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AR038143A1 - Agonistas del receptor 2 del factor liberador de la corticotropina - Google Patents

Agonistas del receptor 2 del factor liberador de la corticotropina

Info

Publication number
AR038143A1
AR038143A1 ARP030100100A ARP030100100A AR038143A1 AR 038143 A1 AR038143 A1 AR 038143A1 AR P030100100 A ARP030100100 A AR P030100100A AR P030100100 A ARP030100100 A AR P030100100A AR 038143 A1 AR038143 A1 AR 038143A1
Authority
AR
Argentina
Prior art keywords
peptide
corticotropine
liberating
agonists
crf2r
Prior art date
Application number
ARP030100100A
Other languages
English (en)
Inventor
Robert Joseph Isfort
Wieslaw Adam Mazur
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of AR038143A1 publication Critical patent/AR038143A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/57509Corticotropin releasing factor [CRF] (Urotensin)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/04Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Neurology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

Abstract

Un péptido no nativo que comprende la secuencia: ZGPPISIDLPX12X13LLRKX18IEIEKQEKEKQQAX32X33NAX36X37X37LX39X40X41, en donde: X12 se selecciona de F, Y, L, I, y T; X13 se selecciona de Q, W, y Y; X18 se selecciona de V y M; X32 se selecciona de T y A; X33 se selecciona de N y T; X36 se selecciona de R y L; X37 se selecciona de L y I; X39 se selecciona de D y A; X40 se selecciona de T y R; X41 se selecciona de I y V; y variantes de éstos. Las correspondientes definiciones y secuencias de dichos sustituyentes se incluyen en la Memoria. Uso para preparar una composición farmacéutica útil para evitar o tratar un trastorno modulado por CRF2R que comprende una cantidad segura y eficaz de dicho péptido. Ácido nucleico aislado que codifica dicho péptido. Anticuerpo aislado específico para dicho péptido. Composición farmacéutica que comprende dicho péptido y un portador farmacéuticamente aceptable. Conjunto o Kit para evitar o tratar un trastorno modulado por CRF2R que comprende dicho péptido en forma de dosis unitaria e instrucciones de uso.
ARP030100100A 2002-01-16 2003-01-15 Agonistas del receptor 2 del factor liberador de la corticotropina AR038143A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US34911702P 2002-01-16 2002-01-16
US37633702P 2002-04-29 2002-04-29
US38889502P 2002-06-14 2002-06-14
US41198802P 2002-09-19 2002-09-19

Publications (1)

Publication Number Publication Date
AR038143A1 true AR038143A1 (es) 2004-12-29

Family

ID=27617822

Family Applications (3)

Application Number Title Priority Date Filing Date
ARP030100100A AR038143A1 (es) 2002-01-16 2003-01-15 Agonistas del receptor 2 del factor liberador de la corticotropina
ARP030100101A AR038144A1 (es) 2002-01-16 2003-01-15 Agonistas del receptor 2 del factor liberador de la corticotropina
ARP030100099A AR038142A1 (es) 2002-01-16 2003-01-15 Agonistas del receptor 2 del factor liberador de la corticotropina

Family Applications After (2)

Application Number Title Priority Date Filing Date
ARP030100101A AR038144A1 (es) 2002-01-16 2003-01-15 Agonistas del receptor 2 del factor liberador de la corticotropina
ARP030100099A AR038142A1 (es) 2002-01-16 2003-01-15 Agonistas del receptor 2 del factor liberador de la corticotropina

Country Status (29)

Country Link
US (7) US6936585B2 (es)
EP (4) EP1724283B1 (es)
JP (3) JP4508648B2 (es)
KR (3) KR100758858B1 (es)
CN (3) CN100475844C (es)
AR (3) AR038143A1 (es)
AT (4) ATE362488T1 (es)
AU (2) AU2003205197B2 (es)
BR (3) BR0306878A (es)
CA (3) CA2470743C (es)
CY (1) CY1106133T1 (es)
DE (4) DE60318547T2 (es)
DK (2) DK1465923T3 (es)
ES (4) ES2299701T3 (es)
IL (5) IL162529A0 (es)
MA (3) MA27592A1 (es)
MX (3) MXPA04006883A (es)
MY (1) MY140306A (es)
NO (3) NO20043366L (es)
NZ (3) NZ533600A (es)
PE (3) PE20030849A1 (es)
PL (3) PL373139A1 (es)
PT (2) PT1465923E (es)
RU (1) RU2294333C2 (es)
SA (3) SA03230564A (es)
SI (1) SI1465921T1 (es)
TW (3) TW200302276A (es)
WO (3) WO2003062268A2 (es)
ZA (1) ZA200404995B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002024732A2 (en) * 2000-09-22 2002-03-28 Max-Planck-Gesellschaft Zur Förderung Der Wissenschaften Methods for improving the antagonistic/agonistic properties of peptidic antagonists/agonists of the corticotropin-releasing factor receptor (crfr)
US6936585B2 (en) * 2002-01-16 2005-08-30 The Procter & Gamble Company Corticotropin releasing factor 2 receptor agonists
WO2005103690A2 (en) * 2004-04-24 2005-11-03 Bayer Healthcare Ag Diagnostics and therapeutics for diseases associated with corticotropin releasing hormone receptor 2 (crhr2)
AU2006235045A1 (en) * 2005-03-30 2006-10-19 J. Craig Venter Institute, Inc. Haemophilus influenzae type b
WO2007090087A2 (en) * 2006-01-27 2007-08-09 Research Development Foundation Use of corticotropin releasing factor receptor-2 inhibitors for treating insulin-related diseases
WO2009033773A2 (en) * 2007-09-11 2009-03-19 Mondobiotech Laboratories Ag Use endothelin 2, alone or combined with a nonapeptide, a peptide as a therapeutic agent
AU2008297874A1 (en) * 2007-09-11 2009-03-19 Mondobiotech Laboratories Ag Use of secretin and optionally urodilatin as therapeutic agents
WO2009046874A1 (en) * 2007-09-11 2009-04-16 Mondobiotech Laboratories Ag Therapeutic combination of trh-potentiating peptide and stresscopin
ES2723098T3 (es) * 2008-11-04 2019-08-21 Janssen Pharmaceutica Nv Agonistas del péptido CRHR2 y usos de los mismos
EP2206726A1 (en) * 2009-01-08 2010-07-14 Universite Joseph Fourier Non-invasive tools for detecting vulnerable atherosclerotic plaques
CN102711801A (zh) * 2009-11-04 2012-10-03 詹森药业有限公司 用顶压素样肽治疗心力衰竭的方法
US9314506B2 (en) 2011-10-24 2016-04-19 Research Development Foundation Methods for increasing insulin secretion by co-stimulation of corticotropin-releasing factor receptors
CN104220098B (zh) * 2012-02-14 2018-04-10 加利福尼亚大学董事会 用于心血管疾病和其它病况的旁分泌基因的全身性递送和受调节的表达
JOP20170153A1 (ar) * 2016-07-15 2019-01-30 Lilly Co Eli نظائر urocortin-2 جديدة معدلة بحمض دهني لعلاج داء السكري وأمراض الكلى المزمنة
EP3528622A4 (en) * 2016-10-20 2020-08-05 Cortene Inc. METHODS OF TREATING ILLNESSES DUE TO IMPROPER STRESS RESPONSE
CN110755434B (zh) * 2018-07-27 2022-03-15 中国医学科学院药物研究所 化合物palosuran防治骨骼肌萎缩等疾病的用途
WO2025184558A1 (en) * 2024-02-28 2025-09-04 Caradon Therapeutics, Inc. Modified urocortin 3
WO2025222010A1 (en) * 2024-04-19 2025-10-23 Neurocrine Biosciences, Inc. Corticotropin releasing factor receptor 2 (crfr2) agonists
WO2025230248A1 (ko) * 2024-04-30 2025-11-06 한미약품 주식회사 Crf2 수용체 작용제와 그 아실화 결합체의 용도

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5235036A (en) * 1991-05-31 1993-08-10 The Salk Institute For Biological Studies Crf analogs
EP0860501A3 (en) 1994-06-14 1999-05-19 Neurocrine Biosciences, Inc. Corticotropin-releasing factor2 receptors
US5786203A (en) * 1994-06-14 1998-07-28 Neurocrine Biosciences, Inc. Isolated nucleic acid encoding corticotropin-releasing factor2 receptors
US5824771A (en) * 1994-12-12 1998-10-20 The Salk Institute For Biological Studies Cyclic CRF agonists
US5663292A (en) * 1994-12-12 1997-09-02 The Salk Institute For Biological Studies Cyclic CRF analogs
US5660824A (en) 1995-05-24 1997-08-26 Grabstein; Kenneth H. Muscle trophic factor
AU6277796A (en) 1995-06-13 1997-01-15 Salk Institute For Biological Studies, The Urocortin peptides
US5869450A (en) 1996-03-06 1999-02-09 The Regents Of The University Of California Anti-inflammatory compositions and method with corticotropin-releasing factor analogs
US6838274B2 (en) 2000-08-04 2005-01-04 Research Development Foundation Urocortin proteins and uses thereof
WO2002024732A2 (en) * 2000-09-22 2002-03-28 Max-Planck-Gesellschaft Zur Förderung Der Wissenschaften Methods for improving the antagonistic/agonistic properties of peptidic antagonists/agonists of the corticotropin-releasing factor receptor (crfr)
US20020082409A1 (en) 2000-10-26 2002-06-27 Hsu Sheau Yu Stresscopins and their uses
US6670140B2 (en) * 2001-03-06 2003-12-30 The Procter & Gamble Company Methods for identifying compounds for regulating muscle mass or function using corticotropin releasing factor receptors
US6936585B2 (en) * 2002-01-16 2005-08-30 The Procter & Gamble Company Corticotropin releasing factor 2 receptor agonists

Also Published As

Publication number Publication date
US7462597B2 (en) 2008-12-09
IL162529A0 (en) 2005-11-20
PT1465923E (pt) 2007-08-06
JP2005525101A (ja) 2005-08-25
TWI300442B (en) 2008-09-01
CA2470731A1 (en) 2003-07-31
IL197774A0 (en) 2009-12-24
ATE362488T1 (de) 2007-06-15
NZ533598A (en) 2007-03-30
EP1465921B1 (en) 2006-07-26
CA2470743C (en) 2011-12-13
MA27590A1 (fr) 2005-11-01
US6936585B2 (en) 2005-08-30
NO20043396L (no) 2004-10-06
AR038144A1 (es) 2004-12-29
US20060025339A1 (en) 2006-02-02
CN1617887A (zh) 2005-05-18
ES2269976T3 (es) 2007-04-01
KR100758858B1 (ko) 2007-09-14
IL162530A0 (en) 2005-11-20
HK1078095A1 (zh) 2006-03-03
DE60307044D1 (de) 2006-09-07
RU2004124847A (ru) 2005-04-20
WO2003062269A3 (en) 2003-11-06
DK1465921T3 (da) 2006-11-27
DE60307044T2 (de) 2007-02-15
NO20043371L (no) 2004-10-06
EP1724283A2 (en) 2006-11-22
WO2003062269A2 (en) 2003-07-31
CN1617886A (zh) 2005-05-18
JP4508649B2 (ja) 2010-07-21
EP1465921A2 (en) 2004-10-13
DK1465923T3 (da) 2007-07-02
CN100475844C (zh) 2009-04-08
DE60313845T2 (de) 2008-01-31
US7192923B2 (en) 2007-03-20
PL373139A1 (en) 2005-08-22
BR0306826A (pt) 2005-09-06
JP4508648B2 (ja) 2010-07-21
PL371364A1 (en) 2005-06-13
US7632933B2 (en) 2009-12-15
SA03230564A (ar) 2005-12-03
EP1465923A1 (en) 2004-10-13
KR100758857B1 (ko) 2007-09-14
CN100391972C (zh) 2008-06-04
ES2299701T3 (es) 2008-06-01
PE20030974A1 (es) 2003-12-26
ES2287484T3 (es) 2007-12-16
KR100735586B1 (ko) 2007-07-04
JP2005522191A (ja) 2005-07-28
MA27591A1 (fr) 2005-11-01
WO2003062277A1 (en) 2003-07-31
EP1724283A3 (en) 2007-04-11
EP1724283B1 (en) 2008-06-18
MXPA04006884A (es) 2004-12-06
PL373529A1 (en) 2005-09-05
JP4489434B2 (ja) 2010-06-23
MXPA04006885A (es) 2004-12-06
BR0306838A (pt) 2005-04-05
US20030148956A1 (en) 2003-08-07
US7897731B2 (en) 2011-03-01
DE60318547D1 (de) 2008-02-21
MY140306A (en) 2009-12-31
ES2309909T3 (es) 2008-12-16
CA2470743A1 (en) 2003-07-31
ZA200404995B (en) 2005-06-29
RU2294333C2 (ru) 2007-02-27
SA03230564B1 (ar) 2006-10-31
DE60313845D1 (de) 2007-06-28
US20100197579A1 (en) 2010-08-05
WO2003062268A3 (en) 2003-11-27
WO2003062268A2 (en) 2003-07-31
CY1106133T1 (el) 2011-06-08
NZ533599A (en) 2007-03-30
ATE334147T1 (de) 2006-08-15
NZ533600A (en) 2007-02-23
ATE383372T1 (de) 2008-01-15
CA2470656C (en) 2011-06-28
DE60318547T2 (de) 2008-12-24
US20080004435A1 (en) 2008-01-03
EP1465922B1 (en) 2008-01-09
PT1465921E (pt) 2006-12-29
PE20030849A1 (es) 2003-12-01
MA27592A1 (fr) 2005-11-01
AR038142A1 (es) 2004-12-29
BR0306878A (pt) 2004-10-26
IL196384A0 (en) 2011-07-31
KR20040082392A (ko) 2004-09-24
KR20040082390A (ko) 2004-09-24
EP1465922A2 (en) 2004-10-13
IL162431A0 (en) 2005-11-20
US7192924B2 (en) 2007-03-20
US20030148958A1 (en) 2003-08-07
NO20043366L (no) 2004-10-06
US7608701B2 (en) 2009-10-27
PE20030747A1 (es) 2003-10-23
SA03230565A (ar) 2005-12-03
AU2003205197B2 (en) 2006-03-02
US20090124793A1 (en) 2009-05-14
MXPA04006883A (es) 2004-12-06
CA2470731C (en) 2011-06-21
DE60321730D1 (de) 2008-07-31
US20030148957A1 (en) 2003-08-07
CN1617885A (zh) 2005-05-18
SA03230565B1 (ar) 2006-10-31
CA2470656A1 (en) 2003-07-31
TW200302277A (en) 2003-08-01
TW200302278A (en) 2003-08-01
KR20040082389A (ko) 2004-09-24
AU2003237419B2 (en) 2006-04-13
SI1465921T1 (sl) 2006-10-31
TW200302276A (en) 2003-08-01
ATE398632T1 (de) 2008-07-15
EP1465923B1 (en) 2007-05-16
JP2005521387A (ja) 2005-07-21

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