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AR055101A1 - 8-(3-amino-piperidin-1-il)-.xantinas, su preparacion y su uso como medicamentos - Google Patents

8-(3-amino-piperidin-1-il)-.xantinas, su preparacion y su uso como medicamentos

Info

Publication number
AR055101A1
AR055101A1 ARP060103275A ARP060103275A AR055101A1 AR 055101 A1 AR055101 A1 AR 055101A1 AR P060103275 A ARP060103275 A AR P060103275A AR P060103275 A ARP060103275 A AR P060103275A AR 055101 A1 AR055101 A1 AR 055101A1
Authority
AR
Argentina
Prior art keywords
piperidin
amino
xantinas
medications
preparation
Prior art date
Application number
ARP060103275A
Other languages
English (en)
Inventor
Waldemar Pfrengle
Peter Sieger
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37102454&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR055101(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of AR055101A1 publication Critical patent/AR055101A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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  • Cardiology (AREA)
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  • Hospice & Palliative Care (AREA)
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Abstract

Se refiere a 8-[3-amino-piperidin-1-il]-xantinas y sus sales fisiologicamente tolerables, en especial a sus hidrocloruros.
ARP060103275A 2005-07-30 2006-07-28 8-(3-amino-piperidin-1-il)-.xantinas, su preparacion y su uso como medicamentos AR055101A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102005035891A DE102005035891A1 (de) 2005-07-30 2005-07-30 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel

Publications (1)

Publication Number Publication Date
AR055101A1 true AR055101A1 (es) 2007-08-08

Family

ID=37102454

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060103275A AR055101A1 (es) 2005-07-30 2006-07-28 8-(3-amino-piperidin-1-il)-.xantinas, su preparacion y su uso como medicamentos

Country Status (32)

Country Link
US (2) US8106060B2 (es)
EP (2) EP2540724B1 (es)
JP (2) JP5145224B2 (es)
KR (1) KR101446692B1 (es)
CN (2) CN101233133B (es)
AR (1) AR055101A1 (es)
BR (1) BRPI0614700B8 (es)
CA (1) CA2617090C (es)
CY (1) CY1114563T1 (es)
DE (1) DE102005035891A1 (es)
DK (1) DK1912990T3 (es)
EA (1) EA013411B1 (es)
EC (1) ECSP088148A (es)
ES (1) ES2428368T3 (es)
HR (1) HRP20130868T1 (es)
IL (1) IL189099A0 (es)
ME (1) ME01593B (es)
MX (1) MX2008000932A (es)
MY (1) MY147274A (es)
NO (1) NO20076510L (es)
NZ (1) NZ566187A (es)
PE (1) PE20070219A1 (es)
PL (1) PL1912990T3 (es)
PT (1) PT1912990E (es)
RS (1) RS52836B (es)
SG (1) SG164390A1 (es)
SI (1) SI1912990T1 (es)
TW (1) TWI393720B (es)
UA (1) UA96577C2 (es)
UY (1) UY29700A1 (es)
WO (1) WO2007014886A1 (es)
ZA (1) ZA200711024B (es)

Families Citing this family (62)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EE05735B1 (et) * 2001-02-24 2015-01-15 Boehringer Ingelheim Pharma Gmbh & Co. Kg Ksantiini derivaadid, nende valmistamine ja kasutamine ravimina
US7074923B2 (en) * 2002-05-31 2006-07-11 Schering Corporation Process for preparing xanthine phosphodiesterase V inhibitors and precursors thereof
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7569574B2 (en) 2002-08-22 2009-08-04 Boehringer Ingelheim Pharma Gmbh & Co. Kg Purine derivatives, the preparation thereof and their use as pharmaceutical compositions
US7495005B2 (en) * 2002-08-22 2009-02-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, their preparation and their use in pharmaceutical compositions
US7482337B2 (en) * 2002-11-08 2009-01-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions
DE10254304A1 (de) * 2002-11-21 2004-06-03 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Xanthinderivate, deren Herstellung und deren Verwendung als Arzneimittel
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