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AR070228A1 - Derivados de 5-fluoro pirimidina - Google Patents

Derivados de 5-fluoro pirimidina

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Publication number
AR070228A1
AR070228A1 ARP090100193A ARP090100193A AR070228A1 AR 070228 A1 AR070228 A1 AR 070228A1 AR P090100193 A ARP090100193 A AR P090100193A AR P090100193 A ARP090100193 A AR P090100193A AR 070228 A1 AR070228 A1 AR 070228A1
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AR
Argentina
Prior art keywords
alkyl
optionally substituted
phenyl
benzyl
haloalkyl
Prior art date
Application number
ARP090100193A
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English (en)
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Dow Agrosciences Llc
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Publication of AR070228A1 publication Critical patent/AR070228A1/es

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
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    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
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    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
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    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/18—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
    • A—HUMAN NECESSITIES
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    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/24—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing the groups, or; Thio analogues thereof
    • A—HUMAN NECESSITIES
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    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/36—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< directly attached to at least one heterocyclic ring; Thio analogues thereof
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    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • A01N47/42—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides containing —N=CX2 groups, e.g. isothiourea
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • A01N47/42—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides containing —N=CX2 groups, e.g. isothiourea
    • A01N47/44—Guanidine; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/26—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-nitrogen bonds
    • A01N57/32—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having phosphorus-to-nitrogen bonds containing heterocyclic radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Health & Medical Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente se refiere al campo de las 5-fluoro pirimidinas y a los derivados de las mismas y al uso de estos compuestos como fungicidas. Composiciones fungicidas y método de control o prevencion de un ataque fungico a una planta. Reivindicacion 1: Un compuesto de la formula 1 en donde R1 es -N(R3)R4; R2 es -OR21; R3 es H, alquilo C1-6 opcionalmente sustituido con 1-3 R5, alquenilo C2-6 opcionalmente sustituido con 1-3 R5, un anillo heteroaromático de 5 o 6 miembros seleccionado a partir del grupo formado por furanilo, piridinilo, piridinil-N-oxido, pirimidinilo, piridazinilo, pirazinilo, tiazolilo, triazinilo, tiadiazolilo, oxazolilo, isoxazolilo, triazolilo, en donde cada anillo heteroaromático es opcionalmente sustituido con 1-3 R30; imidazol fusionado con un anillo aromático o heteroaromático seleccionado entre el grupo formado por benceno, oxazol, isoxazol, furan, tiazol, pirimidina, piridina, pirrol, pirazina, tiofeno, en donde cada anillo aromático heteroaromático es opcionalmente sustituido con 1-3 R30; benzo[1,3]dioxolilo; 3H-isobenzofuran-1-onilo; ciano; alquinilo C3-6 opcionalmente sustituido con 1-3 R5, -C(=O)R6; -C(=S)NHR8 , -OR7; -P(O)(OR15)2; -S(O)2R8, -SR8, -Si(R8)3, -N(R9)R10; -N=C(R15)R16; -(CHR22)mR23; -(CHR24)OR29; -C(=O)N(R8)R10; en donde m es un entero de 1-3; R4 es alquilo C1-6, opcionalmente sustituido con 1-3 R5; o -C=O(R6); -C(=O)N(R8)R10; alternativamente R3 y R4 pueden tomarse juntos para formar: un anillo saturado o insaturado de 5 o 6 miembros que contiene 1-3 heteroátomos en donde cada anillo puede ser opcionalmente sustituido con 1 a 3 R11; =C(R12)N(R13)R14; =C(R13)(R14); o =C(R15)OR15; R5 es independientemente halogeno, alquilo C1-6, haloalquilo C1-4, alcoxi C1-4, haloalcoxi C1-4, alquiltio C1-4, haloalquiltio C1-4, amino, alquilamino C1-3, alcoxicarbonilo C2-6, alquilcarbonilo C2-6, alquilaminocarbonilo C2-6, -OH, N-metil piperazina o trialquilsililo C3-6; R6 es independientemente H, alquilo C1-6, haloalquilo C1-5, alcoxi C1-5, alcoxicarbonilo C2-6; alquilaminocarbonilo C2-6; 1-benzo[1,2,3]tiadiazol-7-ilo, tiazolilo, bencilo, fenilo, fenoxi , o benciloxi en donde tiazol, bencilo, fenilo, fenoxi, o benciloxi pueden ser opcionalmente sustituidos con 1-3 R20; R7 es H, alquilo C1-6, alquenilo C2-6, haloalquilo C1-5, bencilo que pueden ser opcionalmente sustituidos con 1-5 R20, un anillo saturado o insaturado de 5 o 6 miembros que contiene 1-3 heteroátomos en donde cada anillo puede ser opcionalmente sustituido con 1 a 3 R11, o CHR18C(O)OR19; R8 es alquilo C1-6, haloalquilo C1-6, o fenilo opcionalmente sustituido con 1-3 R20; R9 es H, alquil C1-6-haloalquilo C1-6, o fenilo opcionalmente sustituido con 1-3 R20, o -C(=O)R17; R10 es H o alquilo C1-6; haloalquilo C1-6, o fenilo opcionalmente sustituido con 1-3 R20; R11 es independientemente halogeno, alquilo C1-6, alcoxi C1-6, haloalcoxi C1-6, alquiltio C1-6, haloalquiltio C1-6, amino, alquilamino C1-6, dialquilamino C2-6, alcoxicarbonilo C2-6, o alquilcarbonilo C2-6; R12 es H o alquilo C1-4; R13 y R14 son independientemente H, ciano, -OH, alquilo C1-4, alcoxi C1-6, alquilcarbonilo C2-6, fenilo, o bencil en donde el fenilo o bencilo pueden ser opcionalmente sustituidos con 1-3 R20; alternativamente R13 y R14 pueden tomarse conjuntamente para formar: un anillo saturado o insaturado de 5 o 6 miembros que contiene 1-3 heteroátomos en donde cada anillo puede ser opcionalmente sustituido con 1 a 3 R11, o 3,4-dihidro-1H-isoquinolin-2-ilo; R15 es H o alquilo C1-6; R16 es H, alquilo C1-6, fenilo opcionalmente sustituido con 1-3 R20, alternativamente R15 y R16 pueden tomarse conjuntamente como -(CH2)4- o -(CH2)5-; R17 es H, alquilo C1-6, haloalquilo C1-6, alcoxi C1-6, fenilo, fenoxi , o benciloxi en donde cada anillo puede ser opcionalmente sustituido con 1 a 3 R20; R18 es H, alquilo C1-6, o haloalquilo C1-6; R19 es H, alquilo C1-6, haloalquilo C1-6, o bencilo; R20 es independientemente halogeno, ciano, nitro, amino, alcoxialcoxi C1-6, alquilo C1-6, haloalquilo C1-6, hidroxi C1-6 alquilo, alcoxialquilo C2-6, haloalcoxialquilo C2-6, alquenilo C2-6, haloalquenilo C2-6, alquinilo C3-6, haloalquinilo C3-6, hidroxilo, alcoxi C1-6, haloalcoxi C1-6, alqueniloxi C2-6, haloalqueniloxi C2-6, alquiniloxi C3-6, haloalquiniloxi C3-6, alquiltio C1-6, haloalquiltio C1-6, alquilsulfonilo C1-6, haloalquilsulfonilo C1-6, alqueniltio C2-6, haloalqueniltio C2-6, haloalquenilsulfonilo C2-6, alquiniltio C3-6, alquinilsulfonilo C3-6, haloalquinilsulfonilo C3-6, alquilamino C1-6, dialquilamino C2-8, dialquilaminocarbonilo C3-8, trialquilsililo C3-6, 2-[(E)-metoxi imino]-N-metil-acetamidilo, fenilo, bencilo, benciloxi, fenoxi, un anillo heteroaromático de 5 o 6 miembros, en donde cada fenilo, bencilo, benciloxi, fenoxi, o anillo heteroaromático de 5 o 6 miembros puede ser opcionalmente sustituido con 1-3 sustituyentes independientemente seleccionados entre R31; R21 es H, alquilo C1-14; haloalquilo C1-6; alquenilo C2-4; haloalquenilo C2-4; alquinilo C3-4, haloalquinilo C3-4; fenilo, naftilo, o tetrahidroquinolinilo en donde cada uno es opcionalmente sustituido con 1-3 R20; -(CHR22)mR23; -(CHR24)mC(O)OR25; -(CHR24)mC(O)R26; -(CHR24)mC(O)N(R27)R28; -(CHR24)mOR29; -(CHR24)mSR29, -(CHR24)mN(R27)R28, -C(=O)R32; -N=C(R24)(R32); -Si(R8)3; -SO2R33; alcoxi C2-6 carbonilo; alquilaminocarbonilo C2-6, alquilcarbonilo C2-6; azucares seleccionados entre el grupo formado por beta-D-glucosa- tetraacetato, ramnosa, fructosa, y pentosa; o un anillo heteroaromático de 5 o 6 miembros que incluye furanilo, piridinilo, piridinil-N-oxido, pirimidinilo, piridazinilo, pirazinilo, pirazolilo, tiazolilo, triazinilo, tiadiazolilo, oxazolilo, triazolilo o isoxazolilo en donde cada anillo heteroaromático de 5 o 6 miembros puede ser opcionalmente sustituido con 1 a 5 R20; R22 es independientemente H; halogeno; ciano; nitro; alquilo C1-6, haloalquilo C1-6; fenilo o bencilo opcionalmente sustituido con 1-3 R20; hidroxi C1-6 alquilo; alcoxialquilo C2-6; haloalquinilo C3-6; alquenilo C2-6, haloalquenilo C2-6; alquinilo C3-6; alcoxi C1-6; haloalcoxi C1-6, alquiltio C1-6, alquilamino C1-6; dialquilamino C2-8; cicloalquilamino C3-6; alquil C4-6 cicloalquilamino; alquilcarbonilo C2-6, alcoxicarbonilo C2-6; alquilaminocarbonilo C2-6; dialquilaminocarbonilo C3-8; trialquilsililo C3-6; benzo[ 1,3]dioxolilo; anillos heteroaromáticos de anillo fusionado seleccionados entre el grupo formado por benzotiofenilo, quinolinilo, isoquinolinilo, tieno[2,3-b]piridilo, 1-metil-1H-tieno[2,3-c]pirazolilo, y benzoimidazolilo, en donde cada uno de los anillos puede ser además sustituido con 1 a 3 R20; o un anillo heteroaromático de 5 o 6 miembros seleccionado entre el grupo formado por furanilo, piridinilo, piridinil-N-oxido, pirimidinilo, piridazinilo, pirazinilo, tiazolilo, triazinilo, tiadiazolilo, oxazolilo, isoxazolilo, triazolilo o tienilo; R23 es H; halogeno; alquilo C1-6; haloalquilo C1-6; dialquilamino C2-6; fenilo opcionalmente sustituido con 1 a 5 R20; anillo heteroaromáticos de anillo fusionado seleccionados entre el grupo formado por benzotiofenilo, quinolinilo, isoquinolinilo, tieno[2,3-b]piridilo, 1-metil-1H-tieno[2,3-c]pirazolilo, benzofuranil y benzoimidazolilo, en donde cada uno de los anillos puede ser además sustituido con 1 a 3 R20; naftalilo; pirrolidinonilo; oxetanilo; alquiltio C1-6 opcionalmente sustituido con 1 a 5 R20; un anillo saturado o insaturado de 5 o 6 miembros que contiene 1-3 heteroátomos en donde cada anillo puede ser opcionalmente sustituido con 1 a 3 R11, o un anillo heteroaromático de 5 o 6 miembros seleccionado entre el grupo formado por furanilo, piridinilo, piridinil-N-oxido, pirimidinilo, piridazinilo, pirazinilo, pirazolilo, tiazolilo, triazinilo, tiadiazolilo, oxazolilo, isoxazolilo, triazolilo, imidazolilo, tiofeno-2-ilo y tiofen-3-ilo en donde cada anillo heteroaromático puede ser opcionalmente sustituido con 1 a 3 R20; R24 es H, alquilo C1-6, alcoxi C1-6, bencilo, o fenilo en donde cada uno, entre bencilo o fenilo pueden ser opcionalmente sustituidos con 1-3 R20; R25 es H, alquilo C1-6, o bencil opcionalmente sustituido con 1-3 R20; R26 es H; alquilo C1-6, alcoxi C1-6; fenilo opcionalmente sustituido con 1-3 R20; o un anillo heteroaromático de 5 o 6 miembros que incluye furanilo, piridinilo, piridinil-N-oxido, pirimidinilo, piridazinilo, pirazinilo, tiazolilo, triazinilo, tiadiazolilo, oxazolilo, triazolilo o isoxazolilo; R27 y R28 son independientemente H, alquilo C1-6; bencilo, o fenilo en donde cada uno entre bencilo o fenilo puede ser opcionalmente sustituido con 1-3 R20 o un anillo saturado o insaturado de 5 o 6 miembros que contiene 1-3 heteroátomos en donde cada anillo puede ser opcionalmente sustituido con 1 a 3 R11; R29 es H, alquilo C1-6, alcoxialquilo C1-6, alquilcarbonilo, bencilo, o fenilo en donde cada uno entre bencil o fenilo puede ser opcionalmente sustituido con 1-3 R20; y R30 es independientemente halogeno, ciano, nitro, alquilo C1-6, haloalquilo C1-6, hidroxi C1-6 alquilo, alcoxialquilo C2-6, haloalcoxialquilo C2-6, alquenilo C2-6, haloalquenilo C2-6, alquinilo C3-6, haloalquinilo C3-6, hidroxilo, alcoxi C1-6, haloalcoxi C1-6, alqueniloxi C2-6, haloalqueniloxi C2-6, alquiniloxi C3-6, haloalquiniloxi C3-6, alquiltio C1-6, alquilsulfonilo C1-6, haloalquilsulfonilo C1-6, alqueniltio C2-6, haloalqueniltio C2-6, haloalquenilsulfonilo C2-6, alquiniltio C3-6, alquinilsulfonilo C3-6, haloalquinilsulfonilo C3-6, alquilamino C1-6, dialquilamino C2-8, dialquilaminocarbonilo C3-8, trialquilsililo C3-6, tiazolilo, fenilo, pirimidinilo en donde el tiazolilo, fenilo, o pirimidinilo puede ser opcionalmente sustituido con 1 a 3 R20; R31 es independientemente halogeno, ciano, nitro, alquilo C1-6, haloalquilo C1-6, hidroxi C1-6 alquilo, alcoxialquilo C2-6, haloalcoxialquilo C2-6, alquenilo C2-6, haloalquenilo C2-6, alquinilo C3-6, haloalquinilo C3-6, hidroxilo, alcoxi C1-6, haloalcoxi C1-6, alqueniloxi C2-6, haloalqueniloxi C2-6, alquiniloxi C3-6, haloalquiniloxi C3-6, alquilt
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