BR9814765A - Feniluracilas substituìdas - Google Patents
Feniluracilas substituìdasInfo
- Publication number
- BR9814765A BR9814765A BR9814765-0A BR9814765A BR9814765A BR 9814765 A BR9814765 A BR 9814765A BR 9814765 A BR9814765 A BR 9814765A BR 9814765 A BR9814765 A BR 9814765A
- Authority
- BR
- Brazil
- Prior art keywords
- substituted
- alkyl
- amino
- possibly substituted
- pyridine
- Prior art date
Links
- -1 carboxy, cyano, carbamoyl Chemical group 0.000 abstract 7
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical compound C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 abstract 6
- 125000000217 alkyl group Chemical group 0.000 abstract 5
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 239000001257 hydrogen Substances 0.000 abstract 4
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- UMJSCPRVCHMLSP-UHFFFAOYSA-N pyridine Natural products COC1=CC=CN=C1 UMJSCPRVCHMLSP-UHFFFAOYSA-N 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000003282 alkyl amino group Chemical group 0.000 abstract 2
- 125000004414 alkyl thio group Chemical group 0.000 abstract 2
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 2
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 2
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000004183 alkoxy alkyl group Chemical group 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004466 alkoxycarbonylamino group Chemical group 0.000 abstract 1
- 125000004949 alkyl amino carbonyl amino group Chemical group 0.000 abstract 1
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 abstract 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 1
- 125000004644 alkyl sulfinyl group Chemical group 0.000 abstract 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
- 125000004656 alkyl sulfonylamino group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 125000003785 benzimidazolyl group Chemical group N1=C(NC2=C1C=CC=C2)* 0.000 abstract 1
- 125000004618 benzofuryl group Chemical group O1C(=CC2=C1C=CC=C2)* 0.000 abstract 1
- 125000004541 benzoxazolyl group Chemical group O1C(=NC2=C1C=CC=C2)* 0.000 abstract 1
- 125000001316 cycloalkyl alkyl group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000004663 dialkyl amino group Chemical group 0.000 abstract 1
- 125000004598 dihydrobenzofuryl group Chemical group O1C(CC2=C1C=CC=C2)* 0.000 abstract 1
- 125000000532 dioxanyl group Chemical group 0.000 abstract 1
- 125000005879 dioxolanyl group Chemical group 0.000 abstract 1
- LBKPGNUOUPTQKA-UHFFFAOYSA-N ethyl n-phenylcarbamate Chemical class CCOC(=O)NC1=CC=CC=C1 LBKPGNUOUPTQKA-UHFFFAOYSA-N 0.000 abstract 1
- 125000002541 furyl group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical group 0.000 abstract 1
- 239000004009 herbicide Substances 0.000 abstract 1
- 125000002883 imidazolyl group Chemical group 0.000 abstract 1
- 239000013067 intermediate product Substances 0.000 abstract 1
- 125000000842 isoxazolyl group Chemical group 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000002971 oxazolyl group Chemical group 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- PWXJULSLLONQHY-UHFFFAOYSA-N phenylcarbamic acid Chemical class OC(=O)NC1=CC=CC=C1 PWXJULSLLONQHY-UHFFFAOYSA-N 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 125000000168 pyrrolyl group Chemical group 0.000 abstract 1
- 125000002294 quinazolinyl group Chemical group N1=C(N=CC2=CC=CC=C12)* 0.000 abstract 1
- 125000001567 quinoxalinyl group Chemical group N1=C(C=NC2=CC=CC=C12)* 0.000 abstract 1
- 125000003107 substituted aryl group Chemical group 0.000 abstract 1
- 125000000020 sulfo group Chemical group O=S(=O)([*])O[H] 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 125000003718 tetrahydrofuranyl group Chemical group 0.000 abstract 1
- 125000001425 triazolyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Patente de Invenção: <B>"FENILURACILAS SUBSTITUìDAS"<D>. A invenção refere-se a novas feniluracilas substituídas da fórmula geral (I), na qual n representa os números 0, 1, 2 ou 3, Q representa O, S, SO, SO~ 2~, NH ou N (alquila), R¹ representa hidrogênio, amino ou alquila eventualmente substituída, R² representa carbóxi, ciano, carbamoíla, tiocarbamoíla ou alquila ou alcóxialquila eventualmente substituída, R³ representa hidrogênio, halogênio ou alquila eventualmente substituída, R^ 4^ representa nitro, amino ou um dos grupamentos abaixo -NH-CO-R^ 7^ ou -N(CO-R^ 7^)~ 2~, R^ 5^ representa nitro, amino, hidróxi, mercapto, carbóxi, ciano, carbamoíla, tiocarbamoíla, sulfo, clorossulfonila, aminossulfonila hidrogênio ou alquila, alcóxi, alquiltio, alquilsulfinila, alquilsulfonila, alquilamino, alquilcarbonila, alcoxicarbonila, alquilaminocarbonila, alquilaminocarbonilamino, alcoxicarbonilamino, alquilsulfonilamino ou bis-alquilsulfonil-amino eventualmente substituídos, R^ 6^ representa arila eventualmente substituída ou heterociclila eventualmente substituída das séries furila, tetrahidrofurila, benzofurila, dihidrobenzofurila, dioxolanila, dioxanila, benzodioxanila, pirrolila, imidazolila, benzimidazolila, triazolila, oxazolila, isoxazolila, benzoxazolila, tiazolila, isotiazolila, benzotiazolilpiridinila, quinolinila, isoquinolinila, pirimidinila, pirazolila, pirazinila, piridazinila, quinazolinila, quinoxalinila e R^ 7^ representa hidrogênio ou alquila, alcóxi, alquiltio, alquilamino, dialquilamino, alquenila, alquinila, cicloalquila, cicloalquilalquila, arila, arilalquila, heterociclila ou heteroxiciclilalquila eventualmente substituída. A invenção refere-se também ao emprego das feniluracilas da invenção como herbicidas, a um método para produzí-las e a feniluretanas substituídas (fenilcarbamatos) da fórmula geral (III), na qual A² representa alquila, arila ou arilalquila como produtos intermediários.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19752748A DE19752748A1 (de) | 1997-11-28 | 1997-11-28 | Substituierte Phenyluracile |
| PCT/EP1998/007342 WO1999028302A1 (de) | 1997-11-28 | 1998-11-17 | Substituierte phenyluracile |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9814765A true BR9814765A (pt) | 2000-10-03 |
Family
ID=7850080
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9814765-0A BR9814765A (pt) | 1997-11-28 | 1998-11-17 | Feniluracilas substituìdas |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US6432879B1 (pt) |
| EP (1) | EP1066267B1 (pt) |
| JP (1) | JP2001524543A (pt) |
| CN (1) | CN1284068A (pt) |
| AR (1) | AR016705A1 (pt) |
| AT (1) | ATE266645T1 (pt) |
| AU (1) | AU740818B2 (pt) |
| BR (1) | BR9814765A (pt) |
| CA (1) | CA2311557A1 (pt) |
| DE (2) | DE19752748A1 (pt) |
| WO (1) | WO1999028302A1 (pt) |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2842186A1 (de) | 1978-09-28 | 1980-04-10 | Basf Ag | Azofarbstoffe |
| JPH0539272A (ja) | 1991-01-09 | 1993-02-19 | Nissan Chem Ind Ltd | ピリミジンジオン誘導体および除草剤 |
| DE4200259A1 (de) * | 1992-01-08 | 1993-07-15 | Asta Medica Ag | Neue 1,2,4-triaminobenzol-derivate und verfahren zu deren herstellung |
| JPH05202031A (ja) | 1992-01-28 | 1993-08-10 | Nissan Chem Ind Ltd | Ｎ−アミノピリミジンジオン誘導体および除草剤 |
| US5262390A (en) | 1992-08-26 | 1993-11-16 | Fmc Corporation | Herbicical 2-[(4-heterocyclic-phenoxymethyl)phenoxy]-alkanoates |
| US5399543A (en) | 1993-04-21 | 1995-03-21 | Fmc Corporation | 3-[4-(phenylmethoxy)phenyl]-1-substituted-6-haloalkyl-uracil herbicides |
| WO1995017096A1 (en) | 1993-12-22 | 1995-06-29 | Fmc Corporation | Herbicidal haloalkyluracils |
| ES2176617T3 (es) | 1996-03-11 | 2002-12-01 | Sankyo Co | Derivados de anilina con actividad herbicida, su preparacion y su uso. |
| DE19708928A1 (de) | 1997-03-05 | 1998-09-10 | Bayer Ag | Substituierte aromatische Aminoverbindungen |
| DE19715017A1 (de) | 1997-04-11 | 1998-10-15 | Bayer Ag | Substituierte Aryluracile |
| DE19728125A1 (de) | 1997-07-02 | 1999-01-07 | Bayer Ag | Substituierte Aryluracile |
-
1997
- 1997-11-28 DE DE19752748A patent/DE19752748A1/de not_active Withdrawn
-
1998
- 1998-11-17 BR BR9814765-0A patent/BR9814765A/pt not_active IP Right Cessation
- 1998-11-17 DE DE59811399T patent/DE59811399D1/de not_active Expired - Fee Related
- 1998-11-17 JP JP2000523196A patent/JP2001524543A/ja active Pending
- 1998-11-17 US US09/554,965 patent/US6432879B1/en not_active Expired - Fee Related
- 1998-11-17 AT AT98956921T patent/ATE266645T1/de not_active IP Right Cessation
- 1998-11-17 CA CA002311557A patent/CA2311557A1/en not_active Abandoned
- 1998-11-17 AU AU13387/99A patent/AU740818B2/en not_active Ceased
- 1998-11-17 WO PCT/EP1998/007342 patent/WO1999028302A1/de not_active Ceased
- 1998-11-17 EP EP98956921A patent/EP1066267B1/de not_active Expired - Lifetime
- 1998-11-17 CN CN98813386A patent/CN1284068A/zh active Pending
- 1998-11-27 AR ARP980106036A patent/AR016705A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| DE19752748A1 (de) | 1999-06-02 |
| WO1999028302A1 (de) | 1999-06-10 |
| DE59811399D1 (de) | 2004-06-17 |
| CN1284068A (zh) | 2001-02-14 |
| AR016705A1 (es) | 2001-07-25 |
| EP1066267B1 (de) | 2004-05-12 |
| JP2001524543A (ja) | 2001-12-04 |
| AU740818B2 (en) | 2001-11-15 |
| ATE266645T1 (de) | 2004-05-15 |
| AU1338799A (en) | 1999-06-16 |
| EP1066267A1 (de) | 2001-01-10 |
| US6432879B1 (en) | 2002-08-13 |
| CA2311557A1 (en) | 1999-06-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7O E 8O ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1910 DE 14/08/2007. |