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BR0307468A - Derivados tiadiazinona antimicrobianos úteis no tratamento de infecções bacterianas - Google Patents

Derivados tiadiazinona antimicrobianos úteis no tratamento de infecções bacterianas

Info

Publication number
BR0307468A
BR0307468A BR0307468-4A BR0307468A BR0307468A BR 0307468 A BR0307468 A BR 0307468A BR 0307468 A BR0307468 A BR 0307468A BR 0307468 A BR0307468 A BR 0307468A
Authority
BR
Brazil
Prior art keywords
treatment
bacterial infections
antimicrobial
thiadiazinone
derivatives useful
Prior art date
Application number
BR0307468-4A
Other languages
English (en)
Inventor
Gary W Luehr
Mikhail F Gordeev
Dinesh V Patel
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BR0307468A publication Critical patent/BR0307468A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"DERIVADOS TIADIAZINONA ANTIMICROBIANOS úTEIS NO TRATAMENTO DE INFECçõES BACTERIANAS". A presente invenção provê certos derivados tiadiazinona de oxazolidinonas de fórmula (1) e seus sais farmaceuticamente aceitáveis que são agentes antibacterianos. São também descritas composições farmacêuticas contendo derivados tiadiazinona de oxazolidinonas, métodos para sua utilização, e métodos de preparação destes compostos.
BR0307468-4A 2002-02-05 2003-02-04 Derivados tiadiazinona antimicrobianos úteis no tratamento de infecções bacterianas BR0307468A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35459802P 2002-02-05 2002-02-05
PCT/US2003/001082 WO2003066631A1 (en) 2002-02-05 2003-02-04 Antimicrobial thiadiazinone derivatives useful in treatment of bacterial infections

Publications (1)

Publication Number Publication Date
BR0307468A true BR0307468A (pt) 2004-11-09

Family

ID=27734400

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0307468-4A BR0307468A (pt) 2002-02-05 2003-02-04 Derivados tiadiazinona antimicrobianos úteis no tratamento de infecções bacterianas

Country Status (8)

Country Link
US (1) US6828317B2 (pt)
EP (1) EP1472247A1 (pt)
JP (1) JP2005519931A (pt)
AU (1) AU2003209241A1 (pt)
BR (1) BR0307468A (pt)
CA (1) CA2475036A1 (pt)
MX (1) MXPA04007468A (pt)
WO (1) WO2003066631A1 (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7105547B2 (en) 2002-10-10 2006-09-12 Pharmacia And Upjohn Company Antimicrobial 1-aryl dihydropyridone compounds
TW200804358A (en) * 2006-03-31 2008-01-16 Res Found Itsuu Lab Novel compound having heterocycle

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1993009103A1 (en) * 1991-11-01 1993-05-13 The Upjohn Company Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents
SK283420B6 (sk) * 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
DK0673370T3 (da) 1992-12-08 1998-09-07 Upjohn Co Troponsubstituerede phenyloxazolidinoner som antibakterielle midler

Also Published As

Publication number Publication date
US6828317B2 (en) 2004-12-07
JP2005519931A (ja) 2005-07-07
EP1472247A1 (en) 2004-11-03
AU2003209241A1 (en) 2003-09-02
CA2475036A1 (en) 2003-08-14
US20040014746A1 (en) 2004-01-22
MXPA04007468A (es) 2004-11-10
WO2003066631A1 (en) 2003-08-14

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE 4A., 5A., 6A., E 7A. ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2051 DE 27/04/2010.