NO20091234L - Polymorfine krystallformer av et indan-2-ylamino-hydroksyetyl-kinolinonmaleatderivat som beta-adrenoceptoragonist - Google Patents
Polymorfine krystallformer av et indan-2-ylamino-hydroksyetyl-kinolinonmaleatderivat som beta-adrenoceptoragonistInfo
- Publication number
- NO20091234L NO20091234L NO20091234A NO20091234A NO20091234L NO 20091234 L NO20091234 L NO 20091234L NO 20091234 A NO20091234 A NO 20091234A NO 20091234 A NO20091234 A NO 20091234A NO 20091234 L NO20091234 L NO 20091234L
- Authority
- NO
- Norway
- Prior art keywords
- indan
- ylamino
- hydroxyethyl
- polymorphine
- quinolinone
- Prior art date
Links
- 239000013078 crystal Substances 0.000 title abstract 5
- GYPMLKARJPBKQB-BTJKTKAUSA-N OC(=O)\C=C/C(O)=O.C12=CC=CC=C2NC(=O)C(CCO)=C1NC1CC2=CC=CC=C2C1 Chemical class OC(=O)\C=C/C(O)=O.C12=CC=CC=C2NC(=O)C(CCO)=C1NC1CC2=CC=CC=C2C1 GYPMLKARJPBKQB-BTJKTKAUSA-N 0.000 title 1
- 239000000048 adrenergic agonist Substances 0.000 title 1
- 102000015005 beta-adrenergic receptor activity proteins Human genes 0.000 title 1
- 108040006818 beta-adrenergic receptor activity proteins Proteins 0.000 title 1
- IREJFXIHXRZFER-PCBAQXHCSA-N indacaterol maleate Chemical compound OC(=O)\C=C/C(O)=O.N1C(=O)C=CC2=C1C(O)=CC=C2[C@@H](O)CNC1CC(C=C(C(=C2)CC)CC)=C2C1 IREJFXIHXRZFER-PCBAQXHCSA-N 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000000414 obstructive effect Effects 0.000 abstract 1
- 208000023504 respiratory system disease Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/24—Oxygen atoms attached in position 8
- C07D215/26—Alcohols; Ethers thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4704—2-Quinolinones, e.g. carbostyril
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/14—Antitussive agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Vascular Medicine (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Otolaryngology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Quinoline Compounds (AREA)
- Medicinal Preparation (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06119895A EP1914227A1 (en) | 2006-08-31 | 2006-08-31 | Polymorphic crystal form of a indan-2-ylamino-hydroxyethyl-quinolinone maleate derivative as beta-adrenoceptor agonist |
| PCT/EP2007/059039 WO2008025816A1 (en) | 2006-08-31 | 2007-08-30 | Polymorphic crystal form of a indan-2-ylamino-hydroxyethyl-quinolinone maleate derivative as beta-adrenoceptor agonist |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20091234L true NO20091234L (no) | 2009-03-30 |
Family
ID=37714644
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20091234A NO20091234L (no) | 2006-08-31 | 2009-03-24 | Polymorfine krystallformer av et indan-2-ylamino-hydroksyetyl-kinolinonmaleatderivat som beta-adrenoceptoragonist |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US20100010039A1 (ru) |
| EP (2) | EP1914227A1 (ru) |
| JP (1) | JP2010501631A (ru) |
| KR (1) | KR20090049615A (ru) |
| CN (1) | CN101511794A (ru) |
| AR (1) | AR063698A1 (ru) |
| AU (1) | AU2007291270A1 (ru) |
| BR (1) | BRPI0716383A2 (ru) |
| CA (1) | CA2659144A1 (ru) |
| CL (1) | CL2007002525A1 (ru) |
| GT (1) | GT200900037A (ru) |
| IL (1) | IL196805A0 (ru) |
| MA (1) | MA30763B1 (ru) |
| MX (1) | MX2009002301A (ru) |
| NO (1) | NO20091234L (ru) |
