BG60590B1 - Method for the preparation of 9-substituted quanine derivatives - Google Patents

Method for the preparation of 9-substituted quanine derivatives Download PDF

Info

Publication number: BG60590B1
Authority: BG; Bulgaria
Prior art keywords: amino; imidazole; carboxamide; substituted; formula
Prior art date: 1989-03-20

Application number

BG95145A

Other languages

Bulgarian (bg)

English (en)

Other versions

BG95145A (bg

Inventor

Borge Alhede

Finn P Clausen

Jorgen Juhl-Christensen

Klaus K Mccluskey

Herbert Preikschat

Original Assignee

Gea Farmaceutisk Fabrik As

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-03-20

Filing date

1991-09-20

Publication date

1995-09-29

1991-09-20 Application filed by Gea Farmaceutisk Fabrik As filed Critical Gea Farmaceutisk Fabrik As

1993-12-24 Publication of BG95145A publication Critical patent/BG95145A/bg

1995-09-29 Publication of BG60590B1 publication Critical patent/BG60590B1/bg

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/052—Imidazole radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

BG95145A 1989-03-20 1991-09-20 Method for the preparation of 9-substituted quanine derivatives BG60590B1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DK135489A DK135489D0 (da)	1989-03-20	1989-03-20	Fremgangsmaade til fremstilling af 9-substituerede guaninderivater og mellemprodukter til brug ved fremgangsmaaden
PCT/DK1990/000077 WO1990011283A1 (en)	1989-03-20	1990-03-19	A process for the preparation of 9-substituted guanine derivatives and intermediates for use in the process

Publications (2)

Publication Number	Publication Date
BG95145A BG95145A (bg)	1993-12-24
BG60590B1 true BG60590B1 (en)	1995-09-29

Family

ID=8103930

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG95145A BG60590B1 (en)	1989-03-20	1991-09-20	Method for the preparation of 9-substituted quanine derivatives

Country Status (28)

