BRPI0921148A2 - composto, método para tratar uma infecção bacteriana, e, uso de um composto. - Google Patents
composto, método para tratar uma infecção bacteriana, e, uso de um composto.Info
- Publication number
- BRPI0921148A2 BRPI0921148A2 BRPI0921148A BRPI0921148A BRPI0921148A2 BR PI0921148 A2 BRPI0921148 A2 BR PI0921148A2 BR PI0921148 A BRPI0921148 A BR PI0921148A BR PI0921148 A BRPI0921148 A BR PI0921148A BR PI0921148 A2 BRPI0921148 A2 BR PI0921148A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- treating
- bacterial infection
- bacterial
- infection
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US11470608P | 2008-11-14 | 2008-11-14 | |
| US16384809P | 2009-03-26 | 2009-03-26 | |
| PCT/GB2009/051532 WO2010055348A1 (en) | 2008-11-14 | 2009-11-13 | [4- (1-amino-ethyl) -cyclohexyl] -methyl-amines as antibacterials |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0921148A2 true BRPI0921148A2 (pt) | 2016-02-23 |
Family
ID=41463108
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0921148A BRPI0921148A2 (pt) | 2008-11-14 | 2009-11-13 | composto, método para tratar uma infecção bacteriana, e, uso de um composto. |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20110288084A1 (pt) |
| EP (1) | EP2370444A1 (pt) |
| JP (1) | JP2012508789A (pt) |
| KR (1) | KR20110093797A (pt) |
| CN (1) | CN102216308A (pt) |
| AR (1) | AR074340A1 (pt) |
| AU (1) | AU2009315425A1 (pt) |
| BR (1) | BRPI0921148A2 (pt) |
| CA (1) | CA2742520A1 (pt) |
| CO (1) | CO6382113A2 (pt) |
| CR (1) | CR20110256A (pt) |
| CU (1) | CU20110108A7 (pt) |
| EA (1) | EA201100754A1 (pt) |
| EC (1) | ECSP11011053A (pt) |
| IL (1) | IL211941A0 (pt) |
| MX (1) | MX2011005106A (pt) |
| TW (1) | TW201022279A (pt) |
| UY (1) | UY32247A (pt) |
| WO (1) | WO2010055348A1 (pt) |
| ZA (1) | ZA201104395B (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2723737A1 (en) * | 2011-06-27 | 2014-04-30 | Kyorin Pharmaceutical Co., Ltd. | Bridged bicyclic compounds for the treatment of bacterial infections |
| AR096135A1 (es) * | 2013-05-02 | 2015-12-09 | Actelion Pharmaceuticals Ltd | Derivados de la quinolona |
| TW201722965A (zh) * | 2015-08-16 | 2017-07-01 | 葛蘭素史密斯克藍智慧財產發展有限公司 | 用於抗菌應用之化合物 |
| TW201711999A (zh) | 2015-09-03 | 2017-04-01 | 佛瑪治療公司 | ﹝6,6﹞稠合雙環組蛋白脫乙醯基酶8(hdac8)抑制劑 |
| PL3468975T3 (pl) * | 2016-06-08 | 2020-09-07 | Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A. | Nowe związki przeciwbakteryjne |
| FI3634968T3 (fi) * | 2017-06-08 | 2023-04-26 | Bugworks Res Inc | Bakteerilääkkeinä käyttökelpoisia heterosyklisiä yhdisteitä ja menetelmä niiden valmistamiseksi |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY150958A (en) * | 2005-06-16 | 2014-03-31 | Astrazeneca Ab | Compounds for the treatment of multi-drug resistant bacterial infections |
| CA2652501C (en) * | 2006-05-26 | 2014-07-08 | Toyama Chemical Co., Ltd. | Novel heterocyclic compound or salt thereof and intermediate thereof |
| CL2007003693A1 (es) * | 2006-12-22 | 2008-06-27 | Actelion Pharmaceuticals Ltd | Compuestos derivados de pirido [3,2-b] [1,4] tiazina; composicion farmaceutica que contiene dichos compuestos; y su uso en el tratamiento de infecciones bacterianas. |
-
2009
- 2009-11-12 TW TW098138483A patent/TW201022279A/zh unknown
- 2009-11-13 KR KR1020117010967A patent/KR20110093797A/ko not_active Withdrawn
- 2009-11-13 MX MX2011005106A patent/MX2011005106A/es not_active Application Discontinuation
- 2009-11-13 US US13/128,596 patent/US20110288084A1/en not_active Abandoned
- 2009-11-13 AU AU2009315425A patent/AU2009315425A1/en not_active Abandoned
- 2009-11-13 UY UY0001032247A patent/UY32247A/es not_active Application Discontinuation
- 2009-11-13 WO PCT/GB2009/051532 patent/WO2010055348A1/en not_active Ceased
- 2009-11-13 EA EA201100754A patent/EA201100754A1/ru unknown
- 2009-11-13 JP JP2011543815A patent/JP2012508789A/ja active Pending
- 2009-11-13 CN CN2009801457755A patent/CN102216308A/zh active Pending
- 2009-11-13 CA CA2742520A patent/CA2742520A1/en not_active Abandoned
- 2009-11-13 EP EP09753199A patent/EP2370444A1/en not_active Withdrawn
- 2009-11-13 AR ARP090104378A patent/AR074340A1/es unknown
- 2009-11-13 BR BRPI0921148A patent/BRPI0921148A2/pt not_active Application Discontinuation
-
2011
- 2011-03-24 IL IL211941A patent/IL211941A0/en unknown
- 2011-05-11 CO CO11058050A patent/CO6382113A2/es not_active Application Discontinuation
- 2011-05-13 EC EC2011011053A patent/ECSP11011053A/es unknown
- 2011-05-13 CU CU20110108A patent/CU20110108A7/es unknown
- 2011-05-13 CR CR20110256A patent/CR20110256A/es not_active Application Discontinuation
- 2011-06-13 ZA ZA2011/04395A patent/ZA201104395B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TW201022279A (en) | 2010-06-16 |
| US20110288084A1 (en) | 2011-11-24 |
| ZA201104395B (en) | 2012-03-28 |
| EP2370444A1 (en) | 2011-10-05 |
| KR20110093797A (ko) | 2011-08-18 |
| WO2010055348A1 (en) | 2010-05-20 |
| CU20110108A7 (es) | 2012-01-31 |
| CN102216308A (zh) | 2011-10-12 |
| CA2742520A1 (en) | 2010-05-20 |
| EA201100754A1 (ru) | 2012-01-30 |
| ECSP11011053A (es) | 2011-06-30 |
| CR20110256A (es) | 2011-07-04 |
| CO6382113A2 (es) | 2012-02-15 |
| MX2011005106A (es) | 2011-05-30 |
| IL211941A0 (en) | 2011-06-30 |
| UY32247A (es) | 2010-06-30 |
| JP2012508789A (ja) | 2012-04-12 |
| AR074340A1 (es) | 2011-01-12 |
| AU2009315425A1 (en) | 2010-05-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |