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NO332971B1 - Forbedret produksjon av rosuvastatin kalsiumsalt - Google Patents

Forbedret produksjon av rosuvastatin kalsiumsalt

Info

Publication number
NO332971B1
NO332971B1 NO20055730A NO20055730A NO332971B1 NO 332971 B1 NO332971 B1 NO 332971B1 NO 20055730 A NO20055730 A NO 20055730A NO 20055730 A NO20055730 A NO 20055730A NO 332971 B1 NO332971 B1 NO 332971B1
Authority
NO
Norway
Prior art keywords
water
aqueous
isopropyl
solution
calcium salt
Prior art date
Application number
NO20055730A
Other languages
English (en)
Norwegian (no)
Other versions
NO20055730D0 (no
NO20055730L (no
Inventor
Nigel Phillip Taylor
John Horbury
Jeffrey Norman Crabb
Original Assignee
Astrazeneca Uk Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33512687&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO332971(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Uk Ltd filed Critical Astrazeneca Uk Ltd
Publication of NO20055730D0 publication Critical patent/NO20055730D0/no
Publication of NO20055730L publication Critical patent/NO20055730L/no
Publication of NO332971B1 publication Critical patent/NO332971B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO20055730A 2003-06-05 2005-12-05 Forbedret produksjon av rosuvastatin kalsiumsalt NO332971B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0312896.4A GB0312896D0 (en) 2003-06-05 2003-06-05 Chemical process
GBGB0324793.9A GB0324793D0 (en) 2003-06-05 2003-10-24 Chemical process
PCT/GB2004/002373 WO2004108691A1 (en) 2003-06-05 2004-06-03 Improved production of rosuvastatin calcium salt

Publications (3)

Publication Number Publication Date
NO20055730D0 NO20055730D0 (no) 2005-12-05
NO20055730L NO20055730L (no) 2005-12-27
NO332971B1 true NO332971B1 (no) 2013-02-11

Family

ID=33512687

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20055730A NO332971B1 (no) 2003-06-05 2005-12-05 Forbedret produksjon av rosuvastatin kalsiumsalt

Country Status (25)

Country Link
US (1) US8063213B2 (is)
EP (1) EP1633727B1 (is)
JP (1) JP4651615B2 (is)
KR (1) KR101099934B1 (is)
CN (1) CN100422157C (is)
AR (1) AR044773A1 (is)
AT (1) ATE464297T1 (is)
AU (1) AU2004245291B2 (is)
BR (1) BRPI0410922B8 (is)
CA (1) CA2527314C (is)
CO (1) CO5640116A2 (is)
DE (1) DE602004026576D1 (is)
ES (1) ES2341858T3 (is)
GB (2) GB0312896D0 (is)
IL (1) IL172075A (is)
IS (1) IS2751B (is)
MX (1) MXPA05013128A (is)
MY (1) MY140820A (is)
NO (1) NO332971B1 (is)
NZ (1) NZ543962A (is)
RU (1) RU2361864C2 (is)
SA (1) SA04250223B1 (is)
TW (1) TWI341310B (is)
UY (1) UY28341A1 (is)
WO (1) WO2004108691A1 (is)

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Also Published As

Publication number Publication date
RU2361864C2 (ru) 2009-07-20
NZ543962A (en) 2008-09-26
KR101099934B1 (ko) 2011-12-28
MY140820A (en) 2010-01-29
TW200510337A (en) 2005-03-16
ATE464297T1 (de) 2010-04-15
WO2004108691A1 (en) 2004-12-16
DE602004026576D1 (de) 2010-05-27
IS8217A (is) 2006-01-02
CN1798741A (zh) 2006-07-05
HK1087405A1 (en) 2006-10-13
CA2527314A1 (en) 2004-12-16
NO20055730D0 (no) 2005-12-05
AR044773A1 (es) 2005-10-05
JP2006526602A (ja) 2006-11-24
BRPI0410922B8 (pt) 2021-05-25
EP1633727A1 (en) 2006-03-15
US20080221323A1 (en) 2008-09-11
BRPI0410922A (pt) 2006-06-27
AU2004245291A1 (en) 2004-12-16
NO20055730L (no) 2005-12-27
BRPI0410922B1 (pt) 2016-02-23
JP4651615B2 (ja) 2011-03-16
CO5640116A2 (es) 2006-05-31
CN100422157C (zh) 2008-10-01
IS2751B (is) 2011-09-15
RU2005138370A (ru) 2006-07-10
UY28341A1 (es) 2005-01-31
ES2341858T3 (es) 2010-06-29
GB0312896D0 (en) 2003-07-09
TWI341310B (en) 2011-05-01
SA04250223B1 (ar) 2008-12-23
KR20060017848A (ko) 2006-02-27
EP1633727B1 (en) 2010-04-14
MXPA05013128A (es) 2006-03-16
AU2004245291B2 (en) 2008-02-14
CA2527314C (en) 2012-02-21
IL172075A (en) 2011-06-30
GB0324793D0 (en) 2003-11-26
US8063213B2 (en) 2011-11-22

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