AR068835A1 - Derivados sustituidos de azinilo insecticidas - Google Patents
Derivados sustituidos de azinilo insecticidasInfo
- Publication number
- AR068835A1 AR068835A1 ARP080104403A ARP080104403A AR068835A1 AR 068835 A1 AR068835 A1 AR 068835A1 AR P080104403 A ARP080104403 A AR P080104403A AR P080104403 A ARP080104403 A AR P080104403A AR 068835 A1 AR068835 A1 AR 068835A1
- Authority
- AR
- Argentina
- Prior art keywords
- alkyl
- optionally substituted
- maximum amount
- alkoxy
- chlorine
- Prior art date
Links
- 239000002917 insecticide Substances 0.000 title 1
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 12
- 229910052801 chlorine Inorganic materials 0.000 abstract 6
- 239000000460 chlorine Substances 0.000 abstract 6
- 229910052731 fluorine Inorganic materials 0.000 abstract 6
- 125000001153 fluoro group Chemical group F* 0.000 abstract 5
- 125000006274 (C1-C3)alkoxy group Chemical group 0.000 abstract 4
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 3
- 229910052794 bromium Inorganic materials 0.000 abstract 3
- 229910052740 iodine Inorganic materials 0.000 abstract 3
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 2
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 2
- 239000011737 fluorine Substances 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- JCXJVPUVTGWSNB-UHFFFAOYSA-N nitrogen dioxide Inorganic materials O=[N]=O JCXJVPUVTGWSNB-UHFFFAOYSA-N 0.000 abstract 2
- 125000001889 triflyl group Chemical group FC(F)(F)S(*)(=O)=O 0.000 abstract 2
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000000051 benzyloxy group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])O* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000000749 insecticidal effect Effects 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
- A01N47/36—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< directly attached to at least one heterocyclic ring; Thio analogues thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
- C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
- C07D251/12—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D251/26—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
- C07D251/40—Nitrogen atoms
- C07D251/42—One nitrogen atom
- C07D251/46—One nitrogen atom with oxygen or sulfur atoms attached to the two other ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Public Health (AREA)
- Agronomy & Crop Science (AREA)
- Medicinal Chemistry (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pyridine Compounds (AREA)
Abstract
Composicion insecticida y método de control. Reivindicacion 1: Un compuesto de la formula (1) en donde A, B y D representan N, CH o CR3, siempre que al menos uno de A, B o D sea N; R1 representa alquilo C1-4 opcionalmente sustituido con uno a la cantidad máxima de átomos de fluor o de cloro; R2 representa C1, CF3, O(alquilo C1-3), NH(alquilo C1-3) o N(alquilo C1-3)2 en donde cada uno de los grupos alquilo C1-3 anteriores está opcionalmente sustituido con uno a la cantidad máxima de átomos de fluor; R3 representa H, F, Cl, Br, I, alquilo C1-3 u O(alquilo C1-3), en donde cada uno de los grupos alquilo C1-3 anteriores está opcionalmente sustituido con uno a la cantidad máxima de átomos de fluor; representa H, alquilo C1-3 (opcionalmente sustituido con alcoxi, benciloxi u -OC(O)R7) o CO2R6; R5 representa H, alquilo C1-3 (opcionalmente sustituido con alcoxi C1-3, F, CN o CO2R), OH, alcoxi C1-3 o CO2R6 o R4 y R5 tomados juntos representan -CH2CH2- o -C(O)CH2-; R6 representa H o alquilo C1-3; R7 representa alquilo C1-3; W representa O o S; Ar representa un grupo fenilo sustituido con uno a cuatro sustituyentes seleccionados, de modo independiente, de F, Cl, Br, I, NO2, CN, SCF3, SO2CF3, alquilo C1-3 sustituido con uno a la cantidad máxima de átomos de cloro o de fluor o alcoxi C1-3 opcionalmente sustituido con uno a la cantidad máxima de átomos de cloro o de fluor; o representa (2) X e Y representan, de modo independiente, H, F, Cl, Br, I, NO2, CN, SCF3, SO2CF3, alquilo C2-3 sustituido con uno a la cantidad máxima de átomos de cloro o de fluor o alcoxi C1-3 opcionalmente sustituido con uno a la cantidad máxima de átomos de cloro o de fluor.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US99825007P | 2007-10-09 | 2007-10-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR068835A1 true AR068835A1 (es) | 2009-12-09 |
Family
ID=40456231
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080104403A AR068835A1 (es) | 2007-10-09 | 2008-10-08 | Derivados sustituidos de azinilo insecticidas |
Country Status (6)
| Country | Link |
|---|---|
| US (3) | US8013154B2 (es) |
| EP (1) | EP2195302B1 (es) |
| JP (3) | JP5567483B2 (es) |
| AR (1) | AR068835A1 (es) |
| ES (1) | ES2532119T3 (es) |
| WO (1) | WO2009048752A2 (es) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8013154B2 (en) * | 2007-10-09 | 2011-09-06 | Niyaz Noormohamed M | Insecticidal substituted azinyl derivatives |
| EP2595965B1 (en) | 2010-07-20 | 2016-06-22 | Vestaron Corporation | Insecticidal triazines and pyrimidines |
| CA2888225A1 (en) | 2012-11-12 | 2014-05-15 | Dow Agrosciences Llc | Pesticidal pyrimidine compounds |
| WO2015178262A1 (ja) * | 2014-05-22 | 2015-11-26 | 住友化学株式会社 | ピラゾール化合物 |
| CN107530304A (zh) | 2015-02-27 | 2018-01-02 | 科泰纳制药公司 | Olig2活性的抑制 |
| CN106588884B (zh) * | 2016-11-10 | 2019-04-09 | 浙江大学 | 2-多取代芳环-嘧啶类衍生物及制备和医药用途 |
| CN108084158A (zh) * | 2016-11-23 | 2018-05-29 | 江苏豪森药业集团有限公司 | 右兰索拉唑的制备方法 |
| EP3284739A1 (de) * | 2017-07-19 | 2018-02-21 | Bayer CropScience Aktiengesellschaft | Substituierte (het)arylverbindungen als schädlingsbekämpfungsmittel |
| CN114728933B (zh) * | 2020-07-22 | 2023-06-16 | 山东绿叶制药有限公司 | 5-ht2a受体抑制剂或反向激动剂及其制备方法和应用 |
| WO2022046650A1 (en) * | 2020-08-24 | 2022-03-03 | Curtana Pharmaceuticals, Inc. | Combination therapies with olig2 inhibitors |
| JP2025066196A (ja) * | 2022-03-14 | 2025-04-23 | 国立大学法人東北大学 | 認知機能改善剤 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3857883A (en) * | 1972-05-08 | 1974-12-31 | Chevron Res | N-chlorothio urea production |
| JPS51125092A (en) * | 1974-08-26 | 1976-11-01 | Toyama Chem Co Ltd | A process for preparing novel substituted s-triazines |
| JPS56147771A (en) * | 1980-04-15 | 1981-11-16 | Toshihiko Okamoto | N- 2,6-disubstituted-4-pyridyl urea and thiourea |
| US4308054A (en) * | 1979-11-02 | 1981-12-29 | Yo Isogai | N-(2,6-Disubstituted-4-pyridyl)-N'-phenylureas |
| US4747870A (en) * | 1986-05-02 | 1988-05-31 | E. I. Du Pont De Nemours And Company | Herbicidal pyrazole sulfonamides |
| GB8700838D0 (en) * | 1987-01-15 | 1987-02-18 | Shell Int Research | Termiticides |
| US5399564A (en) * | 1991-09-03 | 1995-03-21 | Dowelanco | N-(4-pyridyl or 4-quinolinyl) arylacetamide and 4-(aralkoxy or aralkylamino) pyridine pesticides |
| WO2003030909A1 (en) | 2001-09-25 | 2003-04-17 | Bayer Pharmaceuticals Corporation | 2- and 4-aminopyrimidines n-substtituded by a bicyclic ring for use as kinase inhibitors in the treatment of cancer |
| US6693097B2 (en) * | 2001-11-30 | 2004-02-17 | Synta Pharmaceuticals Corp. | Pyrimidine compounds |
| CA2479037C (en) | 2002-03-15 | 2010-11-09 | Jiri Zemlicka | 2-amino-9[(2-hydroxymethyl)cyclopropylidenemethyl]purines as antiviral agents |
| TW200407315A (en) | 2002-04-23 | 2004-05-16 | Sankyo Co | Pyrimidine derivatives |
| CN1508130A (zh) * | 2002-12-18 | 2004-06-30 | 中国科学院大连化学物理研究所 | N-苯基-n’-嘧啶基取代脲类衍生物的合成方法 |
| CN1510033A (zh) * | 2002-12-24 | 2004-07-07 | 中国科学院大连化学物理研究所 | 一种合成非对称二吡啶基取代脲类衍生物的新方法 |
| WO2008007788A1 (fr) | 2006-07-14 | 2008-01-17 | Asahi Glass Company, Limited | Structure et son procédé de fabrication |
| FR2910477B1 (fr) | 2006-12-22 | 2009-04-10 | Total France Sa | Fluxant et ses applications. |
| US8013154B2 (en) * | 2007-10-09 | 2011-09-06 | Niyaz Noormohamed M | Insecticidal substituted azinyl derivatives |
-
2008
- 2008-09-26 US US12/239,079 patent/US8013154B2/en active Active
- 2008-09-26 ES ES08837395.6T patent/ES2532119T3/es active Active
- 2008-09-26 JP JP2010528937A patent/JP5567483B2/ja not_active Expired - Fee Related
- 2008-09-26 EP EP08837395.6A patent/EP2195302B1/en not_active Not-in-force
- 2008-09-26 WO PCT/US2008/077888 patent/WO2009048752A2/en not_active Ceased
- 2008-10-08 AR ARP080104403A patent/AR068835A1/es unknown
-
2011
- 2011-07-22 US US13/188,568 patent/US8507671B2/en active Active
- 2011-07-22 US US13/188,593 patent/US8455649B2/en active Active
-
2014
- 2014-05-21 JP JP2014105239A patent/JP5826327B2/ja not_active Expired - Fee Related
- 2014-05-21 JP JP2014105238A patent/JP5813825B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20120190684A1 (en) | 2012-07-26 |
| US20090093486A1 (en) | 2009-04-09 |
| JP5567483B2 (ja) | 2014-08-06 |
| US20120190683A1 (en) | 2012-07-26 |
| JP5826327B2 (ja) | 2015-12-02 |
| JP2011500574A (ja) | 2011-01-06 |
| JP5813825B2 (ja) | 2015-11-17 |
| EP2195302A2 (en) | 2010-06-16 |
| JP2014205678A (ja) | 2014-10-30 |
| WO2009048752A2 (en) | 2009-04-16 |
| US8507671B2 (en) | 2013-08-13 |
| EP2195302B1 (en) | 2015-02-18 |
| WO2009048752A3 (en) | 2009-05-28 |
| US8013154B2 (en) | 2011-09-06 |
| JP2014208648A (ja) | 2014-11-06 |
| US8455649B2 (en) | 2013-06-04 |
| ES2532119T3 (es) | 2015-03-24 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR068835A1 (es) | Derivados sustituidos de azinilo insecticidas | |
| AR055053A1 (es) | Compuestos indol sustituidos con actividad inhibidora de nos. composiciones farmaceuticas. | |
| CR10499A (es) | Profarmaco de compuesto de cinamida | |
| CY1113782T1 (el) | Παραγωγα 11-υδροξυ-5η-πυρρολο[2,1-c][1,4]βενζοδιαζεπιν-5-ονης ως ενδιαμεσα κλειδια για την παρασκευη c2 υποκατεστημενων πυρρολοβενζοδιαζεπινων | |
| EP1795536A4 (en) | PHOSPHORAMIDITE COMPOUND AND PROCESS FOR THE PREPARATION OF OLIGO RNA | |
| EA201892191A1 (ru) | Соединения гетероарил-1,2,4-триазола и гетероарил-тетразола для контроля над эктопаразитами | |
| WO2003016291A1 (en) | ACTIVATOR FOR PEROXISOME PROLIFERATOR-RESPONSIVE RECEPTOR δ | |
| RU2009124489A (ru) | Соединения бензоилпиразола, способ их получения и гербициды, содержащие их | |
| MEP24208A (en) | Derivatives of dioxane-2-alkyl carbamates, preparation method thereof and application of same in therapeutics | |
| DK0795025T3 (da) | Enantioselektiv fremstilling af farmaceutisk aktive sulfoxider ved bioreduktion | |
| DK2177503T3 (da) | Modulatorer af cannabinoidreceptorer | |
| NZ581438A (en) | Kallikrein 7 modulators | |
| MY146663A (en) | Organic sulfur compound and its use for controlling harmful arthropod | |
| NZ331123A (en) | 2-(benzo-1,4-oxathiin)- or (benzo-1,4-dithiin)-cyclohexane-1,3-diones and herbicidal compositions | |
| MY160882A (en) | Biocidal composition and method | |
| HRP20040230B1 (hr) | Agonisti muskarina | |
| WO2003097644A3 (en) | Non-nucleoside reverse transcriptase inhibitors | |
| DK1706414T3 (da) | Fremgangsmåde til fluorcytidinderivater | |
| ATE550332T1 (de) | 4-imidazolin-2-onverbindungen als p38-map- kinaseinhibitors | |
| ATE428693T1 (de) | Prostaglandinsynthese | |
| AR054386A1 (es) | Moduladores de quinasas con estructuras de alquiloquinolina y alquilquinazolina | |
| IS7841A (is) | Efnafræðilegt milliefni | |
| HRP20070286T3 (en) | Substituted diketopiperazines and their use as oxytocyn antagonists | |
| GB0326964D0 (en) | Chemical compounds | |
| AR055666A1 (es) | Inhibidores inntr |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |