AP1828A - Muscarinic Acetycholine receptor antagonists - Google Patents

Muscarinic Acetycholine receptor antagonists

Info

Publication number: AP1828A
Authority: AP; ARIPO
Prior art keywords: receptor antagonists; acetycholine receptor; muscarinic; muscarinic acetycholine; antagonists
Prior art date: 2003-10-14

Application number

AP2006003566A

Other languages

English (en)

Other versions

AP2006003566A0 (en

Inventor

Michael R Palovich

Jakob Busch-Petersen

Zehong Wan

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-10-14

Filing date

2004-10-12

Publication date

2008-02-13

2004-10-12 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

2006-04-30 Publication of AP2006003566A0 publication Critical patent/AP2006003566A0/xx

2008-02-13 Application granted granted Critical

2008-02-13 Publication of AP1828A publication Critical patent/AP1828A/xx

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Urology & Nephrology (AREA)
Epidemiology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Emergency Medicine (AREA)
Rheumatology (AREA)
Otolaryngology (AREA)
Pain & Pain Management (AREA)
Immunology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)

AP2006003566A 2003-10-14 2004-10-12 Muscarinic Acetycholine receptor antagonists AP1828A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US51100903P	2003-10-14	2003-10-14
PCT/US2004/033638 WO2005037280A1 (en)	2003-10-14	2004-10-12	Muscarinic acetycholine receptor antagonists

Publications (2)

Publication Number	Publication Date
AP2006003566A0 AP2006003566A0 (en)	2006-04-30
AP1828A true AP1828A (en)	2008-02-13

Family

ID=34465175

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
AP2006003566A AP1828A (en)	2003-10-14	2004-10-12	Muscarinic Acetycholine receptor antagonists
AP2007004239A AP2007004239A0 (en)	2003-10-14	2004-10-12	Muscarinic acetycholine receptor antagonists
AP2007004238A AP2007004238A0 (en)	2003-10-14	2004-10-12	Muscarinic acetycholine receptor antagonists

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
AP2007004239A AP2007004239A0 (en)	2003-10-14	2004-10-12	Muscarinic acetycholine receptor antagonists
AP2007004238A AP2007004238A0 (en)	2003-10-14	2004-10-12	Muscarinic acetycholine receptor antagonists

Country Status (34)

Country	Link
US (3)	US7276521B2 (xx)
EP (1)	EP1677795B1 (xx)
JP (4)	JP2007508390A (xx)
KR (3)	KR20080067023A (xx)
CN (3)	CN1893948A (xx)
AP (3)	AP1828A (xx)
AR (1)	AR046103A1 (xx)
AT (1)	ATE494285T1 (xx)
AU (1)	AU2004281724B2 (xx)
BR (1)	BRPI0415361A (xx)
CA (1)	CA2542657C (xx)
CY (1)	CY1111364T1 (xx)
DE (1)	DE602004030930D1 (xx)
DK (1)	DK1677795T3 (xx)
EA (3)	EA013435B1 (xx)
EC (1)	ECSP066468A (xx)
ES (1)	ES2358673T3 (xx)
HR (1)	HRP20110232T1 (xx)
IL (2)	IL174843A0 (xx)
IS (1)	IS2918B (xx)
MA (1)	MA28110A1 (xx)
MX (1)	MXPA06004244A (xx)
MY (1)	MY143366A (xx)
NO (1)	NO20062042L (xx)
NZ (2)	NZ556424A (xx)
OA (1)	OA13316A (xx)
PE (1)	PE20050963A1 (xx)
PL (1)	PL1677795T3 (xx)
PT (1)	PT1677795E (xx)
SG (1)	SG147436A1 (xx)
SI (1)	SI1677795T1 (xx)
TW (3)	TW200811172A (xx)
UA (2)	UA89734C2 (xx)
WO (1)	WO2005037280A1 (xx)

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WO2010097114A1 (en) *	2009-02-26	2010-09-02	Glaxo Group Limited	Novel combination of therapeutic agents
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HUE026059T2 (en)	2010-09-08	2016-05-30	Glaxosmithkline Ip Dev Ltd	N- [5- [4- (5 - {[(2R, 6S) -2,6-dimethyl-4-morpholinyl] methyl} -1,3-oxazol-2-yl) -1H-indazol-6-yl ] Polymorphs and salts of 2 - (methyloxy) -3-pyridinyl] methanesulfonamide
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2004
- 2004-10-12 TW TW096137868A patent/TW200811172A/zh unknown
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2007
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Patent Citations (2)

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US2800478A (en) *	1955-07-01	1957-07-23	Smith Kline French Lab	3-substituted-8-alkylnortropanes and the acid and quaternary ammonium salts thereof
US2800481A (en) *	1955-07-01	1957-07-23	Smith Kline French Lab	Tertiary alcohol derivatives of 8-alkylnortropanes and the acid and quaternary ammonium salts thereof

Also Published As

Publication number	Publication date
AU2004281724A1 (en)	2005-04-28
US20070105895A1 (en)	2007-05-10
ES2358673T3 (es)	2011-05-12
JP2007508390A (ja)	2007-04-05
KR20080067023A (ko)	2008-07-17
EA013435B1 (ru)	2010-04-30
ATE494285T1 (de)	2011-01-15
DK1677795T3 (da)	2011-04-18
WO2005037280A1 (en)	2005-04-28
UA87473C2 (xx)	2009-07-27
JP4796552B2 (ja)	2011-10-19
EP1677795A4 (en)	2006-12-27
TWI409060B (zh)	2013-09-21
TW200811171A (en)	2008-03-01
EA200702617A1 (ru)	2008-04-28
IL174843A0 (en)	2006-08-20
AP2006003566A0 (en)	2006-04-30
HRP20110232T1 (hr)	2011-05-31
US20070238752A1 (en)	2007-10-11
CA2542657A1 (en)	2005-04-28
DE602004030930D1 (de)	2011-02-17
NZ546312A (en)	2008-09-26
US7579361B2 (en)	2009-08-25
MXPA06004244A (es)	2006-06-28
ECSP066468A (es)	2006-11-16
AU2004281724B2 (en)	2010-07-15
MA28110A1 (fr)	2006-08-01
UA89734C2 (xx)	2010-02-25
CY1111364T1 (el)	2015-08-05
AP2007004239A0 (en)	2007-12-31
EA013689B1 (ru)	2010-06-30
AP2007004238A0 (en)	2007-12-31
AR046103A1 (es)	2005-11-23
BRPI0415361A (pt)	2006-12-12
PT1677795E (pt)	2011-04-01
KR20080065318A (ko)	2008-07-11
SI1677795T1 (sl)	2011-04-29
SG147436A1 (en)	2008-11-28
JP5450509B2 (ja)	2014-03-26
PE20050963A1 (es)	2006-01-11
CN1893948A (zh)	2007-01-10
OA13316A (en)	2007-04-13
PL1677795T3 (pl)	2011-05-31
US20070244150A1 (en)	2007-10-18
CN101230061A (zh)	2008-07-30
IL188112A0 (en)	2008-03-20
IL188112A (en)	2012-10-31
TW200811172A (en)	2008-03-01
CN101230062A (zh)	2008-07-30
TW200522933A (en)	2005-07-16
NO20062042L (no)	2006-05-08
EA009899B1 (ru)	2008-04-28
JP2007314567A (ja)	2007-12-06
MY143366A (en)	2011-04-29
JP2011162556A (ja)	2011-08-25
JP2007277276A (ja)	2007-10-25
CA2542657C (en)	2011-03-01
IS2918B (is)	2015-01-15
EP1677795B1 (en)	2011-01-05
US7276521B2 (en)	2007-10-02
EP1677795A1 (en)	2006-07-12
NZ556424A (en)	2008-12-24
EA200600773A1 (ru)	2008-04-28
EA200702619A1 (ru)	2008-04-28
US7576096B2 (en)	2009-08-18
KR20060106821A (ko)	2006-10-12
IS8441A (is)	2006-05-05

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AP1828A (en)	2008-02-13	Muscarinic Acetycholine receptor antagonists
AU2003261392A8 (en)	2004-02-23	M3muscarinic acetylcholine receptor antagonists
SI1638969T1 (sl)	2009-02-28	Antagonisti cgrp receptorjev
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IL172911A0 (en)	2006-06-11	Muscarinic acetylcholine receptor antagonists
EP1613307A4 (en)	2008-03-12	M SB 3 / SB MUSCARIN ACETYLCHOLINE RECEPTOR ANTAGONISTS
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