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BG61485B1 - N горе 4-оксикарбонил заместени 5'-деокси-5-флуороцитидини - Google Patents

N горе 4-оксикарбонил заместени 5'-деокси-5-флуороцитидини Download PDF

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Publication number
BG61485B1
BG61485B1 BG98304A BG9830493A BG61485B1 BG 61485 B1 BG61485 B1 BG 61485B1 BG 98304 A BG98304 A BG 98304A BG 9830493 A BG9830493 A BG 9830493A BG 61485 B1 BG61485 B1 BG 61485B1
Authority
BG
Bulgaria
Prior art keywords
deoxy
cytidine
fluorocytidine
fluoro
acetyl
Prior art date
Application number
BG98304A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG98304A (bg
Inventor
Motohiro Arasaki
Hideo Ishitsuka
Isami Kuruma
Masanori Miwa
Chikako Murasaki
Nobuo Shimma
Isao Umeda
Original Assignee
F. Hoffmann- La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8210304&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG61485(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by F. Hoffmann- La Roche Ag filed Critical F. Hoffmann- La Roche Ag
Publication of BG98304A publication Critical patent/BG98304A/bg
Publication of BG61485B1 publication Critical patent/BG61485B1/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BG98304A 1992-12-18 1993-12-16 N горе 4-оксикарбонил заместени 5'-деокси-5-флуороцитидини BG61485B1 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP92121538 1992-12-18

Publications (2)

Publication Number Publication Date
BG98304A BG98304A (bg) 1994-01-03
BG61485B1 true BG61485B1 (bg) 1997-09-30

Family

ID=8210304

Family Applications (1)

Application Number Title Priority Date Filing Date
BG98304A BG61485B1 (bg) 1992-12-18 1993-12-16 N горе 4-оксикарбонил заместени 5'-деокси-5-флуороцитидини

Country Status (40)

Country Link
US (1) US5472949A (lt)
EP (1) EP0602454B1 (lt)
JP (1) JP2501297B2 (lt)
KR (1) KR100347218B1 (lt)
CN (1) CN1035617C (lt)
AT (1) ATE137244T1 (lt)
AU (1) AU671491B2 (lt)
BG (1) BG61485B1 (lt)
BR (1) BR9305089A (lt)
CA (1) CA2103324C (lt)
CZ (1) CZ284788B6 (lt)
DE (1) DE69302360T2 (lt)
DK (1) DK0602454T3 (lt)
EE (1) EE03086B1 (lt)
ES (1) ES2086856T3 (lt)
FI (1) FI112365B (lt)
GE (1) GEP20074251B (lt)
GR (1) GR3020286T3 (lt)
HR (1) HRP931430B1 (lt)
HU (2) HU218291B (lt)
IL (1) IL108000A0 (lt)
IS (1) IS4108A (lt)
LT (1) LT3115B (lt)
LV (1) LV10625B (lt)
MY (1) MY109282A (lt)
NO (1) NO300066B1 (lt)
NZ (1) NZ250414A (lt)
PH (1) PH30168A (lt)
PL (1) PL174100B1 (lt)
RO (1) RO112619B1 (lt)
RU (2) RU2458932C2 (lt)
SA (1) SA93140409B1 (lt)
SI (1) SI9300648B (lt)
SK (1) SK281403B6 (lt)
SV (1) SV1993000080A (lt)
TW (1) TW372239B (lt)
UA (1) UA39158C2 (lt)
UY (1) UY23697A1 (lt)
YU (1) YU49411B (lt)
ZA (1) ZA939293B (lt)

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Also Published As

Publication number Publication date
IS4108A (is) 1994-06-19
LTIP1627A (en) 1994-07-15
DE69302360T2 (de) 1996-10-31
EP0602454A1 (en) 1994-06-22
TW372239B (en) 1999-10-21
NO300066B1 (no) 1997-04-01
HRP931430A2 (en) 1998-06-30
UA39158C2 (uk) 2001-06-15
FI935616L (fi) 1994-06-19
RU2458932C2 (ru) 2012-08-20
SI9300648A (en) 1994-09-30
EE03086B1 (et) 1998-04-15
ATE137244T1 (de) 1996-05-15
LT3115B (en) 1994-12-27
RU2493162C1 (ru) 2013-09-20
NO934671L (no) 1994-06-20
CN1035617C (zh) 1997-08-13
AU5069093A (en) 1994-06-30
HUT65757A (en) 1994-07-28
RO112619B1 (ro) 1997-11-28
US5472949A (en) 1995-12-05
BG98304A (bg) 1994-01-03
EP0602454B1 (en) 1996-04-24
YU49411B (sh) 2006-01-16
MY109282A (en) 1996-12-31
CN1094056A (zh) 1994-10-26
CZ284788B6 (cs) 1999-03-17
GR3020286T3 (en) 1996-09-30
ES2086856T3 (es) 1996-07-01
CZ273193A3 (en) 1994-07-13
ZA939293B (en) 1994-06-18
JPH06211891A (ja) 1994-08-02
DK0602454T3 (da) 1996-07-29
JP2501297B2 (ja) 1996-05-29
SI9300648B (sl) 2000-06-30
PL301541A1 (en) 1994-06-27
HU211965A9 (en) 1996-01-29
DE69302360D1 (de) 1996-05-30
CA2103324A1 (en) 1994-06-19
FI112365B (fi) 2003-11-28
AU671491B2 (en) 1996-08-29
CA2103324C (en) 1997-12-23
HU9303525D0 (en) 1994-04-28
SK144493A3 (en) 1994-10-05
BR9305089A (pt) 1994-07-05
GEP20074251B (en) 2007-12-10
HU218291B (en) 2000-07-28
LV10625A (lv) 1995-04-20
HK1005875A1 (en) 1999-01-29
UY23697A1 (es) 1994-06-08
IL108000A0 (en) 1994-04-12
YU77993A (sh) 1996-10-18
SA93140409B1 (ar) 2004-07-24
SK281403B6 (sk) 2001-03-12
FI935616A0 (fi) 1993-12-14
PH30168A (en) 1997-01-21
RU2135511C1 (ru) 1999-08-27
NZ250414A (en) 1995-12-21
HRP931430B1 (en) 1999-08-31
SV1993000080A (es) 1996-01-26
NO934671D0 (no) 1993-12-17
PL174100B1 (pl) 1998-06-30
LV10625B (en) 1996-04-20
KR100347218B1 (ko) 2003-01-24
KR940014428A (ko) 1994-07-18

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