BG108324A - Нафтотиазин положителни алостерични модулатори на амра - рецептор - Google Patents
Нафтотиазин положителни алостерични модулатори на амра - рецептор Download PDFInfo
- Publication number
- BG108324A BG108324A BG108324A BG10832403A BG108324A BG 108324 A BG108324 A BG 108324A BG 108324 A BG108324 A BG 108324A BG 10832403 A BG10832403 A BG 10832403A BG 108324 A BG108324 A BG 108324A
- Authority
- BG
- Bulgaria
- Prior art keywords
- alkyl
- different
- halogen atoms
- optionally substituted
- general formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10123952A DE10123952A1 (de) | 2001-05-17 | 2001-05-17 | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG108324A true BG108324A (bg) | 2004-12-30 |
Family
ID=7685080
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG108324A BG108324A (bg) | 2001-05-17 | 2003-11-07 | Нафтотиазин положителни алостерични модулатори на амра - рецептор |
Country Status (26)
| Country | Link |
|---|---|
| EP (1) | EP1404340A1 (xx) |
| JP (1) | JP2004529980A (xx) |
| KR (1) | KR20040007572A (xx) |
| CN (1) | CN1533278A (xx) |
| AR (1) | AR036332A1 (xx) |
| BG (1) | BG108324A (xx) |
| BR (1) | BR0209796A (xx) |
| CA (1) | CA2449189A1 (xx) |
| CO (1) | CO5550460A2 (xx) |
| CZ (1) | CZ20033112A3 (xx) |
| DE (1) | DE10123952A1 (xx) |
| EA (1) | EA006608B1 (xx) |
| EC (1) | ECSP034852A (xx) |
| EE (1) | EE200300566A (xx) |
| HR (1) | HRP20030933A2 (xx) |
| HU (1) | HUP0401273A3 (xx) |
| IL (1) | IL158642A0 (xx) |
| MX (1) | MXPA03010373A (xx) |
| NO (1) | NO20035088D0 (xx) |
| NZ (1) | NZ530154A (xx) |
| PL (1) | PL364053A1 (xx) |
| SK (1) | SK14222003A3 (xx) |
| UY (1) | UY27290A1 (xx) |
| WO (1) | WO2002100411A1 (xx) |
| YU (1) | YU90403A (xx) |
| ZA (1) | ZA200308466B (xx) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2061471A4 (en) * | 2006-08-31 | 2012-02-01 | Univ Alberta | PROCESS FOR INHIBITING RESTRICTED DEPRESSION WITH POSITIVE ALLOSTER AMPA RECEPTOR MODULATORS |
| CN111518058B (zh) * | 2020-05-29 | 2021-03-09 | 四川大学华西医院 | 一种噁噻嗪类化合物及其用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998012185A1 (en) * | 1996-09-17 | 1998-03-26 | The Regents Of The University Of California | Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor |
| JP2002518498A (ja) * | 1998-06-25 | 2002-06-25 | メルク エンド カムパニー インコーポレーテッド | ナフト［１，８−ｄｅ］チアジン−２−イルメチルカルバペネム抗菌物質 |
| DE10004572A1 (de) * | 2000-02-02 | 2001-08-09 | Boehringer Ingelheim Pharma | Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
-
2001
- 2001-05-17 DE DE10123952A patent/DE10123952A1/de not_active Withdrawn
-
2002
- 2002-05-15 CN CNA028100832A patent/CN1533278A/zh active Pending
- 2002-05-15 CA CA002449189A patent/CA2449189A1/en not_active Abandoned
- 2002-05-15 WO PCT/EP2002/005338 patent/WO2002100411A1/en not_active Ceased
- 2002-05-15 EE EEP200300566A patent/EE200300566A/xx unknown
- 2002-05-15 IL IL15864202A patent/IL158642A0/xx unknown
- 2002-05-15 HR HR20030933A patent/HRP20030933A2/xx not_active Application Discontinuation
- 2002-05-15 NZ NZ530154A patent/NZ530154A/en unknown
- 2002-05-15 PL PL02364053A patent/PL364053A1/xx not_active Application Discontinuation
- 2002-05-15 EA EA200301167A patent/EA006608B1/ru not_active IP Right Cessation
- 2002-05-15 JP JP2003503232A patent/JP2004529980A/ja not_active Abandoned
- 2002-05-15 HU HU0401273A patent/HUP0401273A3/hu unknown
- 2002-05-15 BR BR0209796-6A patent/BR0209796A/pt not_active IP Right Cessation
- 2002-05-15 UY UY27290A patent/UY27290A1/es not_active Application Discontinuation
- 2002-05-15 KR KR10-2003-7014965A patent/KR20040007572A/ko not_active Withdrawn
- 2002-05-15 MX MXPA03010373A patent/MXPA03010373A/es unknown
- 2002-05-15 CZ CZ20033112A patent/CZ20033112A3/cs unknown
- 2002-05-15 EP EP02750931A patent/EP1404340A1/en not_active Withdrawn
- 2002-05-15 SK SK1422-2003A patent/SK14222003A3/sk unknown
- 2002-05-15 YU YU90403A patent/YU90403A/sh unknown
- 2002-05-17 AR ARP020101827A patent/AR036332A1/es unknown
-
2003
- 2003-10-30 ZA ZA200308466A patent/ZA200308466B/en unknown
- 2003-11-07 BG BG108324A patent/BG108324A/bg unknown
- 2003-11-14 NO NO20035088A patent/NO20035088D0/no not_active Application Discontinuation
- 2003-11-17 EC EC2003004852A patent/ECSP034852A/es unknown
- 2003-12-01 CO CO03105591A patent/CO5550460A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2449189A1 (en) | 2002-12-19 |
| UY27290A1 (es) | 2002-12-31 |
| MXPA03010373A (es) | 2004-03-16 |
| JP2004529980A (ja) | 2004-09-30 |
| NO20035088L (no) | 2003-11-14 |
| HUP0401273A3 (en) | 2006-11-28 |
| EA006608B1 (ru) | 2006-02-24 |
| IL158642A0 (en) | 2004-05-12 |
| YU90403A (sh) | 2006-05-25 |
| NO20035088D0 (no) | 2003-11-14 |
| EE200300566A (et) | 2004-02-16 |
| EA200301167A1 (ru) | 2004-06-24 |
| EP1404340A1 (en) | 2004-04-07 |
| ECSP034852A (es) | 2003-12-24 |
| WO2002100411A1 (en) | 2002-12-19 |
| KR20040007572A (ko) | 2004-01-24 |
| AR036332A1 (es) | 2004-09-01 |
| HUP0401273A2 (hu) | 2004-10-28 |
| NZ530154A (en) | 2005-09-30 |
| DE10123952A1 (de) | 2002-11-21 |
| HRP20030933A2 (en) | 2004-04-30 |
| ZA200308466B (en) | 2004-05-24 |
| PL364053A1 (en) | 2004-12-13 |
| CZ20033112A3 (en) | 2004-03-17 |
| BR0209796A (pt) | 2004-06-01 |
| CO5550460A2 (es) | 2005-08-31 |
| SK14222003A3 (sk) | 2004-05-04 |
| CN1533278A (zh) | 2004-09-29 |
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