[go: up one dir, main page]

BE836528A - Nouveaux derives d'acide 3-amino- indazolecarboxylique - Google Patents

Nouveaux derives d'acide 3-amino- indazolecarboxylique

Info

Publication number
BE836528A
BE836528A BE162651A BE162651A BE836528A BE 836528 A BE836528 A BE 836528A BE 162651 A BE162651 A BE 162651A BE 162651 A BE162651 A BE 162651A BE 836528 A BE836528 A BE 836528A
Authority
BE
Belgium
Prior art keywords
amino
new derivatives
indazolecarboxylic acid
indazolecarboxylic
acid
Prior art date
Application number
BE162651A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE836528A publication Critical patent/BE836528A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BE162651A 1974-12-13 1975-12-11 Nouveaux derives d'acide 3-amino- indazolecarboxylique BE836528A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
BE836528A true BE836528A (fr) 1976-06-11

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
BE162651A BE836528A (fr) 1974-12-13 1975-12-11 Nouveaux derives d'acide 3-amino- indazolecarboxylique

Country Status (27)

Country Link
US (1) US4051252A (fr)
JP (1) JPS5182266A (fr)
AT (1) AT343653B (fr)
BE (1) BE836528A (fr)
CA (1) CA1059523A (fr)
CH (1) CH622250A5 (fr)
CS (1) CS189731B2 (fr)
DD (1) DD125484A5 (fr)
DE (1) DE2458965C3 (fr)
DK (1) DK137082C (fr)
ES (1) ES443429A1 (fr)
FI (1) FI753493A7 (fr)
FR (1) FR2293928A1 (fr)
GB (1) GB1490306A (fr)
HK (1) HK52580A (fr)
HU (1) HU173557B (fr)
IE (1) IE42208B1 (fr)
IL (1) IL48642A (fr)
KE (1) KE3078A (fr)
LU (1) LU73993A1 (fr)
NL (1) NL7514521A (fr)
NO (1) NO145382C (fr)
PL (1) PL99858B1 (fr)
SE (1) SE419645B (fr)
SU (1) SU604487A3 (fr)
YU (1) YU315275A (fr)
ZA (1) ZA757777B (fr)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
EP1698627A1 (fr) * 2000-09-15 2006-09-06 Vertex Pharmaceuticals Incorporated Composés de pyrazole comme inhibiteurs de la protéine kinase
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
ES2242771T5 (es) * 2000-09-15 2011-10-14 Vertex Pharmaceuticals Incorporated Compuestos de pirazol útiles como inhibidores de proteína quinasas.
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
ZA200301703B (en) * 2000-09-15 2004-03-02 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
CN102250071A (zh) 2000-12-21 2011-11-23 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡唑化合物
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
CN1556702A (zh) 2001-09-26 2004-12-22 具有作为激酶抑制剂的活性的氨基吲唑衍生物、它们的制备方法和含有它们的药物组合物
CA2475633C (fr) * 2002-02-06 2013-04-02 Vertex Pharmaceuticals Incorporated Composes heteroaryles utiles en tant qu'inhibiteurs de gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
AU2003218215A1 (en) 2002-03-15 2003-09-29 Vertex Pharmaceuticals, Inc. Azolylaminoazines as inhibitors of protein kinases
EP1506176B1 (fr) 2002-05-17 2013-04-24 Pfizer Italia S.r.l. Derives d'aminoindazole agissant comme inhibiteurs de kinase, methode d'obtention et compositions pharmaceutiques les renfermant
MY141867A (en) 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
AU2003257078B2 (en) 2002-08-02 2010-04-01 Vertex Pharmaceuticals Incorporated Pyrazole compositions useful as inhibitors of GSK-3
WO2004041285A1 (fr) * 2002-10-31 2004-05-21 Amgen Inc. Agents anti-inflammatoires
WO2004072029A2 (fr) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Compositions utiles en tant qu'inhibiteurs de proteine kinases
AU2004297235A1 (en) * 2003-12-04 2005-06-23 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
US7737151B2 (en) 2005-08-18 2010-06-15 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
AR056763A1 (es) * 2005-11-03 2007-10-24 Vertex Pharma Aminopirimidinas sustituidas con tiazol o pirazol,utiles como agentes anticancer y composiciones farmaceuticas que las contienen.
KR101118932B1 (ko) * 2006-04-14 2012-02-27 아보트 러보러터리즈 바닐로이드 서브타입 1(vr1) 수용체를 억제하는 인다졸릴우레아의 제조방법
WO2008057940A1 (fr) 2006-11-02 2008-05-15 Vertex Pharmaceuticals Incorporated Aminopyridines et aminopyrimidines utiles en tant qu'inhibiteurs de protéines kinases
CA2673353A1 (fr) 2006-12-19 2008-06-26 Vertex Pharmaceuticals Incorporated Aminopyridines utiles comme inhibiteurs de proteine kinases
JP2010520887A (ja) 2007-03-09 2010-06-17 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリジン
EP2134707B1 (fr) 2007-03-09 2013-09-11 Vertex Pharmaceuticals, Inc. Aminopyrimidines utiles en tant qu'inhibiteurs des protéines kinases
JP5393489B2 (ja) 2007-03-09 2014-01-22 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリミジン
MX2009011059A (es) 2007-04-13 2009-11-26 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasas.
NZ580884A (en) 2007-05-02 2012-02-24 Vertex Pharma Thiazoles and pyrazoles useful as kinase inhibitors
AU2008247594A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
EP2155730A2 (fr) * 2007-05-02 2010-02-24 Vertex Pharmaceuticals Incorporated Aminopyrimidines servant d'inhibiteurs de kinases
AU2008257044A1 (en) * 2007-05-24 2008-12-04 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
AR067762A1 (es) * 2007-07-31 2009-10-21 Vertex Pharma Proceso para preparar 5-fluoro-1h-pirazolo (3,4-b) piridin-3-amina y derivados de la misma
WO2010027921A1 (fr) * 2008-09-03 2010-03-11 Vertex Pharmaceuticals Incorporated Co-cristaux et formulations pharmaceutiques les comprenant
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
LT2890684T (lt) 2012-07-24 2018-05-10 Bial-Portela & Ca, S.A. Šlapalo junginiai ir jų panaudojimas kaip fermentų inhibitorių
WO2014017938A2 (fr) * 2012-07-27 2014-01-30 BIAL - PORTELA & Cª, S.A. Procédé pour la synthèse de composés d'urée substitués
PT3024825T (pt) 2013-07-24 2017-09-28 BIAL - PORTELA & Cª S A Imidazolecarboxamidas e seu uso como inibidores da faah

