AR056475A1 - Formulacion solida estable de sertinodl - Google Patents
Formulacion solida estable de sertinodlInfo
- Publication number
- AR056475A1 AR056475A1 ARP060103764A ARP060103764A AR056475A1 AR 056475 A1 AR056475 A1 AR 056475A1 AR P060103764 A ARP060103764 A AR P060103764A AR P060103764 A ARP060103764 A AR P060103764A AR 056475 A1 AR056475 A1 AR 056475A1
- Authority
- AR
- Argentina
- Prior art keywords
- sertinodl
- solid formulation
- stable solid
- sertindole
- pharmaceutical composition
- Prior art date
Links
- 238000009472 formulation Methods 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 239000007787 solid Substances 0.000 title 1
- GZKLJWGUPQBVJQ-UHFFFAOYSA-N sertindole Chemical compound C1=CC(F)=CC=C1N1C2=CC=C(Cl)C=C2C(C2CCN(CCN3C(NCC3)=O)CC2)=C1 GZKLJWGUPQBVJQ-UHFFFAOYSA-N 0.000 abstract 3
- 229960000652 sertindole Drugs 0.000 abstract 3
- UQSXHKLRYXJYBZ-UHFFFAOYSA-N Iron oxide Chemical compound [Fe]=O UQSXHKLRYXJYBZ-UHFFFAOYSA-N 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 239000003223 protective agent Substances 0.000 abstract 2
- 239000011247 coating layer Substances 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 230000005855 radiation Effects 0.000 abstract 1
- 201000000980 schizophrenia Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2813—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Inorganic Chemistry (AREA)
- Psychiatry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Composicion farmacéutica que comprende sertindol y un agente protector que absorbe radicacion con una longitud de onda por debajo de 400 nm. La presente se refiere también al uso de sertindol para la preparacion de una composicion farmacéutica que comprende sertindol y una capa de recubrimiento que comprende dicho agente protector, tal como oxido de hierro, para el tratamiento de esquizofrenia.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200501255 | 2005-09-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR056475A1 true AR056475A1 (es) | 2007-10-10 |
Family
ID=37697999
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP060103764A AR056475A1 (es) | 2005-09-08 | 2006-08-29 | Formulacion solida estable de sertinodl |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1924261A1 (es) |
| JP (1) | JP2009507051A (es) |
| KR (1) | KR20080042102A (es) |
| CN (1) | CN101257906A (es) |
| AR (1) | AR056475A1 (es) |
| AU (1) | AU2006322460A1 (es) |
| BR (1) | BRPI0615630A2 (es) |
| CA (1) | CA2621866A1 (es) |
| EA (1) | EA013167B1 (es) |
| IL (1) | IL189541A0 (es) |
| MX (1) | MX2008002290A (es) |
| NO (1) | NO20081721L (es) |
| NZ (1) | NZ565330A (es) |
| TW (1) | TW200738239A (es) |
| UA (1) | UA97349C2 (es) |
| WO (1) | WO2007065448A1 (es) |
| ZA (1) | ZA200801169B (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI320783B (en) | 2005-04-14 | 2010-02-21 | Otsuka Pharma Co Ltd | Heterocyclic compound |
| CN106344533A (zh) * | 2009-01-29 | 2017-01-25 | 大日本住友制药株式会社 | 具有内核的口腔崩解片剂 |
| FR2943061B1 (fr) * | 2009-03-13 | 2011-02-25 | Rhodia Operations | Composes organophosphores, systemes catalytiques comprenant ces composes et procede d'hydrocyanation ou d'hydroformylation utilisant ces systemes catalytiques |
| US8883823B2 (en) | 2012-07-16 | 2014-11-11 | Fibrogen, Inc. | Crystalline forms of a prolyl hydroxylase inhibitor |
| JP6491093B2 (ja) | 2012-07-16 | 2019-03-27 | フィブロジェン インコーポレイテッド | プロリルヒドロキシラーゼ阻害剤の結晶形態 |
| DK3003284T3 (da) | 2013-06-06 | 2020-03-30 | Fibrogen Inc | Farmaceutiske formuleringer af en hif-hydroxylase-inhibitor |
| CN105636585B (zh) | 2013-11-19 | 2020-02-07 | 西佳技术公司 | 微粉化特考韦瑞一水化物的再水化 |
| JP2018172361A (ja) * | 2016-10-14 | 2018-11-08 | 大原薬品工業株式会社 | 光安定性を改善した、デュロキセチンを含有する固形製剤 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH04346929A (ja) * | 1991-05-22 | 1992-12-02 | Takada Seiyaku Kk | 光に安定なメシル酸ブロモクリプチン製剤 |
| JP2000507544A (ja) * | 1996-03-25 | 2000-06-20 | イーライ・リリー・アンド・カンパニー | 痛みの治療方法 |
| ZA973433B (en) * | 1996-04-24 | 1997-12-10 | Shionogi & Co | A sertindole-containing preparation and a method for producing the same. |
| ZA977967B (en) * | 1996-09-23 | 1999-03-04 | Lilly Co Eli | Combination therapy for treatment of psychoses |
-
2006
- 2006-06-09 UA UAA200803569A patent/UA97349C2/uk unknown
- 2006-08-17 TW TW095130202A patent/TW200738239A/zh unknown
- 2006-08-29 AR ARP060103764A patent/AR056475A1/es not_active Application Discontinuation
- 2006-09-06 AU AU2006322460A patent/AU2006322460A1/en not_active Abandoned
- 2006-09-06 NZ NZ565330A patent/NZ565330A/en not_active IP Right Cessation
- 2006-09-06 ZA ZA200801169A patent/ZA200801169B/xx unknown
- 2006-09-06 CN CNA2006800323410A patent/CN101257906A/zh active Pending
- 2006-09-06 JP JP2008529472A patent/JP2009507051A/ja not_active Withdrawn
- 2006-09-06 WO PCT/DK2006/050038 patent/WO2007065448A1/en not_active Ceased
- 2006-09-06 EP EP06846966A patent/EP1924261A1/en not_active Withdrawn
- 2006-09-06 BR BRPI0615630A patent/BRPI0615630A2/pt not_active IP Right Cessation
- 2006-09-06 MX MX2008002290A patent/MX2008002290A/es not_active Application Discontinuation
- 2006-09-06 EA EA200800774A patent/EA013167B1/ru not_active IP Right Cessation
- 2006-09-06 CA CA002621866A patent/CA2621866A1/en not_active Abandoned
- 2006-09-06 KR KR1020087004910A patent/KR20080042102A/ko not_active Withdrawn
-
2008
- 2008-02-14 IL IL189541A patent/IL189541A0/en unknown
- 2008-04-08 NO NO20081721A patent/NO20081721L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20080042102A (ko) | 2008-05-14 |
| MX2008002290A (es) | 2008-03-14 |
| BRPI0615630A2 (pt) | 2016-11-16 |
| WO2007065448A1 (en) | 2007-06-14 |
| IL189541A0 (en) | 2008-08-07 |
| CA2621866A1 (en) | 2007-06-14 |
| EA200800774A1 (ru) | 2008-06-30 |
| EA013167B1 (ru) | 2010-02-26 |
| NO20081721L (no) | 2008-04-08 |
| EP1924261A1 (en) | 2008-05-28 |
| AU2006322460A1 (en) | 2007-06-14 |
| TW200738239A (en) | 2007-10-16 |
| JP2009507051A (ja) | 2009-02-19 |
| NZ565330A (en) | 2011-06-30 |
| CN101257906A (zh) | 2008-09-03 |
| ZA200801169B (en) | 2010-07-28 |
| UA97349C2 (uk) | 2012-02-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |