NO970511L - Nye substituerte oksazolidinoner - Google Patents
Nye substituerte oksazolidinonerInfo
- Publication number
- NO970511L NO970511L NO970511A NO970511A NO970511L NO 970511 L NO970511 L NO 970511L NO 970511 A NO970511 A NO 970511A NO 970511 A NO970511 A NO 970511A NO 970511 L NO970511 L NO 970511L
- Authority
- NO
- Norway
- Prior art keywords
- substituted oxazolidinones
- newly substituted
- formula
- drugs
- oxazolidinones
- Prior art date
Links
- IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical class O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 title abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 229940124350 antibacterial drug Drugs 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
- C07F9/6581—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and nitrogen atoms with or without oxygen or sulfur atoms, as ring hetero atoms
- C07F9/6584—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and nitrogen atoms with or without oxygen or sulfur atoms, as ring hetero atoms having one phosphorus atom as ring hetero atom
- C07F9/65842—Cyclic amide derivatives of acids of phosphorus, in which one nitrogen atom belongs to the ring
- C07F9/65844—Cyclic amide derivatives of acids of phosphorus, in which one nitrogen atom belongs to the ring the phosphorus atom being part of a five-membered ring which may be condensed with another ring system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Det blir beskrevet nye substituerte oksazolidinoner med den generelle formel (I). hvor A eksempelvis står for en heterocykl1sk ringstruk-tur bundet over et karbonatom og Rstår for en rest med en av formelene. eller for cyano eller for en 5- til 7-leddes mettet, delvis umettet eller umettet heterocyklus.Forbindelser med formel (I) er anvendelige legemidler, spesielt i antlbakterielle legemidler. Det blir dessuten beskrevet en fremgangsmåte for deres fremstilling.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19604223A DE19604223A1 (de) | 1996-02-06 | 1996-02-06 | Neue substituierte Oxazolidinone |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO970511D0 NO970511D0 (no) | 1997-02-05 |
| NO970511L true NO970511L (no) | 1997-08-07 |
Family
ID=7784633
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO970511A NO970511L (no) | 1996-02-06 | 1997-02-05 | Nye substituerte oksazolidinoner |
Country Status (36)
| Country | Link |
|---|---|
| US (1) | US5792765A (no) |
| EP (1) | EP0789025B1 (no) |
| JP (1) | JPH09316073A (no) |
| KR (1) | KR970061888A (no) |
| CN (1) | CN1160051A (no) |
| AR (1) | AR005703A1 (no) |
| AT (1) | ATE200285T1 (no) |
| AU (1) | AU1251697A (no) |
| BG (1) | BG101193A (no) |
| BR (1) | BR9700885A (no) |
| CA (1) | CA2196862A1 (no) |
| CO (1) | CO4560411A1 (no) |
| CZ (1) | CZ34097A3 (no) |
| DE (2) | DE19604223A1 (no) |
| DK (1) | DK0789025T3 (no) |
| EE (1) | EE9700043A (no) |
| ES (1) | ES2157027T3 (no) |
| GR (1) | GR3036015T3 (no) |
| HR (1) | HRP970048A2 (no) |
| HU (1) | HUP9700358A3 (no) |
| ID (1) | ID15881A (no) |
| IL (1) | IL120125A0 (no) |
| MX (1) | MX9700886A (no) |
| NO (1) | NO970511L (no) |
| NZ (1) | NZ314179A (no) |
| PL (1) | PL318277A1 (no) |
| PT (1) | PT789025E (no) |
| SG (1) | SG50791A1 (no) |
| SI (1) | SI0789025T1 (no) |
| SK (1) | SK15897A3 (no) |
| SV (1) | SV1997000009A (no) |
| TN (1) | TNSN97032A1 (no) |
| TR (1) | TR199700092A2 (no) |
| TW (1) | TW350845B (no) |
| YU (1) | YU4397A (no) |
| ZA (1) | ZA97927B (no) |
Families Citing this family (67)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
| ES2242280T3 (es) | 1997-05-30 | 2005-11-01 | PHARMACIA & UPJOHN COMPANY LLC | Agentes antibacterianos de oxazolidinona que contienen funcionalidad tiocarbonilo. |
| US6255304B1 (en) | 1997-05-30 | 2001-07-03 | Pharmacia & Upjohn Company | Oxazolidinone antibacterial agents having a thiocarbonyl functionality |
| WO1999012914A1 (en) * | 1997-09-11 | 1999-03-18 | Hokuriku Seiyaku Co., Ltd. | Thiourea derivatives |
| KR100619639B1 (ko) * | 1997-11-07 | 2006-09-06 | 파마시아 앤드 업존 캄파니 엘엘씨 | 옥사졸리디논의 제조 방법 |
| DE19802239A1 (de) * | 1998-01-22 | 1999-07-29 | Bayer Ag | Neue mit Bicyclen substituierte Oxazolidinone |
| NZ505902A (en) * | 1998-01-23 | 2003-08-29 | Upjohn Co | Oxazolidinone compounds useful as antimicrobial agents and combinatorial libraries |
| ID30299A (id) * | 1998-06-05 | 2001-11-22 | Astrazeneca Ab | Turunan oksazolidinon, proses pembuatannya dan komposisi farmasi yang mengandungnya |
| GB9821938D0 (en) * | 1998-10-09 | 1998-12-02 | Zeneca Ltd | Chemical compounds |
| JP2000204084A (ja) * | 1998-11-11 | 2000-07-25 | Hokuriku Seiyaku Co Ltd | チオカルバミド酸誘導体 |
| WO2000029409A1 (de) * | 1998-11-17 | 2000-05-25 | Bayer Aktiengesellschaft | Neue heterocyclyl-substituierte oxazolidon-derivate |
| AU1379900A (en) * | 1998-11-17 | 2000-06-05 | Bayer Aktiengesellschaft | Novel substituted phenyloxazolidone derivatives |
| EP1008590B1 (en) | 1998-12-07 | 2006-10-11 | Takasago International Corporation | Process for preparing optically active oxazolidinone derivatives |
| ATE246189T1 (de) * | 1999-05-27 | 2003-08-15 | Upjohn Co | Bizyklische oxazolidinone als antibakterielle mittel |
| BR0012742A (pt) | 1999-07-28 | 2002-06-11 | Upjohn Co | Oxazolidinonas e seus usos como antibiótico |
| US6413981B1 (en) | 1999-08-12 | 2002-07-02 | Ortho-Mcneil Pharamceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| US6297242B1 (en) | 1999-08-12 | 2001-10-02 | Ortho-Mcneil Pharmaceutical, Inc. | N-substituted amidine and guanidine oxazolidinone antibacterials and methods of use thereof |
| US6608081B2 (en) | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
| US6518285B2 (en) | 1999-12-21 | 2003-02-11 | Ortho Mcneil Pharmaceutical, Inc. | Piperidinyloxy and pyrrolidinyloxy oxazolidinone antibacterials |
| ATE243357T1 (de) | 1999-12-23 | 2003-07-15 | Hans-Peter Wilfer | Musikinstrumentbehältnis, insbesondere für gitarren |
| DE19962924A1 (de) | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
| KR100355345B1 (ko) * | 2000-01-21 | 2002-10-12 | 한국과학기술연구원 | 티오펜환을 함유한 신규한 옥사졸리디논 유도체, 그의 제조방법 및 조성물 |
| MY127336A (en) | 2000-03-22 | 2006-11-30 | Upjohn Co | Container for linezolid iv solution |
| US6514529B2 (en) | 2000-03-22 | 2003-02-04 | Pharmacia & Upjohn Company | Oxazolidinone tablet formulation |
| PE20011124A1 (es) | 2000-03-31 | 2001-10-28 | Upjohn Co | Nuevos agentes antibacterianos de benzosultam oxazolidinona |
| GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
| AU2001272961A1 (en) | 2000-06-30 | 2002-01-14 | Pharmacia & Upjohn Company | Compositions for treating bacterial infections containing oxazolidinone compound, sulbactam and an ampicillin |
| PE20030044A1 (es) * | 2000-11-17 | 2003-02-09 | Upjohn Co | Isoxazolinonas biciclicas de formula i |
| AU2002256995A1 (en) * | 2001-02-07 | 2002-08-28 | Ortho-Mcneil Pharmaceutical, Inc. | Pyridoarylphenyl oxazolidinone antibacterials, and related compositions and methods |
| DE10129725A1 (de) * | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
| TW200302095A (en) * | 2002-01-25 | 2003-08-01 | Upjohn Co | Oxazolidinone cotherapy |
| US7141588B2 (en) * | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
| AR038536A1 (es) * | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
| PL372661A1 (en) * | 2002-03-29 | 2005-07-25 | Pharmacia & Upjohn Company Llc. | Parenteral, intravenous, and oral administration of oxazolidinones for treating diabetic foot infections |
| CA2491287A1 (en) * | 2002-08-12 | 2004-02-19 | Pharmacia & Upjohn Company | N-aryl-2-oxazolidinones and their derivatives |
| AU2002339721A1 (en) * | 2002-09-20 | 2004-04-08 | Lupin Limited | Oxazolidinone derivatives, process for their preperation and their use as antimycobacterial agents |
| US7091196B2 (en) * | 2002-09-26 | 2006-08-15 | Rib-X Pharmaceuticals, Inc. | Bifunctional heterocyclic compounds and methods of making and using same |
| ATE344036T1 (de) * | 2002-11-21 | 2006-11-15 | Pharmacia & Upjohn Co Llc | N-(4-(piperazin-1-yl)-phenyl-2-oxazolidinon-5- carbonsäureamid-derivate und verwandte verbindungen als antibakterielle mittel |
| DE10300111A1 (de) | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
| JP2006516989A (ja) * | 2003-02-07 | 2006-07-13 | ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー | 抗菌剤として使用するための二環式環によりn−置換されたオキサゾリジノン誘導体 |
| CA2515311A1 (en) * | 2003-02-07 | 2004-08-19 | Warner-Lambert Company Llc | Antibacterial agents |
| US7012088B2 (en) * | 2003-02-24 | 2006-03-14 | Pharmacia & Upjohn Company | Indolone oxazolidinones and derivatives thereof |
| US20040204463A1 (en) * | 2003-04-01 | 2004-10-14 | Harris Christina Renee | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
| EP1660488A1 (en) * | 2003-08-25 | 2006-05-31 | Warner-Lambert Company LLC | Novel antimicrobial aryloxazolidinone compounds |
| US7304050B2 (en) * | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
| DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
| WO2005082897A1 (en) * | 2004-01-28 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Oxazolidinone antibacterial agents |
| WO2005082900A2 (en) * | 2004-01-28 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Oxazolidinone amidoximes as antibacterial agents |
| US8202843B2 (en) | 2004-02-27 | 2012-06-19 | Rib-X Pharmaceuticals, Inc. | Macrocyclic compounds and methods of making and using the same |
| DE102004062475A1 (de) * | 2004-12-24 | 2006-07-06 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung |
| EP1685841A1 (en) | 2005-01-31 | 2006-08-02 | Bayer Health Care Aktiengesellschaft | Prevention and treatment of thromboembolic disorders |
| AU2006231919A1 (en) | 2005-04-06 | 2006-10-12 | Pharmacia & Upjohn Company Llc | 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents |
| EP3290427A1 (en) * | 2005-08-24 | 2018-03-07 | Melinta Therapeutics, Inc. | Triazole compounds and methods of making and using the same |
| JP2009506063A (ja) | 2005-08-24 | 2009-02-12 | リブ−エックス ファーマシューティカルズ,インコーポレイテッド | トリアゾール化合物ならびにこれを作製する方法および使用する方法 |
| DE102005045518A1 (de) | 2005-09-23 | 2007-03-29 | Bayer Healthcare Ag | 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung |
| DE102005047561A1 (de) | 2005-10-04 | 2007-04-05 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung |
| PT1934208E (pt) | 2005-10-04 | 2011-06-01 | Bayer Schering Pharma Ag | Nova forma polimorfa de 5-cloro-n-({(5s)-2-oxo-3-[4-(3- oxo-4-morfolinil)-fenil]-1,3-oxazolidin-5-il}-metil)-2- tiofenocarboxamida |
| DE102005047558A1 (de) * | 2005-10-04 | 2008-02-07 | Bayer Healthcare Ag | Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen |
| WO2008021309A1 (en) * | 2006-08-15 | 2008-02-21 | Wyeth | Imidazolidin-2-one derivatives useful as pr modulators |
| TW200815428A (en) | 2006-08-15 | 2008-04-01 | Wyeth Corp | Oxazolidone derivatives as PR modulators |
| WO2008021337A1 (en) | 2006-08-15 | 2008-02-21 | Wyeth | Oxazinan-2-one derivatives useful as pr modulators |
| US7649007B2 (en) * | 2006-08-15 | 2010-01-19 | Wyeth Llc | Oxazolidine derivatives as PR modulators |
| DE102006051625A1 (de) * | 2006-11-02 | 2008-05-08 | Bayer Materialscience Ag | Kombinationstherapie substituierter Oxazolidinone |
| US20100298384A1 (en) * | 2006-12-04 | 2010-11-25 | Mohamed Takhi | Novel oxazolidinone compounds as antiinfective agents |
| WO2009104159A1 (en) * | 2008-02-22 | 2009-08-27 | Actelion Pharmaceuticals Ltd | Oxazolidinone derivatives |
| WO2018170664A1 (en) * | 2017-03-20 | 2018-09-27 | Merck Sharp & Dohme Corp. | Oxazolidinone compounds and methods of use thereof as antibacterial agents |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4705799A (en) | 1983-06-07 | 1987-11-10 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents |
| US4965268A (en) * | 1987-10-09 | 1990-10-23 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
| US5032605A (en) * | 1987-10-09 | 1991-07-16 | Du Pont Merck Pharmaceutical Company | Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents |
| US4801600A (en) * | 1987-10-09 | 1989-01-31 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
| US4942183A (en) * | 1987-10-16 | 1990-07-17 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents |
| CA1320730C (en) | 1987-10-16 | 1993-07-27 | The Du Pont Merck Pharmaceutical Company | Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents |
| US5254577A (en) | 1988-07-29 | 1993-10-19 | The Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| US5164510A (en) * | 1988-09-15 | 1992-11-17 | The Upjohn Company | 5'Indolinyl-5β-amidomethyloxazolidin-2-ones |
| JP2865211B2 (ja) | 1988-09-15 | 1999-03-08 | ファルマシア・アンド・アップジョン・カンパニー | 5’―インドリニル―5β―アミドメチルオキサゾリジン―2―オン類、3―(縮合環置換)フェニル―5β―アミドメチルオキサゾリジン―2―オン類および3―(窒素原子置換)フェニル―5β―アミドメチルオキサゾリジン―2―オン類 |
| JP2669579B2 (ja) * | 1991-10-23 | 1997-10-29 | エーザイ株式会社 | オキサゾリドン誘導体 |
| DE4303303C1 (de) | 1993-02-05 | 1994-02-17 | Freudenberg Carl Fa | Antriebsstrang eines Kraftfahrzeugs |
| DE4332384A1 (de) * | 1993-09-23 | 1995-03-30 | Merck Patent Gmbh | Adhäsionsrezeptor-Antagonisten III |
| TW286317B (no) * | 1993-12-13 | 1996-09-21 | Hoffmann La Roche | |
| DE4425612A1 (de) | 1994-07-20 | 1996-04-04 | Bayer Ag | 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone |
| DE4425609A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | Benzofuranyl- und Benzothienyloxazolidinone |
| DE4425613A1 (de) | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
| DE19514313A1 (de) * | 1994-08-03 | 1996-02-08 | Bayer Ag | Benzoxazolyl- und Benzothiazolyloxazolidinone |
| HRP960159A2 (en) | 1995-04-21 | 1997-08-31 | Bayer Ag | Benzocyclopentane oxazolidinones containing heteroatoms |
-
1996
- 1996-02-06 DE DE19604223A patent/DE19604223A1/de not_active Withdrawn
-
1997
- 1997-01-27 HR HR19604223.2A patent/HRP970048A2/hr not_active Application Discontinuation
- 1997-01-31 DE DE59703261T patent/DE59703261D1/de not_active Expired - Fee Related
- 1997-01-31 SI SI9730110T patent/SI0789025T1/xx unknown
- 1997-01-31 PT PT97101509T patent/PT789025E/pt unknown
- 1997-01-31 EP EP97101509A patent/EP0789025B1/de not_active Expired - Lifetime
- 1997-01-31 AT AT97101509T patent/ATE200285T1/de not_active IP Right Cessation
- 1997-01-31 DK DK97101509T patent/DK0789025T3/da active
- 1997-01-31 ES ES97101509T patent/ES2157027T3/es not_active Expired - Lifetime
- 1997-02-03 US US08/794,034 patent/US5792765A/en not_active Expired - Fee Related
- 1997-02-03 NZ NZ314179A patent/NZ314179A/xx unknown
- 1997-02-03 IL IL12012597A patent/IL120125A0/xx unknown
- 1997-02-04 TN TNTNSN97032A patent/TNSN97032A1/fr unknown
- 1997-02-04 MX MX9700886A patent/MX9700886A/es unknown
- 1997-02-04 ID IDP970341A patent/ID15881A/id unknown
- 1997-02-04 AR ARP970100439A patent/AR005703A1/es unknown
- 1997-02-04 AU AU12516/97A patent/AU1251697A/en not_active Abandoned
- 1997-02-04 BG BG101193A patent/BG101193A/xx unknown
- 1997-02-04 PL PL97318277A patent/PL318277A1/xx unknown
- 1997-02-04 TW TW086101259A patent/TW350845B/zh active
- 1997-02-05 EE EE9700043A patent/EE9700043A/xx unknown
- 1997-02-05 SG SG1997000259A patent/SG50791A1/en unknown
- 1997-02-05 TR TR97/00092A patent/TR199700092A2/xx unknown
- 1997-02-05 KR KR1019970003610A patent/KR970061888A/ko not_active Withdrawn
- 1997-02-05 NO NO970511A patent/NO970511L/no unknown
- 1997-02-05 CZ CZ97340A patent/CZ34097A3/cs unknown
- 1997-02-05 SK SK158-97A patent/SK15897A3/sk unknown
- 1997-02-05 CA CA002196862A patent/CA2196862A1/en not_active Abandoned
- 1997-02-05 YU YU4397A patent/YU4397A/sh unknown
- 1997-02-05 HU HU9700358A patent/HUP9700358A3/hu unknown
- 1997-02-05 ZA ZA9700927A patent/ZA97927B/xx unknown
- 1997-02-05 BR BR9700885A patent/BR9700885A/pt not_active Application Discontinuation
- 1997-02-06 JP JP9036908A patent/JPH09316073A/ja active Pending
- 1997-02-06 SV SV1997000009A patent/SV1997000009A/es unknown
- 1997-02-06 CN CN97101879A patent/CN1160051A/zh active Pending
- 1997-02-06 CO CO97006151A patent/CO4560411A1/es unknown
-
2001
- 2001-06-08 GR GR20010400867T patent/GR3036015T3/el not_active IP Right Cessation
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO970511L (no) | Nye substituerte oksazolidinoner | |
| NO975987L (no) | 4-Fenylaminotiazol-derivater, fremgangsmåte for fremstilling av disse og farmasöytiske blandinger inneholdende nevnte derivater | |
| YU49443B (sh) | Derivati benzimidazola, postupci za njihovo pripremanje i primena tih derivata u medicinskoj terapiji, naročito za lečenje ili sprečavanje virusnih infekcija | |
| ATE246190T1 (de) | Heterozyklische verbindungen, verfahren zu ihrer herstellung, pharmazeutische zusammensetzungen die diese enthalten und ihre anwendung in der behandlung von diabetis und verwandten krankheiten | |
| DE59610509D1 (de) | Neue 4-(oxyalkoxyphenyl)-3-oxy-piperidine zur behandlung von herz- und niereninsuffizienz | |
| DK104292D0 (da) | Heterocycliske forbindelser og fremgangsmaade til deres fremstilling | |
| DE69111029D1 (de) | Kondensierte heterocyclische Verbindungen, ihre Herstellung und Verwendung. | |
| NO970512L (no) | Nye heteroaryl-oksazolidinoner | |
| DE3681517D1 (de) | Thiazolidinderivate, verfahren zu deren herstellung und deren anwendung. | |
| DE69709938D1 (de) | N-benzylpiperidin- und tetrahydropyridin-derivate | |
| ATE88894T1 (de) | Methode zur behandlung von kachexie und bestimmte dafuer anzuwendende verbindungen. | |
| NO163855C (no) | Analogifremgangsmaate for fremstilling av terapeutisk aktive arylcyklobutylalkylaminer. | |
| CA2321188A1 (en) | Derivatives of azetidine and pyrrolidine | |
| NO870944D0 (no) | Fremgangsmaate for fremstilling av heteroaryl-oxy-beta-carbolin-derivater. | |
| NO308532B1 (no) | Farmasøytiske piperazinforbindelser | |
| NO170215C (no) | Analogifremgangsmaate ved fremstilling av terapeutisk aktive imidazolderivater | |
| FI922835A0 (fi) | Menetelmä terapeuttisesti aktiivisten piperidiinijohdannaisten valmistamiseksi | |
| FR2449677B1 (fr) | Nouveaux derives de benzoyl-2 glycylanilides substitues, leur preparation et leur application en tant que medicaments anxiolytiques | |
| ATE121383T1 (de) | Polyhydroxycyclopentan derivate, ihre herstellung und ihre therapeutische verwendung. | |
| DE69522118D1 (de) | Thiazolidonon- oder oxazolidinonderivate zur behandlung von angina pectoris und zusammensetzungen die diese als wirkstoffe enthält | |
| ES2131824T3 (es) | Compuestos de piridina sustituidos en 3 y derivados de los mismos como herbicidas. | |
| NO171639C (no) | Analogifremgangsmaate til fremstilling av terapeutisk aktive imidazolpyrazolderivater | |
| NO170630C (no) | Analogifremgangsmaate ved fremstilling av nye, terapeutiskaktive 1-(3-(2-sek.-aminoetoksy)-2-tienyl)-3-fenyl-propanoner og syreaddisjonssalter derav | |
| NO984547L (no) | Nye oksazolidinderivater, fremgangsmÕte for deres fremstilling, samt legemidler inneholdende disse forbindelser | |
| ATE18227T1 (de) | C-homo-9-oxaergolinderivate, ihre salze, verfahren zu ihrer herstellung, ihre verwendung als arzneimittel und diese enthaltende zubereitungen. |