BRPI0817305A2 - Sal de amina orgânica, e, processo para produzir um sal de amina orgânica. - Google Patents
Sal de amina orgânica, e, processo para produzir um sal de amina orgânica.Info
- Publication number
- BRPI0817305A2 BRPI0817305A2 BRPI0817305A BRPI0817305A2 BR PI0817305 A2 BRPI0817305 A2 BR PI0817305A2 BR PI0817305 A BRPI0817305 A BR PI0817305A BR PI0817305 A2 BRPI0817305 A2 BR PI0817305A2
- Authority
- BR
- Brazil
- Prior art keywords
- organic amine
- amine salt
- produce
- salt
- organic
- Prior art date
Links
- -1 amine salt Chemical class 0.000 title 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2007251191 | 2007-09-27 | ||
| JP2007-251191 | 2007-09-27 | ||
| PCT/JP2008/067251 WO2009041473A1 (ja) | 2007-09-27 | 2008-09-25 | 6-フルオロ-3-ヒドロキシ-2-ピラジンカルボニトリルの有機アミン塩およびその製造法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0817305A2 true BRPI0817305A2 (pt) | 2015-03-17 |
| BRPI0817305B1 BRPI0817305B1 (pt) | 2021-10-19 |
Family
ID=40511356
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0817305-2A BRPI0817305B1 (pt) | 2007-09-27 | 2008-09-25 | Sal de dicicloexilamina, e, processo para produzir um sal de dicicloexilamina |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US8168789B2 (pt) |
| EP (1) | EP2192117B1 (pt) |
| JP (1) | JP5550347B2 (pt) |
| KR (2) | KR101574567B1 (pt) |
| CN (2) | CN104672153B (pt) |
| AU (1) | AU2008304956B2 (pt) |
| BR (1) | BRPI0817305B1 (pt) |
| CA (1) | CA2700490C (pt) |
| CY (1) | CY1115218T1 (pt) |
| DK (1) | DK2192117T3 (pt) |
| ES (1) | ES2470740T3 (pt) |
| HR (1) | HRP20140837T1 (pt) |
| IL (1) | IL204516A (pt) |
| MX (1) | MX2010003333A (pt) |
| NZ (1) | NZ584157A (pt) |
| PL (1) | PL2192117T3 (pt) |
| PT (1) | PT2192117E (pt) |
| RU (1) | RU2470924C2 (pt) |
| SI (1) | SI2192117T1 (pt) |
| WO (1) | WO2009041473A1 (pt) |
| ZA (1) | ZA201002001B (pt) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY161429A (en) | 2010-09-30 | 2017-04-14 | Toyama Chemical Co Ltd | Sodium salt of 6-fluoro-3-hydroxy-2-pyrazine carboxamide |
| RS54642B1 (sr) | 2010-09-30 | 2016-08-31 | Toyama Chemical Co., Ltd. | Meglumin so 6-fluor-3-hidroksi-2-pirazin karboksamida |
| MX2013005179A (es) * | 2010-11-12 | 2013-07-05 | Fujifilm Corp | Derivado de pirazino[2,3-d]isoxazol. |
| CN104496917B (zh) * | 2014-12-15 | 2017-06-20 | 南京华威医药科技开发有限公司 | 一种法匹拉韦的合成方法 |
| HK1248236A1 (zh) * | 2015-06-09 | 2018-10-12 | 富士胶片富山化学株式会社 | 6-溴-3-羟基-2-吡嗪甲酰胺的结晶及其制造方法 |
| CN107641106A (zh) * | 2016-07-22 | 2018-01-30 | 大连鸿凯化工科技发展有限公司 | 法匹拉韦中间体以及法匹拉韦的合成方法 |
| CN113248450B (zh) * | 2020-02-07 | 2024-04-12 | 北京四环制药有限公司 | 一种法匹拉韦的制备方法 |
| WO2021260516A1 (en) * | 2020-06-22 | 2021-12-30 | Pi Industries Ltd. | An organic amine salt of favipiravir and a process for the purification of favipiravir |
| KR20230034848A (ko) * | 2020-07-06 | 2023-03-10 | 옵티머스 드럭스 (피) 엘티디 | 파비피라비르의 합성 |
| CN114057656B (zh) * | 2020-08-05 | 2025-11-18 | 广东东阳光药业股份有限公司 | 一种法匹拉韦共晶及其制备方法 |
| CN112645889A (zh) * | 2020-12-24 | 2021-04-13 | 杭州煌森生物科技有限公司 | 一种法匹拉韦的精制方法 |
| CN114478404A (zh) * | 2022-03-17 | 2022-05-13 | 浙江海正药业股份有限公司 | 一种法维拉韦中间体羟基物的纯化方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB879259A (en) | 1956-11-20 | 1961-10-11 | Riker Laboratories Inc | Acid addition salts of 2-dimethylaminoethanol and central nervous system stimulant compositions containing them |
| CZ282939B6 (cs) * | 1992-03-04 | 1997-11-12 | Lonza A.G. | Mikrobiologický způsob hydroxylace dusíkatých heterocyklických karboxylových kyselin |
| PT1256588E (pt) * | 2000-02-16 | 2005-05-31 | Toyama Chemical Co Ltd | Derivados de pirazina originais ou os seus sais, preparacoes farmaceuticas, contendo os derivados ou os seus sais e produtos intermedios para a preparacao de ambos |
| RU2297414C2 (ru) * | 2001-02-14 | 2007-04-20 | Тояма Кемикал Ко., Лтд. | Производные пиразина или их соли, фармацевтическая композиция, содержащая данные соединения, и промежуточные соединения для их получения |
| JP4398631B2 (ja) | 2002-07-12 | 2010-01-13 | 富山化学工業株式会社 | 新規なピラジン誘導体またはその塩並びにそれらを含有する抗ウイルス剤 |
| GB0407908D0 (en) | 2004-04-07 | 2004-05-12 | Univ York | Ionic liquids |
-
2008
- 2008-09-25 PT PT88328166T patent/PT2192117E/pt unknown
- 2008-09-25 SI SI200831283T patent/SI2192117T1/sl unknown
- 2008-09-25 US US12/679,496 patent/US8168789B2/en active Active
- 2008-09-25 AU AU2008304956A patent/AU2008304956B2/en active Active
- 2008-09-25 BR BRPI0817305-2A patent/BRPI0817305B1/pt active IP Right Grant
- 2008-09-25 KR KR1020107006533A patent/KR101574567B1/ko active Active
- 2008-09-25 MX MX2010003333A patent/MX2010003333A/es active IP Right Grant
- 2008-09-25 WO PCT/JP2008/067251 patent/WO2009041473A1/ja not_active Ceased
- 2008-09-25 NZ NZ584157A patent/NZ584157A/en unknown
- 2008-09-25 KR KR1020157022432A patent/KR101686813B1/ko active Active
- 2008-09-25 CA CA2700490A patent/CA2700490C/en active Active
- 2008-09-25 CN CN201510024656.1A patent/CN104672153B/zh active Active
- 2008-09-25 EP EP08832816.6A patent/EP2192117B1/en active Active
- 2008-09-25 DK DK08832816.6T patent/DK2192117T3/da active
- 2008-09-25 CN CN200880109041A patent/CN101809003A/zh active Pending
- 2008-09-25 HR HRP20140837AT patent/HRP20140837T1/hr unknown
- 2008-09-25 PL PL08832816T patent/PL2192117T3/pl unknown
- 2008-09-25 ES ES08832816.6T patent/ES2470740T3/es active Active
- 2008-09-25 JP JP2009534345A patent/JP5550347B2/ja active Active
- 2008-09-25 RU RU2010116390/04A patent/RU2470924C2/ru active
-
2010
- 2010-03-16 IL IL204516A patent/IL204516A/en active IP Right Grant
- 2010-03-19 ZA ZA2010/02001A patent/ZA201002001B/en unknown
-
2014
- 2014-07-01 CY CY20141100481T patent/CY1115218T1/el unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B25A | Requested transfer of rights approved |
Owner name: FUJIFILM TOYAMA CHEMICAL CO., LTD. (JP) |
|
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] |
Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
|
| B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] | ||
| B12B | Appeal against refusal [chapter 12.2 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 25/09/2008, OBSERVADAS AS CONDICOES LEGAIS. PATENTE CONCEDIDA CONFORME ADI 5.529/DF, QUE DETERMINA A ALTERACAO DO PRAZO DE CONCESSAO. |