (es) 2012-11-23

Family

ID=43587001

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2012001686A CL2012001686A1 (es) 2009-12-22 2012-06-21 Analogo peptidico de oxintomodulina, en donde el aminoacido c-terminal es opcionalmente amidado; composicion farmaceutica que lo comprende y su uso en la preparacion de un medicamento para el tratamiento de diabetes no insulinodependiente u obesidad.

Country Status (34)

Country Link
US (1) US8367607B2 (es)
EP (1) EP2515928B1 (es)
JP (1) JP5717759B2 (es)
KR (1) KR101399671B1 (es)
CN (1) CN102740873B (es)
AR (1) AR079345A1 (es)
AU (1) AU2010341651B2 (es)
BR (1) BR112012017348B1 (es)
CA (1) CA2784671C (es)
CL (1) CL2012001686A1 (es)
CO (1) CO6551738A2 (es)
CR (1) CR20120338A (es)
DK (1) DK2515928T3 (es)
DO (1) DOP2012000176A (es)
EA (1) EA022820B1 (es)
ES (1) ES2486675T3 (es)
HN (1) HN2012001321A (es)
HR (1) HRP20140616T1 (es)
IL (1) IL220161B (es)
JO (1) JO2976B1 (es)
MA (1) MA33825B1 (es)
MX (1) MX2012007438A (es)
MY (1) MY160773A (es)
NZ (1) NZ600731A (es)
PE (1) PE20121393A1 (es)
PH (1) PH12012501263B1 (es)
PL (1) PL2515928T3 (es)
PT (1) PT2515928E (es)
RS (1) RS53505B1 (es)
SG (1) SG181430A1 (es)
SI (1) SI2515928T1 (es)
TN (1) TN2012000302A1 (es)
TW (1) TWI423812B (es)
WO (1) WO2011087672A1 (es)

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