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3274203A (en) * 1963-05-31 1966-09-20 Du Pont 1-carbamyl and thiocarbamyl-3-amino-4-nonsubstituted and substituted pyrazoles
NL6707299A (fr) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
ZA757777B (en) 1976-11-24
KE3078A (en) 1980-10-03
IE42208B1 (en) 1980-06-18
DE2458965B2 (de) 1979-02-22
US4051252A (en) 1977-09-27
SE7513990L (sv) 1976-06-14
AU8717075A (en) 1977-06-09
ATA939775A (de) 1977-10-15
DE2458965C3 (de) 1979-10-11
FR2293928A1 (fr) 1976-07-09
ES443429A1 (es) 1977-04-16
CA1059523A (fr) 1979-07-31
CS189731B2 (en) 1979-04-30
IE42208L (en) 1976-06-13
DK137082C (da) 1978-06-19
NO145382B (no) 1981-11-30
FR2293928B1 (fr) 1979-09-21
AT343653B (de) 1978-06-12
SE419645B (sv) 1981-08-17
NL7514521A (nl) 1976-06-15
HU173557B (hu) 1979-06-28
LU73993A1 (fr) 1976-11-11
PL99858B1 (pl) 1978-08-31
DK137082B (da) 1978-01-16
DE2458965A1 (de) 1976-06-16
IL48642A (en) 1979-12-30
YU315275A (en) 1982-02-28
FI753493A7 (fr) 1976-06-14
JPS5182266A (en) 1976-07-19
GB1490306A (en) 1977-11-02
IL48642A0 (en) 1976-02-29
HK52580A (en) 1980-09-26
NO145382C (no) 1982-03-10
DD125484A5 (fr) 1977-04-20
NO754024L (fr) 1976-06-15
SU604487A3 (ru) 1978-04-25
DK567275A (da) 1976-06-14
CH622250A5 (fr) 1981-03-31

Similar Documents

Publication Publication Date Title
BE836528A (fr) Nouveaux derives d'acide 3-amino- indazolecarboxylique
BE851306A (fr) Nouveaux derives de l'acide 3-quinoleine carboxylique
FR2316942A1 (fr) Derives halo-substitues d'acide 1-(alcoyl) inferieur -5-aroylpyrrole-2-acetique
BE827255A (fr) Nouveaux derives de l'amino-3 dihydrothiophenone-2
BE782366A (fr) Nouveaux derives de l'acide cephalosporanique
BE835268A (fr) Derives de l'acide furannehydroxyamique
BE819640A (fr) Nouveaux derives de l'acide phenylbenzoique
BE859846A (fr) Nouveaux derives d'acide alpha-thio-alcanoique
BE809903A (fr) Nouveaux esters o-ethyl-s-n-propyl-o-vinyliques d'acide thionothiolphosphorique
BE822729A (fr) Nouveaux derives de l'acide lysergique
BE821557A (fr) Nouveaux derives de l'acide indane-5-acetique
FR2273806A1 (fr) Derives d'acide barbiturique
BE848023A (fr) Nouveaux derives de l'acide phosphorique,
FR2281101A1 (fr) Derives de l'acide prostanoique
BE828186A (fr) Derives de l'acide prostanoique
BE811209A (fr) Nouveaux derives de l'acide phenylacetique
BE852313A (fr) Nouveaux derives d'acide 4,5-dichlorimidazole-2-carboxylique
FR2305175A1 (fr) Nouveaux derives d'acide prostenoique
BE816343A (fr) Nouveaux derives de l'acide phenyl acetique
BE808969A (fr) Nouveaux derives de l'acide prostanoique
BE852172A (fr) Nouveaux derives de l'acide pyridil-phosphorique
BE782149A (fr) Nouveaux derives de l'acide thiohydroximique
BE823372A (fr) Nouveaux derives de l'acide isonicotinique
FR2100777A1 (fr) Nouveaux derives d'acide benzoique
BE824012A (fr) Derives d'acide butanoique