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BR9916906A - Composto, composição farmacêutica, uso de umcomposto, métodos de tratamento ou profilaxiade, distúrbios psicóticos ou distúrbios deenfraquecimento intelectual, e de tratamento ouprofilaxia de doenças ou condições humanas emque a ativação do receptor alfa-7 nicotìnico ébenéfica, e, processo para preparar um composto - Google Patents

Composto, composição farmacêutica, uso de umcomposto, métodos de tratamento ou profilaxiade, distúrbios psicóticos ou distúrbios deenfraquecimento intelectual, e de tratamento ouprofilaxia de doenças ou condições humanas emque a ativação do receptor alfa-7 nicotìnico ébenéfica, e, processo para preparar um composto

Info

Publication number
BR9916906A
BR9916906A BR9916906-1A BR9916906A BR9916906A BR 9916906 A BR9916906 A BR 9916906A BR 9916906 A BR9916906 A BR 9916906A BR 9916906 A BR9916906 A BR 9916906A
Authority
BR
Brazil
Prior art keywords
compound
alkyl
treatment
prophylaxis
zero
Prior art date
Application number
BR9916906-1A
Other languages
English (en)
Portuguese (pt)
Inventor
James Loch Iii
George Mullen
Eifion Phillips
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BR9916906A publication Critical patent/BR9916906A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34Tobacco-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BR9916906-1A 1999-01-15 1999-12-23 Composto, composição farmacêutica, uso de umcomposto, métodos de tratamento ou profilaxiade, distúrbios psicóticos ou distúrbios deenfraquecimento intelectual, e de tratamento ouprofilaxia de doenças ou condições humanas emque a ativação do receptor alfa-7 nicotìnico ébenéfica, e, processo para preparar um composto BR9916906A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9900100A SE9900100D0 (sv) 1999-01-15 1999-01-15 New compounds
PCT/SE1999/002478 WO2000042044A1 (fr) 1999-01-15 1999-12-23 Nouvelles aralkylamines de spirofuropyridines utiles en therapie

Publications (1)

Publication Number Publication Date
BR9916906A true BR9916906A (pt) 2001-10-30

Family

ID=20414101

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9916906-1A BR9916906A (pt) 1999-01-15 1999-12-23 Composto, composição farmacêutica, uso de umcomposto, métodos de tratamento ou profilaxiade, distúrbios psicóticos ou distúrbios deenfraquecimento intelectual, e de tratamento ouprofilaxia de doenças ou condições humanas emque a ativação do receptor alfa-7 nicotìnico ébenéfica, e, processo para preparar um composto

Country Status (34)

Country Link
US (2) US6995167B2 (fr)
EP (1) EP1147114B1 (fr)
JP (1) JP2002534525A (fr)
KR (1) KR100660496B1 (fr)
CN (1) CN1132837C (fr)
AR (1) AR022283A1 (fr)
AT (1) ATE240960T1 (fr)
AU (1) AU775433B2 (fr)
BR (1) BR9916906A (fr)
CA (1) CA2359990A1 (fr)
CZ (1) CZ20012554A3 (fr)
DE (1) DE69908185T2 (fr)
DK (1) DK1147114T3 (fr)
EE (1) EE04528B1 (fr)
ES (1) ES2200590T3 (fr)
HK (1) HK1040517B (fr)
HU (1) HUP0200513A3 (fr)
ID (1) ID30034A (fr)
IL (1) IL144266A0 (fr)
IS (1) IS6000A (fr)
MY (1) MY118109A (fr)
NO (1) NO20013478L (fr)
NZ (1) NZ512733A (fr)
PT (1) PT1147114E (fr)
RU (1) RU2233282C2 (fr)
SA (1) SA00200987B1 (fr)
SE (1) SE9900100D0 (fr)
SI (1) SI1147114T1 (fr)
SK (1) SK9932001A3 (fr)
TR (1) TR200102042T2 (fr)
TW (2) TW200413387A (fr)
UA (1) UA71598C2 (fr)
WO (1) WO2000042044A1 (fr)
ZA (1) ZA200105527B (fr)

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US6569865B2 (en) 2001-06-01 2003-05-27 Astrazeneca Ab Spiro 1-azabicyclo[2.2.2]octane-3,2′(3′h)-furo[2,3-b]pyridine
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CN1325500C (zh) * 2002-04-18 2007-07-11 阿斯特拉曾尼卡有限公司 呋喃基化合物
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SE0202598D0 (sv) * 2002-09-02 2002-09-02 Astrazeneca Ab Alpha-7 Nicotinic receptor agonists and statins in combination
GB0220581D0 (en) 2002-09-04 2002-10-09 Novartis Ag Organic Compound
EE05516B1 (et) 2002-09-25 2012-02-15 Memory@Pharmaceuticals@Corporation Indasoolid bensotiasoolid ja bensoisotiasoolid nende valmistamine ning kasutamine
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WO2004052365A2 (fr) * 2002-12-06 2004-06-24 North Shore-Long Island Jewish Research Institute Inhibition d'inflammation au moyen d'agonistes cholinergiques se liant au recepteur alpha 7
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AR049401A1 (es) 2004-06-18 2006-07-26 Novartis Ag Aza-biciclononanos
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GB0521508D0 (en) 2005-10-21 2005-11-30 Novartis Ag Organic compounds
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GB0525672D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
GB0525673D0 (en) 2005-12-16 2006-01-25 Novartis Ag Organic compounds
RU2448111C2 (ru) * 2006-08-21 2012-04-20 Дженентек, Инк. Соединения азабензофуранила и способ их применения
TW200901974A (en) 2007-01-16 2009-01-16 Wyeth Corp Compounds, compositions, and methods of making and using them
SA08290475B1 (ar) * 2007-08-02 2013-06-22 Targacept Inc (2s، 3r)-n-(2-((3-بيردينيل)ميثيل)-1-آزا بيسيكلو[2، 2، 2]أوكت-3-يل)بنزو فيوران-2-كربوكساميد، وصور أملاحه الجديدة وطرق استخدامه
CA2728675A1 (fr) 2008-06-20 2009-12-23 Astrazeneca Ab Derives de dibenzothiazepine et leur utilisation
CN105218565A (zh) 2008-10-17 2016-01-06 泽农医药公司 螺羟吲哚化合物及其作为治疗剂的用途
PE20110711A1 (es) 2008-11-19 2011-10-11 Envivo Pharmaceuticals Inc Tratamiento de trastornos cognitivos con (r)-7-cloro-n-(quinuclidin-3-il)benzo[b]tiofeno-2-carboxamida y sales farmaceuticamente aceptables de la misma
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GB201314286D0 (en) 2013-08-08 2013-09-25 Takeda Pharmaceutical Therapeutic Compounds
GB201318222D0 (en) 2013-10-15 2013-11-27 Takeda Pharmaceutical Novel compounds
GB201320905D0 (en) 2013-11-27 2014-01-08 Takeda Pharmaceutical Therapeutic compounds
TW201613864A (en) 2014-02-20 2016-04-16 Takeda Pharmaceutical Novel compounds
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Also Published As

Publication number Publication date
DK1147114T3 (da) 2003-09-15
CA2359990A1 (fr) 2000-07-20
SI1147114T1 (en) 2003-12-31
NO20013478L (no) 2001-09-14
US20030149065A1 (en) 2003-08-07
HUP0200513A2 (en) 2002-06-29
EP1147114A1 (fr) 2001-10-24
UA71598C2 (en) 2004-12-15
AR022283A1 (es) 2002-09-04
US6995167B2 (en) 2006-02-07
KR20010086167A (ko) 2001-09-08
PT1147114E (pt) 2003-10-31
CN1132837C (zh) 2003-12-31
TW200413387A (en) 2004-08-01
KR100660496B1 (ko) 2006-12-22
CN1337964A (zh) 2002-02-27
US7196096B2 (en) 2007-03-27
SA00200987B1 (ar) 2006-11-07
JP2002534525A (ja) 2002-10-15
IL144266A0 (en) 2002-05-23
SK9932001A3 (en) 2002-04-04
AU2334300A (en) 2000-08-01
EP1147114B1 (fr) 2003-05-21
NZ512733A (en) 2003-08-29
TWI227237B (en) 2005-02-01
DE69908185T2 (de) 2004-06-03
HK1040517B (en) 2003-09-05
MY118109A (en) 2004-08-30
DE69908185D1 (de) 2003-06-26
CZ20012554A3 (cs) 2002-01-16
IS6000A (is) 2001-07-12
NO20013478D0 (no) 2001-07-13
ZA200105527B (en) 2002-10-04
EE200100370A (et) 2002-10-15
HUP0200513A3 (en) 2004-07-28
SE9900100D0 (sv) 1999-01-15
TR200102042T2 (tr) 2002-05-21
RU2233282C2 (ru) 2004-07-27
WO2000042044A1 (fr) 2000-07-20
EE04528B1 (et) 2005-08-15
US20050250802A1 (en) 2005-11-10
ES2200590T3 (es) 2004-03-01
ATE240960T1 (de) 2003-06-15
HK1040517A1 (en) 2002-06-14
ID30034A (id) 2001-11-01
AU775433B2 (en) 2004-07-29

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