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AR011986A1 - Un proceso para la produccion de aglomerados y un producto farmaceutico obtenido por dicho proceso - Google Patents

Un proceso para la produccion de aglomerados y un producto farmaceutico obtenido por dicho proceso

Info

Publication number
AR011986A1
AR011986A1 ARP980101197A ARP980101197A AR011986A1 AR 011986 A1 AR011986 A1 AR 011986A1 AR P980101197 A ARP980101197 A AR P980101197A AR P980101197 A ARP980101197 A AR P980101197A AR 011986 A1 AR011986 A1 AR 011986A1
Authority
AR
Argentina
Prior art keywords
agglomerates
production
particles
solid binder
amorphous content
Prior art date
Application number
ARP980101197A
Other languages
English (en)
Inventor
Tsong-Toh Yang
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25232603&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR011986(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of AR011986A1 publication Critical patent/AR011986A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • A61K9/1623Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pulmonology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Otolaryngology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Un proceso para la produccion de aglomerados utilizando partículas de por lo menos un primer material y partículas de por lo menos un aglutinante solido,por lo menos uno de dicho primer material y dicho aglutinante solido, teniendo una cantidadpr eseleccionada del contenido amorfo convetible que es capaz deser convertido a forma cristalina con la exposicion a un estímulo preseleccionado, dicho contenido amorfo convertible siendo proporcionado en unacantidad que es suficientecom o para asegurar la formacion de aglomerados; caracterizado porque las partículas de dicho primer material y dichoaglutinante solido son aglomerados, mientras que se mantienen dicha cantidad preseleccionada de contenido amorfo convertiblea un a forma cristalina. Elproceso involucra la produccion de partículas de aglomerado individuales, y luego la conversion del contenido amorfo convertible de los mismos, siendo laaglomeracion, mediante la aplicacion de por ejemplo, humedad. Serefier e a un proceso para la produccion de aglomerados a partir de una droga, tal como uncorticoesteroide, un beta-antagonista, un anticolinérgico, un antagonista de leucotrieno y una proteína o péptido y un ligante solido tal como otra drogaoun sacá rido, tal como lactosa. Además se contemplan aglomerados capaces de conversion así como también los aglomerados terminados y los sistemas dedosificacion oral y nasal incluyendo los mismos. El proceso produceaglomerados que son ásperospero prod ucirán una fraccion de partícula fina aceptabledurante la dosificacion. También se describe un producto obtenido por dicho proceso.
ARP980101197A 1997-03-20 1998-03-17 Un proceso para la produccion de aglomerados y un producto farmaceutico obtenido por dicho proceso AR011986A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US82112997A 1997-03-20 1997-03-20

Publications (1)

Publication Number Publication Date
AR011986A1 true AR011986A1 (es) 2000-09-13

Family

ID=25232603

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP980101197A AR011986A1 (es) 1997-03-20 1998-03-17 Un proceso para la produccion de aglomerados y un producto farmaceutico obtenido por dicho proceso

Country Status (25)

Country Link
EP (3) EP0969816B1 (es)
JP (5) JP3901738B2 (es)
KR (1) KR100386055B1 (es)
CN (3) CN100518718C (es)
AR (1) AR011986A1 (es)
AT (2) ATE284677T1 (es)
AU (1) AU741783B2 (es)
CA (3) CA2706634C (es)
CL (1) CL2011000050A1 (es)
CZ (1) CZ295460B6 (es)
DE (2) DE69828155T2 (es)
DK (2) DK1393721T3 (es)
ES (2) ES2316681T3 (es)
HU (2) HU226671B1 (es)
ID (1) ID24472A (es)
IL (1) IL131640A0 (es)
MY (1) MY120725A (es)
NO (1) NO328062B1 (es)
NZ (1) NZ337443A (es)
PL (3) PL192441B1 (es)
PT (2) PT1393721E (es)
SK (1) SK284919B6 (es)
TW (1) TWI221778B (es)
WO (1) WO1998041193A1 (es)
ZA (1) ZA982254B (es)

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FI20002215A0 (fi) 2000-10-06 2000-10-06 Orion Yhtymae Oyj Yhdistelmäpartikkelit
FI20002216A0 (fi) 2000-10-06 2000-10-06 Orion Yhtymae Oyj Yhdistelmäpartikkelit astman hoitoon
US6667344B2 (en) 2001-04-17 2003-12-23 Dey, L.P. Bronchodilating compositions and methods
US20030055026A1 (en) 2001-04-17 2003-03-20 Dey L.P. Formoterol/steroid bronchodilating compositions and methods of use thereof
ITMI20012174A1 (it) * 2001-10-18 2003-04-18 Univ Parma Polvere per somministrazione nasale di farmaci
US7931022B2 (en) 2001-10-19 2011-04-26 Respirks, Inc. Method and apparatus for dispensing inhalator medicament
EP1452179A1 (en) * 2003-02-27 2004-09-01 CHIESI FARMACEUTICI S.p.A. Novel medicament combination of a highly potent long-lasting beta2-agonist and a corticosteroid
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JP2007501194A (ja) * 2003-08-05 2007-01-25 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ステロイドとβ模倣薬を含む吸入用薬剤
DE60325906D1 (de) 2003-08-08 2009-03-05 Amgen Fremont Inc Antikörper gegen parath-hormon (pth) und ihre verwendungen
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CA2540005A1 (en) * 2003-09-26 2005-04-07 Schering Corporation Pulmonary disease treatment
US20070053843A1 (en) * 2003-10-28 2007-03-08 Dawson Michelle L Inhalable pharmaceutical formulations employing lactose anhydrate and methods of administering the same
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SI1691787T1 (sl) * 2003-12-04 2008-10-31 Pfizer Prod Inc Postopek za pripravo farmacevtskih produktov iz več delcev
SE528121C2 (sv) * 2004-03-29 2006-09-05 Mederio Ag Preparering av torrpulver för på förhand uppmätt DPI
IL168603A (en) * 2005-05-16 2011-05-31 Resdevco Res And Dev Co Pharmaceutical or cosmetic composition for the prevention and treatment of irritation of mucous cells or skin cells
DE102006030166A1 (de) * 2006-06-29 2008-01-10 Boehringer Ingelheim Pharma Gmbh & Co. Kg Tempern
DE102006053375A1 (de) * 2006-11-10 2008-05-15 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Mischung von Pulvern
TW201024034A (en) 2008-12-30 2010-07-01 Saint Gobain Abrasives Inc Bonded abrasive tool and method of forming
EP2421514A2 (en) * 2009-04-24 2012-02-29 Schering Corporation Agglomerate formulations useful in dry powder inhalers
US8815258B2 (en) 2009-05-29 2014-08-26 Pearl Therapeutics, Inc. Compositions, methods and systems for respiratory delivery of two or more active agents
PL2435024T3 (pl) 2009-05-29 2017-01-31 Pearl Therapeutics, Inc. Dostarczanie substancji czynnych do dróg oddechowych oraz powiązane sposoby i systemy
GB0918150D0 (en) * 2009-10-16 2009-12-02 Jagotec Ag Improved formulations
HRP20180488T1 (hr) * 2010-04-21 2018-07-13 Chiesi Farmaceutici S.P.A. Postupak priprave čestica sa smanjenim elektrostatičkim nabojem
CA2905542C (en) 2013-03-15 2022-05-03 Pearl Therapeutics, Inc. Methods and systems for conditioning of particulate crystalline materials
JP6020489B2 (ja) 2014-02-27 2016-11-02 トヨタ自動車株式会社 昇圧コンバータ及びその制御方法
WO2016067252A1 (en) 2014-10-31 2016-05-06 Glaxosmithkline Intellectual Property Development Limited Powder formulation
EP3400214B1 (en) * 2016-01-08 2024-03-13 Theron Pharmaceuticals, Inc. Dry powder inhaler compositions of 7-azoniabicyclo[2.2.1]heptane derivatives
CN117122585A (zh) * 2023-07-27 2023-11-28 宁波诺丁汉大学 一种通过振动混合制备干粉吸入团聚物处方制剂方法

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GB8334494D0 (en) 1983-12-24 1984-02-01 Tanabe Seiyaku Co Carbostyril derivatives
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JP2924924B2 (ja) * 1992-12-18 1999-07-26 シェリング・コーポレーション 粉末薬物のための吸入器
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Also Published As

Publication number Publication date
CA2282360A1 (en) 1998-09-24
CA2481868C (en) 2010-06-15
DK1393721T3 (da) 2009-03-30
NO328062B1 (no) 2009-11-13
TWI221778B (en) 2004-10-11
CA2481868A1 (en) 1998-09-24
JP2010248260A (ja) 2010-11-04
CA2706634A1 (en) 1998-09-24
HU230274B1 (hu) 2015-11-30
HU226671B1 (en) 2009-06-29
IL131640A0 (en) 2001-01-28
EP1393721B1 (en) 2008-11-26
DK0969816T3 (da) 2005-03-14
PL208480B1 (pl) 2011-05-31
PT1393721E (pt) 2009-02-02
EP0969816A1 (en) 2000-01-12
EP2036544A1 (en) 2009-03-18
MY120725A (en) 2005-11-30
CZ295460B6 (cs) 2005-08-17
CA2706634C (en) 2012-10-23
JP3901738B2 (ja) 2007-04-04
EP2036544B1 (en) 2016-12-28
NO994519L (no) 1999-11-19
ATE415149T1 (de) 2008-12-15
AU6537898A (en) 1998-10-12
KR100386055B1 (ko) 2003-06-09
ES2234102T3 (es) 2005-06-16
CN1903179A (zh) 2007-01-31
HK1021323A1 (en) 2000-06-09
PL192441B1 (pl) 2006-10-31
JP2010275316A (ja) 2010-12-09
HK1061359A1 (en) 2004-09-17
CN100518718C (zh) 2009-07-29
SK284919B6 (sk) 2006-02-02
CN100548277C (zh) 2009-10-14
ID24472A (id) 2000-07-20
PT969816E (pt) 2005-04-29
DE69828155T2 (de) 2005-12-22
KR20010005520A (ko) 2001-01-15
CL2011000050A1 (es) 2011-06-24
DE69828155D1 (de) 2005-01-20
NO994519D0 (no) 1999-09-17
CA2282360C (en) 2004-11-09
HU0600845D0 (en) 2007-01-29
HUP0002029A2 (hu) 2000-11-28
JP2006152000A (ja) 2006-06-15
PL335742A1 (en) 2000-05-08
CZ323399A3 (cs) 2000-02-16
AU741783B2 (en) 2001-12-06
DE69840277D1 (de) 2009-01-08
ATE284677T1 (de) 2005-01-15
CN1149076C (zh) 2004-05-12
CN1257423A (zh) 2000-06-21
PL204480B1 (pl) 2010-01-29
JP5523240B2 (ja) 2014-06-18
NZ337443A (en) 2001-04-27
ZA982254B (en) 1998-09-17
WO1998041193A1 (en) 1998-09-24
CN1552310A (zh) 2004-12-08
JP2014037446A (ja) 2014-02-27
HUP0002029A3 (en) 2001-02-28
EP1393721A1 (en) 2004-03-03
EP0969816B1 (en) 2004-12-15
JP2000510478A (ja) 2000-08-15
ES2316681T3 (es) 2009-04-16
SK128099A3 (en) 2000-06-12

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