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BR9806801A - Utilização de um antagonista de receptores cb1, composição farmacêutica, e, estojo para o tratamento de distúrbios da apetência - Google Patents

Utilização de um antagonista de receptores cb1, composição farmacêutica, e, estojo para o tratamento de distúrbios da apetência

Info

Publication number
BR9806801A
BR9806801A BR9806801-6A BR9806801A BR9806801A BR 9806801 A BR9806801 A BR 9806801A BR 9806801 A BR9806801 A BR 9806801A BR 9806801 A BR9806801 A BR 9806801A
Authority
BR
Brazil
Prior art keywords
treatment
pharmaceutical composition
receptor antagonist
kit
disorders
Prior art date
Application number
BR9806801-6A
Other languages
English (en)
Inventor
Jeanne Maruani
Philippe Soubrie
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of BR9806801A publication Critical patent/BR9806801A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Addiction (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)

Abstract

"UTILIZAçãO DE UM ANTAGONISTA DE RECEPTORES CB1, COMPOSIçãO FARMACêUTICA, E, ESTOJO PARA O TRATAMENTO DE DISTúRBIOS DA APETêNCIA". A invenção refere-se à utilização de um antagonista de receptores de canabinóides centrais, sozinhos ou em associação com um composto regulador dos distúrbios metabólicos, notadamente um agonista de receptor <225>~ 3~ adrenérgico, para a preparação de medicamentos úteis no tratamento de distúrbios da apetência.
BR9806801-6A 1997-01-28 1998-01-28 Utilização de um antagonista de receptores cb1, composição farmacêutica, e, estojo para o tratamento de distúrbios da apetência BR9806801A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9700870A FR2758723B1 (fr) 1997-01-28 1997-01-28 Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour la preparation de medicaments
PCT/FR1998/000154 WO1998032441A1 (fr) 1997-01-28 1998-01-28 Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour reguler l'appetance

Publications (1)

Publication Number Publication Date
BR9806801A true BR9806801A (pt) 2000-05-16

Family

ID=9503028

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9806801-6A BR9806801A (pt) 1997-01-28 1998-01-28 Utilização de um antagonista de receptores cb1, composição farmacêutica, e, estojo para o tratamento de distúrbios da apetência

Country Status (31)

Country Link
US (3) US6344474B1 (pt)
EP (2) EP0969835B1 (pt)
JP (1) JP3676383B2 (pt)
AR (1) AR011776A1 (pt)
AT (1) ATE358480T1 (pt)
AU (1) AU6219398A (pt)
BR (1) BR9806801A (pt)
CA (1) CA2278661A1 (pt)
DE (1) DE69837473T2 (pt)
DK (1) DK0969835T3 (pt)
DZ (1) DZ2405A1 (pt)
EE (1) EE04630B1 (pt)
ES (1) ES2285760T3 (pt)
FR (1) FR2758723B1 (pt)
GT (1) GT199800021A (pt)
HR (1) HRP980042A2 (pt)
ID (1) ID22216A (pt)
IS (1) IS5113A (pt)
LV (1) LV12354B (pt)
ME (1) MEP26508A (pt)
MY (1) MY117251A (pt)
NO (1) NO323696B1 (pt)
PT (1) PT969835E (pt)
RS (1) RS49830B (pt)
SA (1) SA98181113B1 (pt)
SK (1) SK99799A3 (pt)
TR (1) TR199901721T2 (pt)
TW (1) TW450808B (pt)
UY (1) UY24847A1 (pt)
WO (1) WO1998032441A1 (pt)
ZA (1) ZA98691B (pt)

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IS5113A (is) 1999-07-12
NO993634D0 (no) 1999-07-27
MEP26508A (en) 2010-06-10
SK99799A3 (en) 2000-06-12
AU6219398A (en) 1998-08-18
DE69837473T2 (de) 2007-12-13
ATE358480T1 (de) 2007-04-15
NO323696B1 (no) 2007-06-25
EP1795194A3 (fr) 2008-04-30
FR2758723B1 (fr) 1999-04-23
AR011776A1 (es) 2000-09-13
LV12354B (en) 2000-02-20
TW450808B (en) 2001-08-21
EP0969835A1 (fr) 2000-01-12
US6344474B1 (en) 2002-02-05
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NO993634L (no) 1999-09-27
WO1998032441A1 (fr) 1998-07-30
MY117251A (en) 2004-06-30
TR199901721T2 (xx) 1999-10-21
LV12354A (lv) 1999-10-20
DE69837473D1 (de) 2007-05-16
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US20050026986A1 (en) 2005-02-03
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US20020128302A1 (en) 2002-09-12
FR2758723A1 (fr) 1998-07-31
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EP1795194A2 (fr) 2007-06-13
CA2278661A1 (en) 1998-07-30
SA98181113B1 (ar) 2006-06-25
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