NO974603L - Anvendelse av imidazo£1,2-a|pyridin-3-acetamidderivater for terapeutisk behandling av neuropsykiatriske syndromer assosiert med disfunksjon av de sentrale områder av de basale ganglia - Google Patents
Anvendelse av imidazo£1,2-a|pyridin-3-acetamidderivater for terapeutisk behandling av neuropsykiatriske syndromer assosiert med disfunksjon av de sentrale områder av de basale gangliaInfo
- Publication number
- NO974603L NO974603L NO974603A NO974603A NO974603L NO 974603 L NO974603 L NO 974603L NO 974603 A NO974603 A NO 974603A NO 974603 A NO974603 A NO 974603A NO 974603 L NO974603 L NO 974603L
- Authority
- NO
- Norway
- Prior art keywords
- imidazo
- dysfunction
- therapeutic treatment
- basal ganglia
- central regions
- Prior art date
Links
- YDHIMEXEGOCNHU-UHFFFAOYSA-N 2-pyridin-3-ylacetamide Chemical class NC(=O)CC1=CC=CN=C1 YDHIMEXEGOCNHU-UHFFFAOYSA-N 0.000 title 1
- 206010071323 Neuropsychiatric syndrome Diseases 0.000 title 1
- 210000004227 basal ganglia Anatomy 0.000 title 1
- 230000004064 dysfunction Effects 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Psychology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT95RM000223A IT1276522B1 (it) | 1995-04-07 | 1995-04-07 | Uso dello zolpidem per il trattamento terapeudico di sindromi neuropsichiatriche associate a disfunsione e di circuiti neurali dei |
| PCT/IT1996/000063 WO1996031210A1 (en) | 1995-04-07 | 1996-04-02 | USE OF IMIDAZO[1,2-a]PYRIDINE-3-ACETAMIDE DERIVATIVES FOR THE THERAPEUTIC TREATMENT OF NEUROPSYCHIATRIC SYNDROMES ASSOCIATED WITH DISFUNCTION OF THE NEURAL CIRCUITS OF THE BASAL GANGLIA |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO974603D0 NO974603D0 (no) | 1997-10-06 |
| NO974603L true NO974603L (no) | 1997-11-24 |
| NO315408B1 NO315408B1 (no) | 2003-09-01 |
Family
ID=11403250
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19974603A NO315408B1 (no) | 1995-04-07 | 1997-10-06 | Anvendelse av imidazo[1,2-a]pyridin-3-acetamidderivater for terapeutisk behandling av neuropsykiatriske syndromer assosiert med disfunksjonav de sentraleområder av de basale ganglia |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US5891891A (no) |
| EP (1) | EP0819002B1 (no) |
| JP (1) | JP4049390B2 (no) |
| KR (1) | KR100425628B1 (no) |
| CN (1) | CN1198612C (no) |
| AR (1) | AR003414A1 (no) |
| AT (1) | ATE222763T1 (no) |
| AU (1) | AU707759B2 (no) |
| CA (1) | CA2217590C (no) |
| CZ (1) | CZ292020B6 (no) |
| DE (1) | DE69623271T2 (no) |
| DK (1) | DK0819002T3 (no) |
| EA (1) | EA000396B1 (no) |
| ES (1) | ES2182967T3 (no) |
| HU (1) | HUP9900733A3 (no) |
| IL (1) | IL117824A (no) |
| IT (1) | IT1276522B1 (no) |
| MX (1) | MX9707712A (no) |
| NO (1) | NO315408B1 (no) |
| NZ (1) | NZ304107A (no) |
| PL (1) | PL322647A1 (no) |
| PT (1) | PT819002E (no) |
| TW (1) | TW450816B (no) |
| WO (1) | WO1996031210A1 (no) |
| ZA (1) | ZA962711B (no) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7632517B2 (en) * | 1997-10-01 | 2009-12-15 | Novadel Pharma Inc. | Buccal, polar and non-polar spray containing zolpidem |
| US6333345B1 (en) | 1999-05-14 | 2001-12-25 | Sepracor, Inc. | Methods of using and compositions comprising N-desmethylzolpidem |
| US6399621B1 (en) | 1999-08-10 | 2002-06-04 | American Cyanamid Company | N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1, 5-α]-pyrimidin-7-yl}phenyl)acetamide and compositions and methods related thereto |
| US20030091632A1 (en) * | 1999-08-26 | 2003-05-15 | Neurocrine Biosciences, Inc. | Controlled-release sedative-hypnotic compositions and methods related thereto |
| US6485746B1 (en) | 2000-08-25 | 2002-11-26 | Neurocrine Biosciences, Inc. | Controlled-release sedative-hypnotic compositions and methods related thereto |
| US6384221B1 (en) | 1999-09-02 | 2002-05-07 | Neurocrine Biosciences, Inc. | Polymorphs of N-methyl-N-(3-{3-[2-thienylcarbonyl]-pyrazol-[1,5-α]-pyrimidin-7-yl}phenyl)acetamide and compositions and methods related thereto |
| AU5066101A (en) * | 2000-04-13 | 2001-10-30 | Synthon B.V. | Modified release formulations containing a hypnotic agent |
| PT1475093E (pt) * | 2000-04-24 | 2006-11-30 | Teva Pharma | Hemitartarato de zolpidem micronizado |
| DE10041478A1 (de) * | 2000-08-24 | 2002-03-14 | Sanol Arznei Schwarz Gmbh | Neue pharmazeutische Zusammensetzung |
| DE10117183A1 (de) * | 2001-04-05 | 2002-10-10 | Gruenenthal Gmbh | Verwendung von substituierten Imidazo[1,2-a]-pyridinverbindungen als Arzneimittel |
| GB0311457D0 (en) * | 2003-05-19 | 2003-06-25 | Sciencom Ltd | New therapeutic use |
| EP1624867A1 (en) * | 2003-05-19 | 2006-02-15 | Sciencom Ltd | Further therapeutic use of zolpidem |
| DE10334187A1 (de) * | 2003-07-26 | 2005-03-03 | Schwarz Pharma Ag | Substituierte 2-Aminotetraline zur Behandlung von Depressionen |
| DE10334188B4 (de) | 2003-07-26 | 2007-07-05 | Schwarz Pharma Ag | Verwendung von Rotigotin zur Behandlung von Depressionen |
| DK1691811T3 (da) | 2003-12-11 | 2014-10-20 | Sunovion Pharmaceuticals Inc | Kombination af et sedativ og en neurotransmittermodulator og fremgangsmåder til forbedring af søvnkvaliteten og behandling af depression |
| DE10361258A1 (de) | 2003-12-24 | 2005-07-28 | Schwarz Pharma Ag | Verwendung von substituierten 2-Aminotetralinen zur vorbeugenden Behandlung von Morbus Parkinson |
| WO2005079851A2 (en) | 2004-02-18 | 2005-09-01 | Sepracor, Inc. | Dopamine-agonist combination therapy with sedatives for improving sleep quality |
| DE102004014841B4 (de) * | 2004-03-24 | 2006-07-06 | Schwarz Pharma Ag | Verwendung von Rotigotin zur Behandlung und Prävention des Parkinson-Plus-Syndroms |
| AU2006322314A1 (en) * | 2005-11-18 | 2007-06-14 | Synthon B.V. | Zolpidem tablets |
| GB2443928A (en) * | 2006-11-08 | 2008-05-21 | Regen Therapeutics Plc | Transdermal pharmaceutical composition comprising Zolpidem |
| GB0809936D0 (en) * | 2008-05-30 | 2008-07-09 | Regen Therapeutics Plc | Therapeutic use of zolpidem |
| WO2017214442A1 (en) | 2016-06-08 | 2017-12-14 | President And Fellows Of Harvard College | Methods and compositions for reducing tactile dysfunction and anxiety associated with autism spectrum disorder, rett syndrome, and fragile x syndrome |
| CA3099751A1 (en) | 2018-05-22 | 2019-11-28 | President And Fellows Of Harvard College | Compositions and methods for reducing tactile dysfunction, anxiety, and social impairment |
| EP3801512A4 (en) | 2018-05-29 | 2022-01-19 | President and Fellows of Harvard College | COMPOSITIONS AND METHODS TO REDUCE TACTILE DYSFUNCTION, ANXIETY AND SOCIAL DISABILITIES |
| WO2020198275A1 (en) | 2019-03-25 | 2020-10-01 | President And Fellows Of Harvard College | Compositions and methods for reducing tactile dysfunction, anxiety, and social impairment |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2492382A1 (fr) * | 1980-10-22 | 1982-04-23 | Synthelabo | Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique |
| US5032595A (en) * | 1989-11-24 | 1991-07-16 | Fidia-Georgetown Institute For The Neurosciences | Method of stimulating steroidogenesis with alpidem |
| US5206382A (en) * | 1991-06-27 | 1993-04-27 | Fidia Georgetown Institute For The Neurosciences | Indole derivatives, pharmaceutical compositions and methods of treating neurological and psychiatric disorders |
-
1995
- 1995-04-07 IT IT95RM000223A patent/IT1276522B1/it active IP Right Grant
-
1996
- 1996-04-02 AU AU51200/96A patent/AU707759B2/en not_active Ceased
- 1996-04-02 EA EA199700308A patent/EA000396B1/ru not_active IP Right Cessation
- 1996-04-02 NZ NZ304107A patent/NZ304107A/xx not_active IP Right Cessation
- 1996-04-02 JP JP53016596A patent/JP4049390B2/ja not_active Expired - Fee Related
- 1996-04-02 US US08/930,644 patent/US5891891A/en not_active Expired - Lifetime
- 1996-04-02 CA CA002217590A patent/CA2217590C/en not_active Expired - Lifetime
- 1996-04-02 DK DK96907656T patent/DK0819002T3/da active
- 1996-04-02 CZ CZ19973167A patent/CZ292020B6/cs not_active IP Right Cessation
- 1996-04-02 PT PT96907656T patent/PT819002E/pt unknown
- 1996-04-02 DE DE69623271T patent/DE69623271T2/de not_active Expired - Lifetime
- 1996-04-02 CN CNB961937815A patent/CN1198612C/zh not_active Expired - Fee Related
- 1996-04-02 MX MX9707712A patent/MX9707712A/es unknown
- 1996-04-02 PL PL96322647A patent/PL322647A1/xx unknown
- 1996-04-02 KR KR1019970707107A patent/KR100425628B1/ko not_active Expired - Fee Related
- 1996-04-02 WO PCT/IT1996/000063 patent/WO1996031210A1/en not_active Ceased
- 1996-04-02 HU HU9900733A patent/HUP9900733A3/hu unknown
- 1996-04-02 ES ES96907656T patent/ES2182967T3/es not_active Expired - Lifetime
- 1996-04-02 AT AT96907656T patent/ATE222763T1/de active
- 1996-04-02 EP EP96907656A patent/EP0819002B1/en not_active Expired - Lifetime
- 1996-04-03 IL IL11782496A patent/IL117824A/xx not_active IP Right Cessation
- 1996-04-04 ZA ZA962711A patent/ZA962711B/xx unknown
- 1996-04-08 AR ARP960102094A patent/AR003414A1/es unknown
- 1996-04-15 TW TW085104484A patent/TW450816B/zh not_active IP Right Cessation
-
1997
- 1997-10-06 NO NO19974603A patent/NO315408B1/no not_active IP Right Cessation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |