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BRPI1009090A2 - composto, pró-droga, medicamento, métodos, e, uso do composto - Google Patents

composto, pró-droga, medicamento, métodos, e, uso do composto

Info

Publication number
BRPI1009090A2
BRPI1009090A2 BRPI1009090A BRPI1009090A BRPI1009090A2 BR PI1009090 A2 BRPI1009090 A2 BR PI1009090A2 BR PI1009090 A BRPI1009090 A BR PI1009090A BR PI1009090 A BRPI1009090 A BR PI1009090A BR PI1009090 A2 BRPI1009090 A2 BR PI1009090A2
Authority
BR
Brazil
Prior art keywords
compound
prodrug
medicine
methods
compound use
Prior art date
Application number
BRPI1009090A
Other languages
English (en)
Inventor
Haruyuki Nishida
Ikuo Fujimori
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of BRPI1009090A2 publication Critical patent/BRPI1009090A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BRPI1009090A 2009-03-26 2010-03-25 composto, pró-droga, medicamento, métodos, e, uso do composto BRPI1009090A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2009077078 2009-03-26
PCT/JP2010/055257 WO2010110378A1 (ja) 2009-03-26 2010-03-25 ピラゾール化合物

Publications (1)

Publication Number Publication Date
BRPI1009090A2 true BRPI1009090A2 (pt) 2016-03-01

Family

ID=42781069

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1009090A BRPI1009090A2 (pt) 2009-03-26 2010-03-25 composto, pró-droga, medicamento, métodos, e, uso do composto

Country Status (25)

Country Link
US (1) US8895588B2 (pt)
EP (1) EP2412713B1 (pt)
JP (1) JP5552481B2 (pt)
KR (1) KR101656906B1 (pt)
CN (1) CN102448953B (pt)
AU (1) AU2010228220B2 (pt)
BR (1) BRPI1009090A2 (pt)
CA (1) CA2756086A1 (pt)
CL (1) CL2011002351A1 (pt)
CO (1) CO6460700A2 (pt)
CR (1) CR20110533A (pt)
DO (1) DOP2011000296A (pt)
EA (1) EA019853B1 (pt)
EC (1) ECSP11011419A (pt)
GE (1) GEP20156222B (pt)
IL (1) IL215235A (pt)
MA (1) MA33214B1 (pt)
MX (1) MX2011009943A (pt)
NZ (1) NZ595890A (pt)
PE (1) PE20120618A1 (pt)
SG (1) SG174476A1 (pt)
TN (1) TN2011000474A1 (pt)
UA (1) UA107457C2 (pt)
WO (1) WO2010110378A1 (pt)
ZA (1) ZA201107435B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014003199A1 (en) 2012-06-27 2014-01-03 Takeda Pharmaceutical Company Limited Liquid preparations of amines and organic acids stabilized by salts
EP3524260B1 (en) 2012-09-27 2023-09-13 Elanco Animal Health Incorporated Pharmaceutical compositions for treatment of inappetence
KR20180108916A (ko) 2015-01-28 2018-10-04 아라타나 세라퓨틱스, 인크. 체중-증량 화합물의 장기 사용을 위한 조성물 및 방법
CN105067814A (zh) * 2015-07-24 2015-11-18 中国科学院成都生物研究所 解旋酶水解atp活性测定方法
US11767311B2 (en) * 2020-06-17 2023-09-26 Ildong Pharmaceutical Co., Ltd. Acid secretion inhibitor and use thereof

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3285991A (en) 1963-03-26 1966-11-15 Union Carbide Corp Polyepoxides cured with the reaction product of a dihydroxydiphenylsul-fone, an amine, and an aldehyde
US4847289A (en) 1987-06-08 1989-07-11 Merck & Co., Inc. Thiophene sulfonamide antiglaucoma agents
MX9205392A (es) 1991-10-29 1993-04-01 Du Pont Triazolcarbozamidas herbicidas y procedimiento para su obtencion.
PL183931B1 (pl) 1994-09-26 2002-08-30 Shionogi & Co Nowe związki, pochodne imidazolu i kompozycje farmaceutyczne je zawierające
JPH0948778A (ja) 1995-08-04 1997-02-18 Sagami Chem Res Center 2−置換−3−アルコキシ−5−(ピロール−2−イル)フラン誘導体
WO1997017070A1 (en) 1995-11-06 1997-05-15 University Of Pittsburgh Inhibitors of protein isoprenyl transferases
ATE443698T1 (de) 1996-12-23 2009-10-15 Bristol Myers Squibb Pharma Co Stickstoffhaltige heterocyclen als faktor xa- hemmer
AU1918299A (en) 1998-02-23 1999-09-06 Warner-Lambert Company Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
AU2003254282A1 (en) 2002-08-01 2004-02-23 Nitromed, Inc. Nitrosated proton pump inhibitors, compositions and methods of use
EP1633348B1 (en) 2003-05-02 2008-10-08 Elan Pharmaceuticals, Inc. 4- BROMO - 5 - (2- CHLORO - BENZOYLAMINO) - 1H - PYRAZOLE - 3 - CARBOXYLIC ACID AMIDE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ B sb 1 /sb RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES
EP1628957B1 (en) 2003-05-26 2010-09-29 Takeda Pharmaceutical Company Limited Sulfopyrroles
CA2532800C (en) 2003-07-23 2013-06-18 Exelixis, Inc. Anaplastic lymphoma kinase modulators and methods of use
KR101178747B1 (ko) 2004-09-30 2012-09-03 다케다 야쿠힌 고교 가부시키가이샤 프로톤 펌프 저해제
PT1919865E (pt) 2005-08-30 2011-07-11 Takeda Pharmaceutical Derivados de 1h-pirrole substituídos com 1-heterociclilsulfonilo, 2-aminometilo, 5-(hetero)arilo como inibidores da secreção ácida
EP2005957B1 (en) 2006-03-31 2012-05-30 Takeda Pharmaceutical Company Limited Acid secretion inhibitor
US8933105B2 (en) 2007-02-28 2015-01-13 Takeda Pharmaceutical Company Limited Pyrrole compounds
JP2009077078A (ja) 2007-09-19 2009-04-09 Brother Ind Ltd 位置検出システム
TW200920366A (en) * 2007-09-28 2009-05-16 Takeda Pharmaceutical 5-membered heterocyclic compound
US8334301B2 (en) 2007-09-28 2012-12-18 Takeda Pharmaceutical Company Limited 5-Membered heterocyclic compound
PE20091846A1 (es) 2008-05-19 2009-12-16 Plexxikon Inc DERIVADOS DE PIRROLO[2,3-d]-PIRIMIDINA COMO MODULADORES DE CINASAS
AU2009272486A1 (en) 2008-07-18 2010-01-21 Takeda Pharmaceutical Company Limited. Benzazepine derivatives and their use as hstamine H3 antagonists

Also Published As

Publication number Publication date
EP2412713A4 (en) 2014-04-02
JPWO2010110378A1 (ja) 2012-10-04
CO6460700A2 (es) 2012-06-15
DOP2011000296A (es) 2011-10-15
IL215235A (en) 2014-07-31
MA33214B1 (fr) 2012-04-02
SG174476A1 (en) 2011-10-28
NZ595890A (en) 2013-09-27
AU2010228220A1 (en) 2011-11-17
US20120095057A1 (en) 2012-04-19
ECSP11011419A (es) 2011-11-30
ZA201107435B (en) 2012-08-29
US8895588B2 (en) 2014-11-25
EP2412713B1 (en) 2016-11-30
CA2756086A1 (en) 2010-09-30
AU2010228220A2 (en) 2011-11-24
PE20120618A1 (es) 2012-06-05
AU2010228220B2 (en) 2015-05-21
GEP20156222B (en) 2015-01-26
WO2010110378A1 (ja) 2010-09-30
IL215235A0 (en) 2011-12-29
CR20110533A (es) 2012-02-13
EA019853B1 (ru) 2014-06-30
CN102448953B (zh) 2014-05-07
KR101656906B1 (ko) 2016-09-12
MX2011009943A (es) 2011-10-06
KR20110130483A (ko) 2011-12-05
CL2011002351A1 (es) 2012-07-13
UA107457C2 (uk) 2015-01-12
JP5552481B2 (ja) 2014-07-16
EP2412713A1 (en) 2012-02-01
TN2011000474A1 (en) 2013-03-27
CN102448953A (zh) 2012-05-09
EA201171168A1 (ru) 2012-05-30

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]
B350 Update of information on the portal [chapter 15.35 patent gazette]