Country	Link
US (1)	US5223619A (pt)
EP (1)	EP0464112B1 (pt)
KR (1)	KR0142098B1 (pt)
AR (1)	AR245719A1 (pt)
AT (1)	ATE112568T1 (pt)
BG (1)	BG60590B1 (pt)
BR (1)	BR9007230A (pt)
CA (1)	CA2047217A1 (pt)
CS (1)	CS275359B2 (pt)
DD (1)	DD293116A5 (pt)
DE (1)	DE69013146T2 (pt)
DK (2)	DK135489D0 (pt)
ES (1)	ES2061023T3 (pt)
FI (1)	FI97387C (pt)
GE (1)	GEP19971014B (pt)
GR (1)	GR1001096B (pt)
HR (1)	HRP920907B1 (pt)
HU (1)	HU206715B (pt)
IE (1)	IE62042B1 (pt)
LT (1)	LT3183B (pt)
LV (1)	LV10455B (pt)
NO (1)	NO178497C (pt)
PL (1)	PL163313B1 (pt)
RO (1)	RO109737B1 (pt)
RU (2)	RU2090566C1 (pt)
SI (1)	SI9010545A (pt)
WO (1)	WO1990011283A1 (pt)
YU (1)	YU47343B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IT1264599B1 (it) *	1993-06-14	1996-10-04	Solar Chem Sa	Processo per la sintesi della 9-(2-idrossietossimetil)- guanina
GB9520364D0 (en) *	1995-10-05	1995-12-06	Chiroscience Ltd	Compouundds
JP4525883B2 (ja) *	1998-07-23	2010-08-18	アステラス製薬株式会社	イミダゾール化合物
US6872243B2 (en)	2002-09-04	2005-03-29	Xerox Corporation	Phase change inks containing gelator additives
US6860928B2 (en)	2002-09-04	2005-03-01	Xerox Corporation	Alkylated urea and triaminotriazine compounds and phase change inks containing same
US6761758B2 (en)	2002-09-04	2004-07-13	Xerox Corporation	Alkylated tetrakis(triaminotriazine) compounds and phase change inks containing same
US6811595B2 (en)	2002-09-04	2004-11-02	Xerox Corporation	Guanidinopyrimidinone compounds and phase change inks containing same
US7144450B2 (en)	2004-12-04	2006-12-05	Xerox Corporation	Phase change inks containing trans-1,2-cyclohexane bis(urea-urethane) compounds
US7317122B2 (en)	2004-12-04	2008-01-08	Xerox Corporation	Curable trans-1,2-cyclohexane bis(urea-urethane) compounds
US7314949B2 (en)	2004-12-04	2008-01-01	Xerox Corporation	Trans-1,2-cyclohexane bis(urea-urethane) compounds
US7153349B2 (en)	2004-12-04	2006-12-26	Xerox Corporation	Phase change inks containing curable trans-1,2-cyclohexane bis(urea-urethane) compounds
US7220300B2 (en)	2004-12-04	2007-05-22	Xerox Corporation	Phase change inks containing bis(urea-urethane) compounds
US7560587B2 (en)	2004-12-04	2009-07-14	Xerox Corporation	Bis[urea-urethane] compounds
KR102277174B1 (ko)	2013-10-29	2021-07-14	스웹 인터네셔널 에이비이	스크린 프린티드 브레이징재를 이용한 판형 열교환기 브레이징 방법 및 그 방법으로 제조된 판형 열교환기
CN115504977B (zh) *	2022-09-23	2024-02-09	海南锦瑞制药有限公司	更昔洛韦的制备方法及注射用更昔洛韦的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS56152437U (pt) *	1980-04-14	1981-11-14
US4602089A (en) *	1982-03-12	1986-07-22	Newport Pharmaceuticals, Inc.	Process for preparing purine compounds
US4451478A (en) *	1982-03-12	1984-05-29	Newport Pharmaceuticals International, Inc.	Imidazole compounds
JPS6055071B2 (ja) *	1982-04-16	1985-12-03	四国化成工業株式会社	イミダゾリル琥珀酸化合物および該化合物を用いるエポキシ樹脂硬化方法
HUT36464A (en) *	1983-05-24	1985-09-30	Newport Pharmaceuticals	Process for producing erythro-4-amino-3-/2-hydroxy-3-alkyl/-imidazol-5-carboxamide
EP0219838A3 (en) *	1985-10-22	1988-04-06	Takeda Chemical Industries, Ltd.	Carbocyclic purine nucleosides, their production and use
MY101126A (en) *	1985-12-13	1991-07-31	Beecham Group Plc	Novel compounds

1989
- 1989-03-20 DK DK135489A patent/DK135489D0/da not_active Application Discontinuation
1990
- 1990-03-16 IE IE99490A patent/IE62042B1/en unknown
- 1990-03-19 RO RO148411A patent/RO109737B1/ro unknown
- 1990-03-19 EP EP90905442A patent/EP0464112B1/en not_active Expired - Lifetime
- 1990-03-19 HU HU902874A patent/HU206715B/hu not_active IP Right Cessation
- 1990-03-19 WO PCT/DK1990/000077 patent/WO1990011283A1/en not_active Ceased
- 1990-03-19 DE DE69013146T patent/DE69013146T2/de not_active Expired - Fee Related
- 1990-03-19 ES ES90905442T patent/ES2061023T3/es not_active Expired - Lifetime
- 1990-03-19 RU RU9093004872A patent/RU2090566C1/ru active
- 1990-03-19 CA CA002047217A patent/CA2047217A1/en not_active Abandoned
- 1990-03-19 AT AT90905442T patent/ATE112568T1/de not_active IP Right Cessation
- 1990-03-19 DK DK90905442.1T patent/DK0464112T3/da active
- 1990-03-19 KR KR1019910701187A patent/KR0142098B1/ko not_active Expired - Fee Related
- 1990-03-19 BR BR909007230A patent/BR9007230A/pt not_active Application Discontinuation
- 1990-03-19 US US07/761,890 patent/US5223619A/en not_active Expired - Fee Related
- 1990-03-20 YU YU54590A patent/YU47343B/sh unknown
- 1990-03-20 SI SI9010545A patent/SI9010545A/sl unknown
- 1990-03-20 DD DD90338906A patent/DD293116A5/de not_active IP Right Cessation
- 1990-03-20 GR GR900100212A patent/GR1001096B/el unknown
- 1990-03-20 CS CS901365A patent/CS275359B2/cs unknown
- 1990-03-20 AR AR90316421A patent/AR245719A1/es active
- 1990-03-20 PL PL90284379A patent/PL163313B1/pl unknown
1991
- 1991-09-19 FI FI914418A patent/FI97387C/fi active
- 1991-09-19 RU SU915001705A patent/RU2042668C1/ru active
- 1991-09-19 NO NO913686A patent/NO178497C/no unknown
- 1991-09-20 BG BG95145A patent/BG60590B1/bg unknown
1992
- 1992-10-02 HR HRP-545/90A patent/HRP920907B1/xx not_active IP Right Cessation
- 1992-12-02 LV LVP-92-250A patent/LV10455B/en unknown
1993
- 1993-01-27 LT LTIP297A patent/LT3183B/lt not_active IP Right Cessation
- 1993-08-25 GE GEAP19931494A patent/GEP19971014B/en unknown

Also Published As

Publication number	Publication date
FI97387B (fi)	1996-08-30
LV10455B (en)	1995-08-20
HU206715B (en)	1992-12-28
NO178497C (no)	1996-04-10
ATE112568T1 (de)	1994-10-15
CS9001365A3 (en)	1992-02-19
HUT59141A (en)	1992-04-28
LTIP297A (en)	1994-08-25
NO178497B (no)	1996-01-02
NO913686D0 (no)	1991-09-19
LT3183B (en)	1995-03-27
YU54590A (sh)	1992-12-21
EP0464112A1 (en)	1992-01-08
SI9010545A (en)	1997-08-31
RO109737B1 (ro)	1995-05-30
IE900994L (en)	1990-09-20
YU47343B (sh)	1995-01-31
FI914418A0 (fi)	1991-09-19
NO913686L (no)	1991-09-19
HRP920907B1 (en)	1998-06-30
HRP920907A2 (hr)	1994-04-30
FI97387C (fi)	1996-12-10
GEP19971014B (en)	1997-04-18
DD293116A5 (de)	1991-08-22
US5223619A (en)	1993-06-29
RU2090566C1 (ru)	1997-09-20
RU2042668C1 (ru)	1995-08-27
ES2061023T3 (es)	1994-12-01
CA2047217A1 (en)	1990-09-21
BR9007230A (pt)	1992-02-25
AR245719A1 (es)	1994-02-28
DE69013146D1 (de)	1994-11-10
EP0464112B1 (en)	1994-10-05
IE62042B1 (en)	1994-12-14
CS275359B2 (en)	1992-02-19
DK135489D0 (da)	1989-03-20
BG95145A (bg)	1993-12-24
KR0142098B1 (ko)	1998-06-01
KR920701208A (ko)	1992-08-11
WO1990011283A1 (en)	1990-10-04
LV10455A (lv)	1995-02-20
PL163313B1 (pl)	1994-03-31
GR1001096B (el)	1993-04-28
DK0464112T3 (da)	1995-03-13
DE69013146T2 (de)	1995-02-16
GR900100212A (en)	1990-07-31
HU902874D0 (en)	1991-12-30

Publication	Publication Date	Title
BG60590B1 (en)	1995-09-29	Method for the preparation of 9-substituted quanine derivatives
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PL148969B1 (en)	1989-12-30	Method of obtaining novel derivatives of 9-/2-hydroxymethyl/quanine