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AR086688A2 - Composicion farmaceutica con excipiente liquido modificado, un metodo para producir una composicion farmaceutica y el uso de dicha composicion para preparar un medicamento - Google Patents

Composicion farmaceutica con excipiente liquido modificado, un metodo para producir una composicion farmaceutica y el uso de dicha composicion para preparar un medicamento

Info

Publication number
AR086688A2
AR086688A2 ARP120101998A ARP120101998A AR086688A2 AR 086688 A2 AR086688 A2 AR 086688A2 AR P120101998 A ARP120101998 A AR P120101998A AR P120101998 A ARP120101998 A AR P120101998A AR 086688 A2 AR086688 A2 AR 086688A2
Authority
AR
Argentina
Prior art keywords
composition
pharmaceutical composition
liquid carrier
producing
oil
Prior art date
Application number
ARP120101998A
Other languages
English (en)
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of AR086688A2 publication Critical patent/AR086688A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/65Tetracyclines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dermatology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines Containing Plant Substances (AREA)

Abstract

Una composición farmacéutica que comprende: (a) uno o más agentes biológicamente activos; y (b) un excipiente líquido modificado; en donde se proporciona una composición que inmediatamente después de fabricada puede administrarse a un huésped de manera tal que uno o más agentes biológicamente activos se liberan al huésped en forma continua y predecible; un método para producir una composición farmacéutica y el uso de dicha composición para preparar un medicamento para tratar o prevenir una enfermedad en un mamífero.Reivindicación 1: Una composición farmacéutica caracterizada porque comprende: (a) ácido libre de ceftiofur cristalino; y (b) un portador líquido, dicho portador líquido comprende un aceite insaturado que tiene un valor de peróxido de entre 0.1 y 600 miliequivalentes (mEq) de peróxido por 1000 gramos de aceite. Reivindicación 2: La composición según la reivindicación 1 caracterizada porque dicho portador líquido comprende una mezcla de un aceite insaturado con un aceite saturado. Reivindicación 8: La composición de la reivindicación 1, caracterizada porque dicho portador líquido comprende una mezcla de dicho aceite insaturado con un vehículo no oxidante.
ARP120101998A 2000-09-12 2012-06-06 Composicion farmaceutica con excipiente liquido modificado, un metodo para producir una composicion farmaceutica y el uso de dicha composicion para preparar un medicamento AR086688A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23176700P 2000-09-12 2000-09-12

Publications (1)

Publication Number Publication Date
AR086688A2 true AR086688A2 (es) 2014-01-15

Family

ID=22870572

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP010104286A AR030648A1 (es) 2000-09-12 2001-09-11 Composicion farmaceutica con excipiente modificado
ARP120101998A AR086688A2 (es) 2000-09-12 2012-06-06 Composicion farmaceutica con excipiente liquido modificado, un metodo para producir una composicion farmaceutica y el uso de dicha composicion para preparar un medicamento

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP010104286A AR030648A1 (es) 2000-09-12 2001-09-11 Composicion farmaceutica con excipiente modificado

Country Status (18)

Country Link
US (1) US20020110561A1 (es)
EP (1) EP1317256B1 (es)
JP (1) JP4738713B2 (es)
AR (2) AR030648A1 (es)
AT (1) ATE412405T1 (es)
AU (2) AU8832301A (es)
BR (1) BRPI0113372B8 (es)
CA (1) CA2416566C (es)
DE (1) DE60136367D1 (es)
DK (1) DK1317256T3 (es)
ES (1) ES2313981T3 (es)
MX (1) MXPA03002055A (es)
NZ (1) NZ524694A (es)
PE (1) PE20030046A1 (es)
PT (1) PT1317256E (es)
TW (1) TWI284046B (es)
WO (1) WO2002022107A2 (es)
ZA (1) ZA200300617B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040033938A1 (en) * 2000-09-12 2004-02-19 Britten Nancy J. Cyclooxygenase-2 inhibitor and antibacterial agent combination for intramammary treatment of mastitis
KR20040015622A (ko) * 2002-08-13 2004-02-19 대한뉴팜(주) 세프티오푸르나트륨을 활성성분으로 함유하는 현탁주사액조성물
US7659061B2 (en) * 2002-11-19 2010-02-09 Pharmacia & Upjohn Company Pharmaceutical compositions having a modified vehicle
US7842791B2 (en) * 2002-12-19 2010-11-30 Nancy Jean Britten Dispersible pharmaceutical compositions
US20080153894A1 (en) * 2002-12-19 2008-06-26 Pharmacia Corporation Cyclooxygenase-2 inhibitor and antibacterial agent combination for intramammary treatment of mastitis
CA2743551C (en) * 2008-11-19 2017-08-15 Merial Limited Formulations comprising ceftiofur and ketoprofen or ceftiofur and benzyl alcohol
BRPI0903778B1 (pt) 2009-07-17 2017-04-18 Cargill Agrícola S A composição alimentícia de gordura vegetal, processo de preparação de uma composição alimentícia de gordura vegetal e uso de uma composição alimentícia de gordura vegetal na preparação de recheio
MX340951B (es) * 2011-09-29 2016-07-29 Plx Pharma Inc Portadores dependientes del ph para la liberacion dirigida de productos farmaceuticos a lo largo del tracto gastrointestinal, composiciones de los mismos, y fabricación y uso de las mismas.
CA2968320A1 (en) 2014-11-19 2016-05-26 Cassandra K JONES Chemical mitigants in animal feed and feed ingredients
PH12021551973A1 (en) 2019-03-06 2022-05-23 Zoetis Services Llc Ready-to-use injectable formulations

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE122005000055I2 (de) * 1993-03-12 2008-06-05 Upjohn Co Kristallines ceftiofur (freie säure)
US5736151A (en) * 1996-12-09 1998-04-07 Pharmacia & Upjohn Company Antibiotic oil suspensions
US6074657A (en) * 1997-03-20 2000-06-13 Pharmacia & Upjohn Company Administration of an injectable antibiotic in the ear of an animal

Also Published As

Publication number Publication date
US20020110561A1 (en) 2002-08-15
CA2416566C (en) 2011-05-31
BRPI0113372B1 (pt) 2017-08-01
NZ524694A (en) 2005-05-27
JP2004508395A (ja) 2004-03-18
PT1317256E (pt) 2008-12-17
EP1317256A2 (en) 2003-06-11
CA2416566A1 (en) 2002-03-21
JP4738713B2 (ja) 2011-08-03
DE60136367D1 (de) 2008-12-11
EP1317256B1 (en) 2008-10-29
ATE412405T1 (de) 2008-11-15
AU2001288323B2 (en) 2006-11-23
ZA200300617B (en) 2004-04-22
ES2313981T3 (es) 2009-03-16
BRPI0113372A8 (es) 2003-06-24
BRPI0113372B8 (pt) 2021-10-13
PE20030046A1 (es) 2003-02-14
MXPA03002055A (es) 2004-12-13
DK1317256T3 (da) 2009-01-26
TWI284046B (en) 2007-07-21
AU8832301A (en) 2002-03-26
WO2002022107A2 (en) 2002-03-21
WO2002022107A3 (en) 2003-01-16
AR030648A1 (es) 2003-08-27
BR0113372A (pt) 2003-06-24

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal