BRPI0911659B8 - composto 3-fenilpirazolo[5,1-b]tiazol e composição farmacêutica compreendendo o mesmo - Google Patents

composto 3-fenilpirazolo[5,1-b]tiazol e composição farmacêutica compreendendo o mesmo

Info

Publication number: BRPI0911659B8
Authority: BR; Brazil
Prior art keywords: phenylpyrazolo; same; pharmaceutical composition; thiazole compound; cycloalkyl
Prior art date: 2008-04-15

Application number

BRPI0911659A

Other languages

English (en)

Portuguese (pt)

Inventor

Inomata Akira

Shibata Hisashi

Shikata Kodo

Shin Kogyoku

Takeda Kunitoshi

Hashizume Minako

Terauchi Taro

Takahashi Yoshinori

Original Assignee

Eisai R&D Man Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-04-15

Filing date

2009-04-09

Publication date

2021-05-25

2009-04-09 Application filed by Eisai R&D Man Co Ltd filed Critical Eisai R&D Man Co Ltd

2015-10-13 Publication of BRPI0911659A2 publication Critical patent/BRPI0911659A2/pt

2020-08-25 Publication of BRPI0911659B1 publication Critical patent/BRPI0911659B1/pt

2021-05-25 Publication of BRPI0911659B8 publication Critical patent/BRPI0911659B8/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Psychiatry (AREA)
Heart & Thoracic Surgery (AREA)
Addiction (AREA)
Cardiology (AREA)
Pain & Pain Management (AREA)
Vascular Medicine (AREA)
Anesthesiology (AREA)
Hospice & Palliative Care (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)

BRPI0911659A 2008-04-15 2009-04-09 composto 3-fenilpirazolo[5,1-b]tiazol e composição farmacêutica compreendendo o mesmo BRPI0911659B8 (pt)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
US4508408P	2008-04-15	2008-04-15
US61/045,084		2008-04-15
JP2008106080		2008-04-15
JP2008-106080		2008-04-15
PCT/JP2009/057270 WO2009128383A1 (fr)	2008-04-15	2009-04-09	COMPOSÉ DE 3-PHÉNYLPYRAZOLO[5,1-b]THIAZOLE

Publications (3)

Publication Number	Publication Date
BRPI0911659A2 BRPI0911659A2 (pt)	2015-10-13
BRPI0911659B1 BRPI0911659B1 (pt)	2020-08-25
BRPI0911659B8 true BRPI0911659B8 (pt)	2021-05-25

Family

ID=41164535

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0911659A BRPI0911659B8 (pt)	2008-04-15	2009-04-09	composto 3-fenilpirazolo[5,1-b]tiazol e composição farmacêutica compreendendo o mesmo

Country Status (28)

Country	Link
US (1)	US8431603B2 (fr)
EP (1)	EP2266990B1 (fr)
JP (1)	JP4654325B2 (fr)
KR (1)	KR101601994B1 (fr)
CN (1)	CN102007133B (fr)
AR (1)	AR071655A1 (fr)
AU (1)	AU2009237050B2 (fr)
BR (1)	BRPI0911659B8 (fr)
CA (1)	CA2721670C (fr)
CL (1)	CL2009000896A1 (fr)
CY (1)	CY1113484T1 (fr)
DK (1)	DK2266990T3 (fr)
ES (1)	ES2396126T3 (fr)
HR (1)	HRP20121021T1 (fr)
IL (1)	IL208393A (fr)
MX (1)	MX2010011089A (fr)
MY (1)	MY152687A (fr)
NZ (1)	NZ588376A (fr)
PE (1)	PE20091890A1 (fr)
PL (1)	PL2266990T3 (fr)
PT (1)	PT2266990E (fr)
RS (1)	RS52561B (fr)
RU (1)	RU2482120C2 (fr)
SI (1)	SI2266990T1 (fr)
TW (1)	TW201004964A (fr)
UA (1)	UA101836C2 (fr)
WO (1)	WO2009128383A1 (fr)
ZA (1)	ZA201006764B (fr)

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BRPI0313976B8 (pt)	2002-10-22	2021-05-25	Eisai Co Ltd	compostos de 7-fenilpirazolopiridina e uso dos mesmos na preparação de agente terapêutico ou profilático para doenças associadas com o crf ou seus receptores
WO2005063756A1 (fr) *	2003-12-22	2005-07-14	Sb Pharmco Puerto Rico Inc	Antagonistes du recepteur de crf et procedes correspondants
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PL2266990T3 (pl)	2008-04-15	2013-03-29	Eisai R&D Man Co Ltd	ZWIĄZEK 3-FENYLOPIRAZOLO[5,1-b] TIAZOLOWY
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TWI358017B (en)	2009-12-17	2012-02-11	Askey Computer Corp	Electronic device loading base

2009
- 2009-04-09 PL PL09732907T patent/PL2266990T3/pl unknown
- 2009-04-09 CA CA2721670A patent/CA2721670C/fr active Active
- 2009-04-09 RS RS20120562A patent/RS52561B/sr unknown
- 2009-04-09 KR KR1020107019769A patent/KR101601994B1/ko not_active Expired - Fee Related
- 2009-04-09 AU AU2009237050A patent/AU2009237050B2/en not_active Ceased
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- 2009-04-09 NZ NZ588376A patent/NZ588376A/en not_active IP Right Cessation
- 2009-04-09 US US12/421,182 patent/US8431603B2/en not_active Expired - Fee Related
- 2009-04-09 WO PCT/JP2009/057270 patent/WO2009128383A1/fr not_active Ceased
- 2009-04-09 EP EP09732907A patent/EP2266990B1/fr active Active
- 2009-04-09 JP JP2010508183A patent/JP4654325B2/ja not_active Expired - Fee Related
- 2009-04-09 SI SI200930453T patent/SI2266990T1/sl unknown
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- 2009-04-09 BR BRPI0911659A patent/BRPI0911659B8/pt not_active IP Right Cessation
- 2009-04-09 DK DK09732907.2T patent/DK2266990T3/da active
- 2009-04-09 HR HRP20121021AT patent/HRP20121021T1/hr unknown
- 2009-04-09 ES ES09732907T patent/ES2396126T3/es active Active
- 2009-04-09 RU RU2010146240/04A patent/RU2482120C2/ru active
- 2009-04-09 MX MX2010011089A patent/MX2010011089A/es active IP Right Grant
- 2009-04-09 PT PT97329072T patent/PT2266990E/pt unknown
- 2009-04-10 TW TW098112062A patent/TW201004964A/zh unknown
- 2009-04-13 PE PE2009000505A patent/PE20091890A1/es not_active Application Discontinuation
- 2009-04-13 AR ARP090101280A patent/AR071655A1/es not_active Application Discontinuation
- 2009-04-14 CL CL2009000896A patent/CL2009000896A1/es unknown
- 2009-09-04 UA UAA201013461A patent/UA101836C2/ru unknown
2010
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Also Published As

Publication number	Publication date
US20090259049A1 (en)	2009-10-15
UA101836C2 (en)	2013-05-13
ES2396126T3 (es)	2013-02-19
CN102007133B (zh)	2013-06-12
BRPI0911659B1 (pt)	2020-08-25
TW201004964A (en)	2010-02-01
EP2266990B1 (fr)	2012-09-26
PE20091890A1 (es)	2009-12-20
CN102007133A (zh)	2011-04-06
RS52561B (sr)	2013-04-30
CA2721670A1 (fr)	2009-10-22
HRP20121021T1 (hr)	2013-01-31
EP2266990A4 (fr)	2011-08-03
BRPI0911659A2 (pt)	2015-10-13
IL208393A0 (en)	2010-12-30
IL208393A (en)	2013-08-29
AU2009237050B2 (en)	2013-04-11
SI2266990T1 (sl)	2013-01-31
PT2266990E (pt)	2012-12-27
HK1150310A1 (en)	2011-11-25
HK1151797A1 (en)	2012-02-10
US8431603B2 (en)	2013-04-30
JP4654325B2 (ja)	2011-03-16
ZA201006764B (en)	2012-03-28
RU2482120C2 (ru)	2013-05-20
AU2009237050A1 (en)	2009-10-22
RU2010146240A (ru)	2012-05-20
CY1113484T1 (el)	2016-06-22
MY152687A (en)	2014-10-31
CA2721670C (fr)	2013-09-10
AR071655A1 (es)	2010-07-07
DK2266990T3 (da)	2013-01-07
JPWO2009128383A1 (ja)	2011-08-04
MX2010011089A (es)	2010-11-05
KR20110002007A (ko)	2011-01-06
WO2009128383A1 (fr)	2009-10-22
KR101601994B1 (ko)	2016-03-17
PL2266990T3 (pl)	2013-03-29
NZ588376A (en)	2011-06-30
EP2266990A1 (fr)	2010-12-29
CL2009000896A1 (es)	2010-04-16

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BR122013025375B8 (pt)	2021-05-25	compostos orgânicos, seus métodos de preparo e uso, bem como composições farmacêuticas
DK2074120T3 (da)	2010-06-14	Tropan-forbindelser
BRPI1009637A2 (pt)	2019-04-30	composto, composição e uso de um composto
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BR112012009861A2 (pt)	2015-09-29	composto, composição farmacêutica, e, uso do composto.
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