DK1123291T3 - Fremgangsmåde til fremstilling af 3-(substitueret phenyl)-5-thienyl (eller furyl)-1,2,4-triazoler og hidtil ukendte mellemprodukter anvendt derved - Google Patents
Fremgangsmåde til fremstilling af 3-(substitueret phenyl)-5-thienyl (eller furyl)-1,2,4-triazoler og hidtil ukendte mellemprodukter anvendt dervedInfo
- Publication number
- DK1123291T3 DK1123291T3 DK99970990T DK99970990T DK1123291T3 DK 1123291 T3 DK1123291 T3 DK 1123291T3 DK 99970990 T DK99970990 T DK 99970990T DK 99970990 T DK99970990 T DK 99970990T DK 1123291 T3 DK1123291 T3 DK 1123291T3
- Authority
- DK
- Denmark
- Prior art keywords
- triazoles
- furyl
- thienyl
- substituted phenyl
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C327/00—Thiocarboxylic acids
- C07C327/58—Derivatives of thiocarboxylic acids, the doubly-bound oxygen atoms being replaced by nitrogen atoms, e.g. imino-thio ethers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10531498P | 1998-10-23 | 1998-10-23 | |
| PCT/US1999/024860 WO2000024738A1 (en) | 1998-10-23 | 1999-10-22 | Process for preparing 3-(substituted phenyl)-5-thienyl or furyl)-1,2,4-triazoles and novel intermediates utilized therein |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1123291T3 true DK1123291T3 (da) | 2007-11-05 |
Family
ID=22305135
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK99970990T DK1123291T3 (da) | 1998-10-23 | 1999-10-22 | Fremgangsmåde til fremstilling af 3-(substitueret phenyl)-5-thienyl (eller furyl)-1,2,4-triazoler og hidtil ukendte mellemprodukter anvendt derved |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US6329528B1 (da) |
| EP (1) | EP1123291B1 (da) |
| JP (1) | JP4610740B2 (da) |
| KR (1) | KR100795030B1 (da) |
| CN (1) | CN1136218C (da) |
| AT (1) | ATE367388T1 (da) |
| AU (1) | AU769981B2 (da) |
| BR (1) | BR9914673B1 (da) |
| DE (1) | DE69936592T2 (da) |
| DK (1) | DK1123291T3 (da) |
| HU (1) | HU228839B1 (da) |
| IL (1) | IL142599A (da) |
| WO (1) | WO2000024738A1 (da) |
| ZA (1) | ZA200102719B (da) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0302094D0 (en) | 2003-01-29 | 2003-02-26 | Pharmagene Lab Ltd | EP4 receptor antagonists |
| GB0324269D0 (en) | 2003-10-16 | 2003-11-19 | Pharmagene Lab Ltd | EP4 receptor antagonists |
| EP2474546A1 (en) | 2006-01-23 | 2012-07-11 | Vertex Pharmaceuticals Inc. | Thiophene-carboxamides useful as inhibitors of protein kinases |
| JP2009533452A (ja) | 2006-04-13 | 2009-09-17 | バーテックス ファーマシューティカルズ インコーポレイテッド | タンパク質キナーゼの阻害剤として有用なチオフェン−カルボキサミド |
| CN101495474A (zh) | 2006-05-23 | 2009-07-29 | 沃泰克斯药物股份有限公司 | 可用作蛋白激酶抑制剂的噻吩-甲酰胺类 |
| JP2009538309A (ja) | 2006-05-23 | 2009-11-05 | バーテックス ファーマシューティカルズ インコーポレイテッド | プロテインキナーゼのインヒビターとして有用なチオフェンカルボキサミド |
| US9073881B2 (en) | 2011-09-23 | 2015-07-07 | Hoffmann-La Roche Inc. | Benzoic acid derivatives |
| CN104016962A (zh) * | 2014-06-16 | 2014-09-03 | 商丘凯瑞达化工有限公司 | 2-噻吩乙酰氯合成工艺 |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1039459A (en) * | 1965-04-01 | 1966-08-17 | Shell Int Research | Novel derivatives of 2,6-dichlorothiobenzamide, methods for their preparation, and herbicidal compositions containing them |
| SU508198A3 (ru) * | 1971-07-22 | 1976-03-25 | Группо Лепетит С.П.А. (Фирма) | Способ получени производных 1,2,4-триазола |
| AR241530A1 (es) | 1984-12-21 | 1992-08-31 | Ciba Geigy A G Cesionaria De F | 1,2,4-triazoles, composicion para el control de pestes y procedimiento para la preparacion de 1,2,4-triazoles. |
| ZA859576B (en) * | 1984-12-21 | 1986-08-27 | Hoffmann La Roche | Heterocyclic compounds |
| JPS6284046A (ja) * | 1985-09-09 | 1987-04-17 | シンテツクス（ユ−・エス・エイ）インコ−ポレイテツド | ナフタレン系抗乾癬剤 |
| JP2729810B2 (ja) * | 1988-09-27 | 1998-03-18 | クミアイ化学工業株式会社 | フェニルトリアゾール誘導体及び殺虫剤 |
| JP3217846B2 (ja) * | 1992-03-04 | 2001-10-15 | クミアイ化学工業株式会社 | トリアゾール誘導体及び殺虫剤 |
| JPH05310712A (ja) | 1992-04-03 | 1993-11-22 | Kumiai Chem Ind Co Ltd | ジフェニルトリアゾール誘導体及び殺虫、殺ダニ剤 |
| JP3443134B2 (ja) * | 1992-05-29 | 2003-09-02 | クミアイ化学工業株式会社 | トリアゾール誘導体及び殺虫、殺ダニ剤 |
| TW226993B (da) | 1992-05-29 | 1994-07-21 | Kumiai Chemical Industry Co | |
| JPH0641093A (ja) * | 1992-07-24 | 1994-02-15 | Kumiai Chem Ind Co Ltd | シクロアルキルトリアゾール誘導体および害虫防除剤 |
| EP0609459B1 (en) | 1992-07-24 | 1996-10-09 | Kumiai Chemical Industry Co., Ltd. | Triazole derivative, process for producing the same, pest control agent, and pest control method |
| JP3161827B2 (ja) * | 1992-07-31 | 2001-04-25 | クミアイ化学工業株式会社 | アルケニルトリアゾール誘導体及び害虫防除剤 |
| JPH0641094A (ja) * | 1992-07-24 | 1994-02-15 | Kumiai Chem Ind Co Ltd | シクロアルケニルトリアゾール誘導体および有害生物防除剤 |
| JP3682075B2 (ja) * | 1993-04-16 | 2005-08-10 | クミアイ化学工業株式会社 | トリアゾール誘導体及び殺虫、殺ダニ剤 |
| JPH0776577A (ja) * | 1993-07-14 | 1995-03-20 | Kumiai Chem Ind Co Ltd | ジフェニルトリアゾール誘導体及び殺虫、殺ダニ剤 |
| JP3496078B2 (ja) * | 1993-07-20 | 2004-02-09 | イハラケミカル工業株式会社 | 新規なヒドラゾン誘導体及びその製造法 |
| AU2630495A (en) * | 1994-06-09 | 1996-01-04 | Nippon Soda Co., Ltd. | Triazole compound, production process, and pest control agent |
| JPH07330742A (ja) * | 1994-06-09 | 1995-12-19 | Nippon Soda Co Ltd | トリアゾール誘導体、製法及び有害生物防除剤 |
| JP3407088B2 (ja) * | 1994-06-27 | 2003-05-19 | イハラケミカル工業株式会社 | トリアゾール誘導体の製造方法およびその中間体 |
| KR100199123B1 (ko) * | 1994-07-01 | 1999-06-15 | 쓰끼하시 다미까따 | 트리아졸 화합물, 그의 제법 및 유해 생물 방제제 |
| JPH0892224A (ja) * | 1994-09-16 | 1996-04-09 | Kumiai Chem Ind Co Ltd | ３，５−置換フェニルトリアゾール誘導体および殺虫、殺ダニ剤 |
| JPH08245315A (ja) * | 1995-03-16 | 1996-09-24 | Nippon Soda Co Ltd | トリアゾール誘導体および有害生物防除剤 |
| JPH08283261A (ja) * | 1995-04-07 | 1996-10-29 | Kumiai Chem Ind Co Ltd | ３−フェニルトリアゾール誘導体および殺虫、殺ダニ剤 |
| EP0922043B1 (en) * | 1997-04-24 | 2002-01-30 | Dow AgroSciences LLC | Pesticidal 3-(substituted phenyl)-5-(thienyl or furyl)-1,2,4-triazoles |
-
1999
- 1999-10-22 AT AT99970990T patent/ATE367388T1/de active
- 1999-10-22 DK DK99970990T patent/DK1123291T3/da active
- 1999-10-22 WO PCT/US1999/024860 patent/WO2000024738A1/en not_active Ceased
- 1999-10-22 BR BRPI9914673-8A patent/BR9914673B1/pt not_active IP Right Cessation
- 1999-10-22 DE DE69936592T patent/DE69936592T2/de not_active Expired - Lifetime
- 1999-10-22 AU AU12253/00A patent/AU769981B2/en not_active Ceased
- 1999-10-22 EP EP99970990A patent/EP1123291B1/en not_active Expired - Lifetime
- 1999-10-22 CN CNB998124990A patent/CN1136218C/zh not_active Expired - Fee Related
- 1999-10-22 JP JP2000578308A patent/JP4610740B2/ja not_active Expired - Fee Related
- 1999-10-22 US US09/426,076 patent/US6329528B1/en not_active Expired - Fee Related
- 1999-10-22 KR KR1020017005099A patent/KR100795030B1/ko not_active Expired - Fee Related
- 1999-10-22 HU HU0104115A patent/HU228839B1/hu not_active IP Right Cessation
-
2001
- 2001-04-03 ZA ZA2001/02719A patent/ZA200102719B/en unknown
- 2001-04-15 IL IL142599A patent/IL142599A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DE69936592D1 (de) | 2007-08-30 |
| IL142599A (en) | 2006-08-20 |
| ZA200102719B (en) | 2002-06-26 |
| HUP0104115A2 (hu) | 2002-02-28 |
| HUP0104115A3 (en) | 2002-12-28 |
| ATE367388T1 (de) | 2007-08-15 |
| EP1123291B1 (en) | 2007-07-18 |
| BR9914673A (pt) | 2001-07-17 |
| KR20010087378A (ko) | 2001-09-15 |
| WO2000024738A1 (en) | 2000-05-04 |
| HU228839B1 (hu) | 2013-06-28 |
| CN1324356A (zh) | 2001-11-28 |
| JP4610740B2 (ja) | 2011-01-12 |
| BR9914673B1 (pt) | 2010-12-14 |
| JP2002528450A (ja) | 2002-09-03 |
| AU769981B2 (en) | 2004-02-12 |
| US6329528B1 (en) | 2001-12-11 |
| AU1225300A (en) | 2000-05-15 |
| EP1123291A1 (en) | 2001-08-16 |
| DE69936592T2 (de) | 2008-04-30 |
| CN1136218C (zh) | 2004-01-28 |
| KR100795030B1 (ko) | 2008-01-16 |
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