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AR057885A1 - Acido 1-(1-(2- etoxietil) - 1- etil-7-(4- metilpiridin -2- ilamino)- 1h pirazolo (4,3-d) pirimidin -5- il) piperidina -4- carboxilico y las sales del mismo. composiciones farmaceuticas. - Google Patents

Acido 1-(1-(2- etoxietil) - 1- etil-7-(4- metilpiridin -2- ilamino)- 1h pirazolo (4,3-d) pirimidin -5- il) piperidina -4- carboxilico y las sales del mismo. composiciones farmaceuticas.

Info

Publication number
AR057885A1
AR057885A1 ARP060104894A ARP060104894A AR057885A1 AR 057885 A1 AR057885 A1 AR 057885A1 AR P060104894 A ARP060104894 A AR P060104894A AR P060104894 A ARP060104894 A AR P060104894A AR 057885 A1 AR057885 A1 AR 057885A1
Authority
AR
Argentina
Prior art keywords
etoxietil
methylpiridin
pirazolo
pirimidin
etil
Prior art date
Application number
ARP060104894A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of AR057885A1 publication Critical patent/AR057885A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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Abstract

Reivindicacion 1: Un compuesto, y las sales farmacéuticamente aceptables del compuesto que tiene la formula (1).
ARP060104894A 2005-11-10 2006-11-08 Acido 1-(1-(2- etoxietil) - 1- etil-7-(4- metilpiridin -2- ilamino)- 1h pirazolo (4,3-d) pirimidin -5- il) piperidina -4- carboxilico y las sales del mismo. composiciones farmaceuticas. AR057885A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73532005P 2005-11-10 2005-11-10

Publications (1)

Publication Number Publication Date
AR057885A1 true AR057885A1 (es) 2007-12-26

Family

ID=37685872

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060104894A AR057885A1 (es) 2005-11-10 2006-11-08 Acido 1-(1-(2- etoxietil) - 1- etil-7-(4- metilpiridin -2- ilamino)- 1h pirazolo (4,3-d) pirimidin -5- il) piperidina -4- carboxilico y las sales del mismo. composiciones farmaceuticas.

Country Status (29)

Country Link
US (2) US20090156618A1 (es)
EP (1) EP1948661B1 (es)
JP (1) JP4208959B1 (es)
KR (1) KR101012592B1 (es)
CN (1) CN101305007B (es)
AP (1) AP2008004437A0 (es)
AR (1) AR057885A1 (es)
AT (1) ATE435865T1 (es)
AU (1) AU2006313486B2 (es)
BR (1) BRPI0618284A2 (es)
CA (1) CA2629339C (es)
CR (1) CR9966A (es)
DE (1) DE602006007728D1 (es)
DK (1) DK1948661T3 (es)
DO (1) DOP2006000248A (es)
EA (1) EA200800920A1 (es)
EC (1) ECSP088441A (es)
ES (1) ES2326919T3 (es)
IL (1) IL190456A (es)
MA (1) MA29943B1 (es)
NL (1) NL2000291C2 (es)
NO (1) NO20082593L (es)
PE (1) PE20070764A1 (es)
RS (1) RS20080197A (es)
TN (1) TNSN08209A1 (es)
TW (1) TW200738723A (es)
UY (1) UY29909A1 (es)
WO (1) WO2007054778A1 (es)
ZA (1) ZA200803173B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2732628A1 (en) * 2008-08-01 2010-02-04 Biocryst Pharmaceuticals, Inc. Therapeutic agents
WO2010043633A1 (en) * 2008-10-15 2010-04-22 Palau Pharma, S. A. 2h-pyrazolo [4,3-d]pyrimidin-5-amine derivatives as h4 histamine receptor antagonists for the treatment of allergic, immunological and inflammatory diseases
CN102970965A (zh) * 2010-04-05 2013-03-13 Sk化学公司 含有pde5抑制剂的减少皮肤皱纹的合成物
CN103402542B (zh) * 2011-02-28 2017-05-03 独立行政法人国立循环器病研究中心 恶性肿瘤转移抑制用药物
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US20110059993A1 (en) 2011-03-10
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