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AR027038A1 - Metodo y composicion para el tratamiento del dolor - Google Patents

Metodo y composicion para el tratamiento del dolor

Info

Publication number
AR027038A1
AR027038A1 ARP000106798A ARP000106798A AR027038A1 AR 027038 A1 AR027038 A1 AR 027038A1 AR P000106798 A ARP000106798 A AR P000106798A AR P000106798 A ARP000106798 A AR P000106798A AR 027038 A1 AR027038 A1 AR 027038A1
Authority
AR
Argentina
Prior art keywords
composition
pain
pain treatment
mitigate
compound according
Prior art date
Application number
ARP000106798A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of AR027038A1 publication Critical patent/AR027038A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • A61K31/5025Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • A61K31/503Pyridazines; Hydrogenated pyridazines spiro-condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541Non-condensed thiazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se describe un método para el tratamiento del dolor que comprende la administracion de una cantidad efectiva para mitigar el dolor de cualquier compuestode acuerdo con el diagrama estructural (1) en el cual A, D y R1 son como se los definiera en la m emoria. También se describen composiciones farmacéuticas quecomprenden una cantidad efectiva para mitigar el dolor de uncompuesto de acuerdo con el diagrama estructural (1).
ARP000106798A 1999-12-23 2000-12-20 Metodo y composicion para el tratamiento del dolor AR027038A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17190699P 1999-12-23 1999-12-23
US23683500P 2000-09-29 2000-09-29

Publications (1)

Publication Number Publication Date
AR027038A1 true AR027038A1 (es) 2003-03-12

Family

ID=26867559

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000106798A AR027038A1 (es) 1999-12-23 2000-12-20 Metodo y composicion para el tratamiento del dolor

Country Status (23)

Country Link
US (1) US20030162783A1 (es)
EP (1) EP1248621A1 (es)
JP (1) JP2003518499A (es)
KR (1) KR20020062983A (es)
CN (1) CN1434714A (es)
AR (1) AR027038A1 (es)
AU (1) AU783499B2 (es)
BG (1) BG106832A (es)
BR (1) BR0016646A (es)
CA (1) CA2394561A1 (es)
CO (1) CO5271687A1 (es)
EE (1) EE200200348A (es)
HK (1) HK1048767A1 (es)
HU (1) HUP0300043A3 (es)
IL (1) IL150202A0 (es)
IS (1) IS6428A (es)
MX (1) MXPA02006154A (es)
NO (1) NO20022990L (es)
NZ (1) NZ519389A (es)
PL (1) PL355850A1 (es)
RU (1) RU2238094C2 (es)
SK (1) SK8802002A3 (es)
WO (1) WO2001047523A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1325004A1 (en) * 2000-09-29 2003-07-09 AstraZeneca AB 1,2,5,10-tetrahydropyridazino[4,5-b]quinoline-1,10-diones and their use for the treatment of pain
DE60119949T2 (de) * 2000-09-29 2007-04-26 Astrazeneca Ab 1,2,5,10-TETRAHYDROPYRIDAZINOi4,5-BöCHINOLIN-1,10-DIONE UND IHRE ANWENDUNG IN DER BEHANDLUNG VON SCHMERZEN
AU2002214441A1 (en) * 2000-09-29 2002-04-08 Astrazeneca Ab 1,2,5,10-tetrahydropyridazino(4,5-b)quinoline-1,10-diones and their use for the treatment of pain
SE0403172D0 (sv) * 2004-12-23 2004-12-23 Astrazeneca Ab Manufacturing process

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9420590D0 (en) * 1993-10-22 1994-11-30 Zeneca Ltd Pyridazino quinoline compounds
US6730675B2 (en) * 1999-12-23 2004-05-04 Astrazeneca Ab Compounds and methods for the treatment of pain
JP2003519148A (ja) * 1999-12-23 2003-06-17 アストラゼネカ・アクチエボラーグ 痛みの処置のための化合物および方法
EP1244664A1 (en) * 1999-12-23 2002-10-02 AstraZeneca AB Compounds and methods for the treatment of pain

Also Published As

Publication number Publication date
EP1248621A1 (en) 2002-10-16
US20030162783A1 (en) 2003-08-28
NO20022990L (no) 2002-08-20
BG106832A (bg) 2003-03-31
HUP0300043A2 (en) 2003-05-28
RU2238094C2 (ru) 2004-10-20
PL355850A1 (en) 2004-05-31
NO20022990D0 (no) 2002-06-20
KR20020062983A (ko) 2002-07-31
AU2566001A (en) 2001-07-09
HK1048767A1 (zh) 2003-04-17
NZ519389A (en) 2004-05-28
CA2394561A1 (en) 2001-07-05
JP2003518499A (ja) 2003-06-10
IL150202A0 (en) 2002-12-01
SK8802002A3 (en) 2003-06-03
CN1434714A (zh) 2003-08-06
HUP0300043A3 (en) 2007-05-02
EE200200348A (et) 2003-08-15
IS6428A (is) 2002-06-19
CO5271687A1 (es) 2003-04-30
MXPA02006154A (es) 2002-12-05
BR0016646A (pt) 2002-10-08
AU783499B2 (en) 2005-11-03
WO2001047523A1 (en) 2001-07-05

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal