AR065108A1 - Proceso para elaborar (r)-5-(2-aminoetil)-1-(6,8-difluorocromo-3-il)-1,3-dihidroimidazol-2-tiona - Google Patents
Proceso para elaborar (r)-5-(2-aminoetil)-1-(6,8-difluorocromo-3-il)-1,3-dihidroimidazol-2-tionaInfo
- Publication number
- AR065108A1 AR065108A1 ARP080100396A ARP080100396A AR065108A1 AR 065108 A1 AR065108 A1 AR 065108A1 AR P080100396 A ARP080100396 A AR P080100396A AR P080100396 A ARP080100396 A AR P080100396A AR 065108 A1 AR065108 A1 AR 065108A1
- Authority
- AR
- Argentina
- Prior art keywords
- difluorocromo
- aminoetil
- tiona
- dihydroimidazol
- prepare
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Reivindicacion 1: un proceso para elaborar un compuesto de la formula 1; que comprende hacer reaccionar un compuesto de la formula 2; con dihidroxiacetona y un tiocianato soluble en agua, y un acido organico presencia de un disolvente.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0701965.6A GB0701965D0 (en) | 2007-02-01 | 2007-02-01 | Process |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR065108A1 true AR065108A1 (es) | 2009-05-13 |
Family
ID=37891142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP080100396A AR065108A1 (es) | 2007-02-01 | 2008-01-31 | Proceso para elaborar (r)-5-(2-aminoetil)-1-(6,8-difluorocromo-3-il)-1,3-dihidroimidazol-2-tiona |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20100113799A1 (es) |
| EP (1) | EP2114926A1 (es) |
| JP (1) | JP2010517999A (es) |
| KR (1) | KR20090104898A (es) |
| CN (1) | CN101627032A (es) |
| AR (1) | AR065108A1 (es) |
| AU (1) | AU2008211846A1 (es) |
| BR (1) | BRPI0806402A2 (es) |
| CA (1) | CA2677203A1 (es) |
| GB (1) | GB0701965D0 (es) |
| IL (1) | IL200178A0 (es) |
| MX (1) | MX2009008244A (es) |
| RU (1) | RU2009132668A (es) |
| WO (1) | WO2008094055A1 (es) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5438150A (en) * | 1994-04-26 | 1995-08-01 | Syntex (U.S.A.) Inc. | Process for making 1-benzocycloalkyl-1,3-dihydroimidazole-2-thione derivatives |
| US7125904B2 (en) * | 2002-10-11 | 2006-10-24 | Portela & C.A., S.A. | Peripherally-selective inhibitors of dopamine-β-hydroxylase and method of their preparation |
| JP2010517998A (ja) * | 2007-02-01 | 2010-05-27 | バイアル−ポルテラ アンド シーエー,エス.エー. | 化合物 |
-
2007
- 2007-02-01 GB GBGB0701965.6A patent/GB0701965D0/en not_active Ceased
-
2008
- 2008-01-31 AU AU2008211846A patent/AU2008211846A1/en not_active Abandoned
- 2008-01-31 AR ARP080100396A patent/AR065108A1/es unknown
- 2008-01-31 CN CN200880003908A patent/CN101627032A/zh active Pending
- 2008-01-31 EP EP08712687A patent/EP2114926A1/en not_active Withdrawn
- 2008-01-31 US US12/525,007 patent/US20100113799A1/en not_active Abandoned
- 2008-01-31 KR KR1020097017870A patent/KR20090104898A/ko not_active Withdrawn
- 2008-01-31 MX MX2009008244A patent/MX2009008244A/es not_active Application Discontinuation
- 2008-01-31 BR BRPI0806402-4A patent/BRPI0806402A2/pt not_active IP Right Cessation
- 2008-01-31 JP JP2009548188A patent/JP2010517999A/ja active Pending
- 2008-01-31 WO PCT/PT2008/000005 patent/WO2008094055A1/en not_active Ceased
- 2008-01-31 CA CA002677203A patent/CA2677203A1/en not_active Abandoned
- 2008-01-31 RU RU2009132668/04A patent/RU2009132668A/ru not_active Application Discontinuation
-
2009
- 2009-07-30 IL IL200178A patent/IL200178A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB0701965D0 (en) | 2007-03-14 |
| AU2008211846A1 (en) | 2008-08-07 |
| AU2008211846A2 (en) | 2009-09-10 |
| WO2008094055A1 (en) | 2008-08-07 |
| CA2677203A1 (en) | 2008-08-07 |
| US20100113799A1 (en) | 2010-05-06 |
| MX2009008244A (es) | 2009-08-12 |
| BRPI0806402A2 (pt) | 2011-09-06 |
| KR20090104898A (ko) | 2009-10-06 |
| CN101627032A (zh) | 2010-01-13 |
| JP2010517999A (ja) | 2010-05-27 |
| EP2114926A1 (en) | 2009-11-11 |
| RU2009132668A (ru) | 2011-03-10 |
| IL200178A0 (en) | 2010-04-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |