AR041747A1 - Ciclopropil-tienil-carboxamida y su uso como funguicida - Google Patents
Ciclopropil-tienil-carboxamida y su uso como funguicidaInfo
- Publication number
- AR041747A1 AR041747A1 ARP030104010A ARP030104010A AR041747A1 AR 041747 A1 AR041747 A1 AR 041747A1 AR P030104010 A ARP030104010 A AR P030104010A AR P030104010 A ARP030104010 A AR P030104010A AR 041747 A1 AR041747 A1 AR 041747A1
- Authority
- AR
- Argentina
- Prior art keywords
- optionally substituted
- hydrogen
- compounds
- preparation
- alkyl
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 4
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 239000001257 hydrogen Substances 0.000 abstract 4
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 4
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 abstract 2
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 2
- 239000004480 active ingredient Substances 0.000 abstract 2
- 125000002947 alkylene group Chemical group 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- 239000000543 intermediate Substances 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 abstract 1
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 1
- QWENRTYMTSOGBR-UHFFFAOYSA-N 1H-1,2,3-Triazole Chemical compound C=1C=NNN=1 QWENRTYMTSOGBR-UHFFFAOYSA-N 0.000 abstract 1
- 125000002373 5 membered heterocyclic group Chemical group 0.000 abstract 1
- 125000004070 6 membered heterocyclic group Chemical group 0.000 abstract 1
- 241000233866 Fungi Species 0.000 abstract 1
- 206010061217 Infestation Diseases 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 239000003905 agrochemical Substances 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 230000000855 fungicidal effect Effects 0.000 abstract 1
- 239000000417 fungicide Substances 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 238000003898 horticulture Methods 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 244000005700 microbiome Species 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 230000003032 phytopathogenic effect Effects 0.000 abstract 1
- 125000005017 substituted alkenyl group Chemical group 0.000 abstract 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 1
- 125000004426 substituted alkynyl group Chemical group 0.000 abstract 1
- 125000005346 substituted cycloalkyl group Chemical group 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 239000011593 sulfur Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/36—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D411/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Un compuesto activo como fungicida de la fórmula (1): donde X es (X1), (X2) o (X3); Het es un anillo heterocíclico de 5 o 6 miembros que contiene entre uno y tres heteroátomos, cada uno seleccionado en forma independiente entre oxígeno, nitrógeno y azufre, con la condición de que el anillo no sea 1,2,3-triazol, donde el anillo está sustituido con los grupos R4, R5 y R6; R1 y R2 son cada uno, en forma independiente, hidrógeno, halo o metilo; R3 es C2-12 alquilo opcionalmente sustituido, C2-12 alquenilo opcionalmente sustituido, C2-12 alquinilo opcionalmente sustituido C3-12 cicloalquilo opcionalmente sustituido, fenilo opcionalmente sustituido o heterociclilo opcionalmente sustituido; R4, R5 y R6 se seleccionan, cada uno en forma independiente, entre hidrógeno, halo, ciano, nitro, C1-4 alquilo, C1-4 haloalquilo, C1-4 alcoxi(C1-4)alquileno y C1-4 haloalcoxi(C1-4)alquileno, con la condición de que al menos uno de R4, R5 y R6 no sea hidrógeno; y R7 y R8 son cada uno, en forma independiente, hidrógeno, halógeno, C1-4 alquilo o C1-4 haloalquilo; también hace referencia a la preparación de estos compuestos, a intermediarios utilizados en la preparación de estos compuestos, a la preparación de intermediarios, a composiciones agroquímicas que comprenden al menos uno de los compuestos como ingrediente activo y al uso de los ingredientes activos o composiciones de agricultura u horticultura con el fin de controlar o prevenir la infestación de plantas por parte de microorganismos fitopatogénicos, preferentemente hongos.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0225554.5A GB0225554D0 (en) | 2002-11-01 | 2002-11-01 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR041747A1 true AR041747A1 (es) | 2005-05-26 |
Family
ID=9947074
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP030104010A AR041747A1 (es) | 2002-11-01 | 2003-10-31 | Ciclopropil-tienil-carboxamida y su uso como funguicida |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US7312179B2 (es) |
| EP (1) | EP1556377B1 (es) |
| JP (1) | JP4673061B2 (es) |
| KR (1) | KR101000731B1 (es) |
| CN (1) | CN100526310C (es) |
| AR (1) | AR041747A1 (es) |
| AT (1) | ATE331714T1 (es) |
| AU (1) | AU2003286140A1 (es) |
| BR (1) | BR0315857A (es) |
| CA (1) | CA2501739C (es) |
| CO (1) | CO5550397A2 (es) |
| DE (1) | DE60306540T2 (es) |
| DK (1) | DK1556377T3 (es) |
| EC (1) | ECSP055770A (es) |
| ES (1) | ES2266881T3 (es) |
| GB (1) | GB0225554D0 (es) |
| GT (1) | GT200300236A (es) |
| MX (1) | MXPA05004463A (es) |
| PT (1) | PT1556377E (es) |
| RU (1) | RU2005116974A (es) |
| TW (1) | TW200412848A (es) |
| WO (1) | WO2004039799A1 (es) |
| ZA (1) | ZA200502644B (es) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0418047D0 (en) | 2004-08-12 | 2004-09-15 | Syngenta Participations Ag | Fungicidal compositions |
| DE102005025989A1 (de) * | 2005-06-07 | 2007-01-11 | Bayer Cropscience Ag | Carboxamide |
| EP1956909A1 (en) * | 2005-11-15 | 2008-08-20 | Syngeta Participations AG | Microbiocides |
| US7820830B2 (en) | 2005-11-15 | 2010-10-26 | Syngenta Crop Protection, Inc. | Process for the production of carboxanilides |
| DK2563776T3 (en) | 2010-04-27 | 2016-09-19 | Calcimedica Inc | Relations that modulate intracellular calcium |
| US10703722B2 (en) | 2010-04-27 | 2020-07-07 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| JP2013525448A (ja) | 2010-04-27 | 2013-06-20 | カルシメディカ，インク． | 細胞内カルシウムを調節する化合物 |
| WO2012027710A2 (en) * | 2010-08-27 | 2012-03-01 | Calcimedica Inc. | Compounds that modulate intracellular calcium |
| US20130231303A1 (en) * | 2010-11-15 | 2013-09-05 | Bayer Intellectual Property Gmbh | 5-halogenopyrazole(thio)carboxamides |
| WO2012170931A2 (en) | 2011-06-10 | 2012-12-13 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| WO2013059677A1 (en) | 2011-10-19 | 2013-04-25 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| WO2014059333A1 (en) | 2012-10-12 | 2014-04-17 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| TWI835179B (zh) | 2015-02-27 | 2024-03-11 | 美商鈣系醫藥公司 | 胰腺炎治療 |
| DK3331525T3 (da) | 2015-08-07 | 2020-12-14 | Calcimedica Inc | Anvendelse af CRAC-kanal-inhibitorer til behandling af slagtilfælde og traumatisk hjerneskade |
| CN106977457A (zh) * | 2016-12-22 | 2017-07-25 | 浙江海正化工股份有限公司 | 一种3‑二氟甲基‑1‑甲基‑吡唑‑4‑甲酸及其合成方法 |
| CR20200641A (es) * | 2018-07-05 | 2021-02-16 | Bayer Ag | Tiofenocarboxamidas sustituidas y analogos como agentes antibacterianos |
| EP4243813A4 (en) | 2020-11-13 | 2024-07-17 | Calcimedica, Inc. | IMPROVED SYNTHESIS OF CRAC CHANNEL INHIBITORS |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2385721A1 (fr) * | 1977-03-31 | 1978-10-27 | Hexachimie | Cyclopropyl-6 dihydro-1,3 methyl-1 phenyl-5 oxo-2 2 h-thieno (2,3-e) diazepine, son procede de preparation et son application en therapeutique |
| GB2126587A (en) * | 1982-09-13 | 1984-03-28 | Sandoz Ltd | Fungicidal thiophene derivatives |
| GB2192631A (en) * | 1986-07-16 | 1988-01-20 | Ici Plc | Fungicidal heterocyclic tertiary amine compounds containing a cyclopropane ring |
| GB8617378D0 (en) * | 1986-07-16 | 1986-08-20 | Ici Plc | Tertiary amine compounds |
| DE69618370T2 (de) | 1995-04-11 | 2002-09-26 | Mitsui Chemicals, Inc. | Substituierte Thiophenderivate und diese als aktiver Bestandteil enthaltenden Fungizide für Land- und Gartenbauwirtschaft |
| GB9817548D0 (en) * | 1998-08-12 | 1998-10-07 | Novartis Ag | Organic compounds |
| GB9930750D0 (en) * | 1999-12-29 | 2000-02-16 | Novartis Ag | Organic compounds |
| HK1079785B (zh) * | 2002-03-05 | 2007-08-10 | 辛根塔参与股份公司 | 邻环丙基-n-甲酰苯胺及其作为杀菌剂的用途 |
| ATE516275T1 (de) | 2002-08-22 | 2011-07-15 | Syngenta Participations Ag | Microbiozide (z.b. fungizide) 1,2,3- triazolderivate |
-
2002
- 2002-11-01 GB GBGB0225554.5A patent/GB0225554D0/en not_active Ceased
-
2003
- 2003-10-24 DK DK03776869T patent/DK1556377T3/da active
- 2003-10-24 RU RU2005116974/04A patent/RU2005116974A/ru not_active Application Discontinuation
- 2003-10-24 MX MXPA05004463A patent/MXPA05004463A/es active IP Right Grant
- 2003-10-24 KR KR1020057007633A patent/KR101000731B1/ko not_active Expired - Fee Related
- 2003-10-24 AT AT03776869T patent/ATE331714T1/de not_active IP Right Cessation
- 2003-10-24 CN CNB2003801021700A patent/CN100526310C/zh not_active Expired - Fee Related
- 2003-10-24 BR BR0315857-8A patent/BR0315857A/pt not_active Application Discontinuation
- 2003-10-24 EP EP03776869A patent/EP1556377B1/en not_active Expired - Lifetime
- 2003-10-24 JP JP2004547558A patent/JP4673061B2/ja not_active Expired - Fee Related
- 2003-10-24 AU AU2003286140A patent/AU2003286140A1/en not_active Abandoned
- 2003-10-24 ES ES03776869T patent/ES2266881T3/es not_active Expired - Lifetime
- 2003-10-24 CA CA2501739A patent/CA2501739C/en not_active Expired - Fee Related
- 2003-10-24 DE DE60306540T patent/DE60306540T2/de not_active Expired - Lifetime
- 2003-10-24 PT PT03776869T patent/PT1556377E/pt unknown
- 2003-10-24 US US10/532,847 patent/US7312179B2/en not_active Expired - Fee Related
- 2003-10-24 WO PCT/EP2003/011805 patent/WO2004039799A1/en not_active Ceased
- 2003-10-27 TW TW092129757A patent/TW200412848A/zh unknown
- 2003-10-30 GT GT200300236A patent/GT200300236A/es unknown
- 2003-10-31 AR ARP030104010A patent/AR041747A1/es unknown
-
2005
- 2005-04-01 ZA ZA200502644A patent/ZA200502644B/en unknown
- 2005-04-29 EC EC2005005770A patent/ECSP055770A/es unknown
- 2005-04-29 CO CO05040972A patent/CO5550397A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004039799A1 (en) | 2004-05-13 |
| DE60306540T2 (de) | 2007-06-28 |
| US7312179B2 (en) | 2007-12-25 |
| MXPA05004463A (es) | 2005-07-26 |
| DE60306540D1 (en) | 2006-08-10 |
| US20060030567A1 (en) | 2006-02-09 |
| DK1556377T3 (da) | 2006-10-23 |
| ATE331714T1 (de) | 2006-07-15 |
| JP4673061B2 (ja) | 2011-04-20 |
| CN1708496A (zh) | 2005-12-14 |
| GB0225554D0 (en) | 2002-12-11 |
| BR0315857A (pt) | 2005-09-20 |
| GT200300236A (es) | 2004-06-23 |
| ECSP055770A (es) | 2005-08-11 |
| AU2003286140A1 (en) | 2004-05-25 |
| CA2501739C (en) | 2011-04-12 |
| ES2266881T3 (es) | 2007-03-01 |
| TW200412848A (en) | 2004-08-01 |
| CO5550397A2 (es) | 2005-08-31 |
| EP1556377B1 (en) | 2006-06-28 |
| ZA200502644B (en) | 2005-11-23 |
| CA2501739A1 (en) | 2004-05-13 |
| RU2005116974A (ru) | 2006-03-27 |
| JP2006508089A (ja) | 2006-03-09 |
| KR101000731B1 (ko) | 2010-12-14 |
| KR20050071648A (ko) | 2005-07-07 |
| PT1556377E (pt) | 2006-10-31 |
| CN100526310C (zh) | 2009-08-12 |
| EP1556377A1 (en) | 2005-07-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |