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GB879259A - Acid addition salts of 2-dimethylaminoethanol and central nervous system stimulant compositions containing them - Google Patents

Acid addition salts of 2-dimethylaminoethanol and central nervous system stimulant compositions containing them

Info

Publication number
GB879259A
GB879259A GB35979/57A GB3597957A GB879259A GB 879259 A GB879259 A GB 879259A GB 35979/57 A GB35979/57 A GB 35979/57A GB 3597957 A GB3597957 A GB 3597957A GB 879259 A GB879259 A GB 879259A
Authority
GB
United Kingdom
Prior art keywords
acid
dimethylaminoethanol
neutral
salts
addition salts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB35979/57A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Riker Laboratories Inc
Original Assignee
Riker Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Riker Laboratories Inc filed Critical Riker Laboratories Inc
Publication of GB879259A publication Critical patent/GB879259A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/20Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/14Quaternary ammonium compounds, e.g. edrophonium, choline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/205Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • A61K31/24Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
    • A61K31/245Amino benzoic acid types, e.g. procaine, novocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Adsorbates of 2-dimethylaminoethanol or cation-exchange resins include the adsorbates or "Dowex" 1-150 (a sulphonated copolymer of styrene and divinyl benzene) and "Amberlite" IRC-50 (a copolymer material having free carboxylic groups). ("Amberlite" and "Dowex" are Registered Trade Marks).ALSO:The invention comprises the lactate, acetate, ascorbate, nicotinate, neutral and acid citrates, neutral and acid tartarates, salicylate, adenosinate, creatinate, succinate, neutral and acid fumarates, phthalate, l-methionine, l-arginine, l-tryptophane, d-pantothenate, benzoate propionate, pyruvate, betaresorcylate, p-acetylaminobenzoate, 3,4,5,-trimethoxybenzoate ortho-aminosalicylate, meta-aminosalicylate and para-aminosalicylate salts of 2-dimethylaminoethanol, an adsorbate of 2-dimethylaminoethanol or a cation-exchange resin (see Group IV(a)) and pharmaceutical preparations containing salts of dimethylaminoethanol (see Group VI). The specific salts of the invention are prepared from the base and the appropriate acid.ALSO:Pharmaceutical compositions comprise either 2-dimethylamino ethanol or acid addition salts thereof and a pharmaceutical carrier in unit closage form or 2-dimethylamino ethanol acid addition salts other than the gallate or the p-aminobenzoate and a pharmaceutical carrier. The compositions may contain other active ingredients such as d-pantothenic acid, l-methionine, pyridoxine or cyanocobalamin. Examples are given of a tablet containing the acid tartrate, an elixir containing the betaresorcylate, an aqueous sterile solution for injection containing the neutral tartrate. A dry filled capsule containing the gallate, a capsule containing a solution of the salicylate in peanut oil, an aerosol preparation containing the base, a tablet containing the p-acetylamino benzoate together with pyridoxine, d-calcium pantothenate and l-methionine and a sterile solution for injection containing the hydrochloride salt, cyanocobaltamin, d-calcium pantathenate and pyridoxine.
GB35979/57A 1956-11-20 1957-11-19 Acid addition salts of 2-dimethylaminoethanol and central nervous system stimulant compositions containing them Expired GB879259A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US879259XA 1956-11-20 1956-11-20

Publications (1)

Publication Number Publication Date
GB879259A true GB879259A (en) 1961-10-11

Family

ID=22208091

Family Applications (1)

Application Number Title Priority Date Filing Date
GB35979/57A Expired GB879259A (en) 1956-11-20 1957-11-19 Acid addition salts of 2-dimethylaminoethanol and central nervous system stimulant compositions containing them

Country Status (1)

Country Link
GB (1) GB879259A (en)

Cited By (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3275643A (en) * 1963-07-19 1966-09-27 Irwin I Lubowe Allantoin-pantothenate compounds
FR2068522A1 (en) * 1969-08-28 1971-08-27 Newport Pharmaceuticals
FR2168245A1 (en) * 1972-01-21 1973-08-31 Eurap Sa Dimethylamino ethanol pyridinecarboxylate - cholinergic and antiinflammatory
FR2295742A1 (en) * 1974-12-24 1976-07-23 Francaise Coop Pharma N-methyl colamine pantothenate compsns - used to stimulate acetyl choline synthesis, e.g. to treat atropinic side effects of drugs
EP0217258A3 (en) * 1985-09-28 1989-12-13 Massachusetts Institute Of Technology The use of choline or choline releasing compounds in the production of pharmacological compositions capable of reducing fatigue
FR2684297A1 (en) * 1991-11-28 1993-06-04 Bfb USE OF SULFUR AMINO ACID FOR THE PREPARATION OF A MEDICINAL PRODUCT FOR THE TREATMENT OF ECZEMA.
US5364885A (en) * 1992-11-13 1994-11-15 Ahluwalia Gurpreet S Reduction of hair growth
WO1996012696A1 (en) * 1994-10-20 1996-05-02 Prospa B.V. Salts of omega-3-polyunsaturated fatty acids and pharmaceutical formulations containing them
WO2005074946A1 (en) * 2004-02-10 2005-08-18 Adenobio N.V. Stable and active complexes of adenosine and adenosine phosphates with aminoalcohols for the treatment of pulmonary artery hypertension, cardiac failure and other diseases
WO2008044099A1 (en) * 2006-10-09 2008-04-17 Carlo Ghisalberti Charge transfer complexes in the treatment of inflammatory bowel diseases
CN102344379A (en) * 2004-04-07 2012-02-08 约克大学 Ionic liquids containing nitrogen-containing cations
US8168789B2 (en) 2007-09-27 2012-05-01 Toyama Chemical Co., Ltd. Organic amine salt of 6-fluoro-3-hydroxy-2-pyrazinecarbonitrile and method for producing the same
CN108658793A (en) * 2018-06-25 2018-10-16 安徽大学 Synthesis process of di (dimethylaminoethyl) phthalate

Cited By (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3275643A (en) * 1963-07-19 1966-09-27 Irwin I Lubowe Allantoin-pantothenate compounds
FR2068522A1 (en) * 1969-08-28 1971-08-27 Newport Pharmaceuticals
FR2168245A1 (en) * 1972-01-21 1973-08-31 Eurap Sa Dimethylamino ethanol pyridinecarboxylate - cholinergic and antiinflammatory
FR2295742A1 (en) * 1974-12-24 1976-07-23 Francaise Coop Pharma N-methyl colamine pantothenate compsns - used to stimulate acetyl choline synthesis, e.g. to treat atropinic side effects of drugs
EP0217258A3 (en) * 1985-09-28 1989-12-13 Massachusetts Institute Of Technology The use of choline or choline releasing compounds in the production of pharmacological compositions capable of reducing fatigue
FR2684297A1 (en) * 1991-11-28 1993-06-04 Bfb USE OF SULFUR AMINO ACID FOR THE PREPARATION OF A MEDICINAL PRODUCT FOR THE TREATMENT OF ECZEMA.
EP0545759A1 (en) * 1991-11-28 1993-06-09 Société BFB Use of a sulfur containing amino acid, eventually in combination with pyridoxine, for the preparation of a medicament for the treatment of eczema
US5364885A (en) * 1992-11-13 1994-11-15 Ahluwalia Gurpreet S Reduction of hair growth
WO1996012696A1 (en) * 1994-10-20 1996-05-02 Prospa B.V. Salts of omega-3-polyunsaturated fatty acids and pharmaceutical formulations containing them
WO2005074946A1 (en) * 2004-02-10 2005-08-18 Adenobio N.V. Stable and active complexes of adenosine and adenosine phosphates with aminoalcohols for the treatment of pulmonary artery hypertension, cardiac failure and other diseases
US7585850B2 (en) 2004-02-10 2009-09-08 Adenobio N.V. Stable and active complexes of adenosine and adenosine phosphates with aminoalcohols for the treatment of pulmonary artery hypertension, cardiac failure and other diseases
CN102344379A (en) * 2004-04-07 2012-02-08 约克大学 Ionic liquids containing nitrogen-containing cations
US8784686B2 (en) 2004-04-07 2014-07-22 Innovia Films Limited Liquids
US8992798B2 (en) 2004-04-07 2015-03-31 Innovia Films Limited Liquids
US9328220B2 (en) 2004-04-07 2016-05-03 Innovia Films Limited Liquids
WO2008044099A1 (en) * 2006-10-09 2008-04-17 Carlo Ghisalberti Charge transfer complexes in the treatment of inflammatory bowel diseases
US8168789B2 (en) 2007-09-27 2012-05-01 Toyama Chemical Co., Ltd. Organic amine salt of 6-fluoro-3-hydroxy-2-pyrazinecarbonitrile and method for producing the same
CN108658793A (en) * 2018-06-25 2018-10-16 安徽大学 Synthesis process of di (dimethylaminoethyl) phthalate

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