| PE (1) | PE20080923A1 (ru) |
| RU (1) | RU2009111389A (ru) |
| TN (1) | TN2009000056A1 (ru) |
| TW (1) | TW200817333A (ru) |
| WO (1) | WO2008025816A1 (ru) |
| ZA (1) | ZA200900264B (ru) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2481738A1 (en) * | 2009-09-25 | 2012-08-01 | Kyorin Pharmaceutical Co., Ltd. | Maleic acid salt and crystal thereof |
| ES2626829T3 (es) | 2013-03-27 | 2017-07-26 | Laboratorios Lesvi, S.L. | Procedimiento para la fabricación de (R)-5[2-(5,6-dietil-indan-2-ilamino)-1-hidroxietil]-8-hidroxi-(1H)-quinolin-2-ona |
| CN103830195A (zh) * | 2014-03-11 | 2014-06-04 | 熊妲妮 | 一种茚达特罗片及其制备方法 |
| CN103830193A (zh) * | 2014-03-11 | 2014-06-04 | 熊妲妮 | 茚达特罗片制剂及其制备方法 |
| EP3347345B1 (en) | 2015-09-29 | 2019-07-31 | Inke, S.A. | Mixed solvate of (r)-5-[2-(5,6-diethylindan-2-ylamino)-1-hydroxyethyl]-8-hydroxy-1h-quinolin-2-one l-tartrate |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9913083D0 (en) * | 1999-06-04 | 1999-08-04 | Novartis Ag | Organic compounds |
| GB0413960D0 (en) * | 2004-06-22 | 2004-07-28 | Novartis Ag | Organic compounds |
-
2006
- 2006-08-31 EP EP06119895A patent/EP1914227A1/en not_active Ceased
-
2007
- 2007-08-28 PE PE2007001166A patent/PE20080923A1/es not_active Application Discontinuation
- 2007-08-29 AR ARP070103832A patent/AR063698A1/es unknown
- 2007-08-30 EP EP07803048A patent/EP2066639A1/en not_active Withdrawn
- 2007-08-30 US US12/438,407 patent/US20100010039A1/en not_active Abandoned
- 2007-08-30 MX MX2009002301A patent/MX2009002301A/es not_active Application Discontinuation
- 2007-08-30 RU RU2009111389/04A patent/RU2009111389A/ru not_active Application Discontinuation
- 2007-08-30 CA CA002659144A patent/CA2659144A1/en not_active Abandoned
- 2007-08-30 TW TW096132295A patent/TW200817333A/zh unknown
- 2007-08-30 AU AU2007291270A patent/AU2007291270A1/en not_active Withdrawn
- 2007-08-30 WO PCT/EP2007/059039 patent/WO2008025816A1/en not_active Ceased
- 2007-08-30 CN CNA2007800319674A patent/CN101511794A/zh active Pending
- 2007-08-30 BR BRPI0716383-5A2A patent/BRPI0716383A2/pt not_active Application Discontinuation
- 2007-08-30 CL CL200702525A patent/CL2007002525A1/es unknown
- 2007-08-30 KR KR1020097006531A patent/KR20090049615A/ko not_active Withdrawn
- 2007-08-30 JP JP2009526104A patent/JP2010501631A/ja active Pending
-
2009
- 2009-01-13 ZA ZA200900264A patent/ZA200900264B/xx unknown
- 2009-01-29 IL IL196805A patent/IL196805A0/en unknown
- 2009-02-20 TN TN2009000056A patent/TN2009000056A1/fr unknown
- 2009-02-20 GT GT200900037A patent/GT200900037A/es unknown
- 2009-03-13 MA MA31713A patent/MA30763B1/fr unknown
- 2009-03-24 NO NO20091234A patent/NO20091234L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EP1914227A1 (en) | 2008-04-23 |
| RU2009111389A (ru) | 2010-10-10 |
| KR20090049615A (ko) | 2009-05-18 |
| MA30763B1 (fr) | 2009-10-01 |
| IL196805A0 (en) | 2009-11-18 |
| TN2009000056A1 (en) | 2010-08-19 |
| ZA200900264B (en) | 2010-05-26 |
| CN101511794A (zh) | 2009-08-19 |
| CL2007002525A1 (es) | 2008-07-11 |
| TW200817333A (en) | 2008-04-16 |
| BRPI0716383A2 (pt) | 2013-09-24 |
| CA2659144A1 (en) | 2008-03-06 |
| AU2007291270A1 (en) | 2008-03-06 |
| JP2010501631A (ja) | 2010-01-21 |
| GT200900037A (es) | 2010-03-11 |
| WO2008025816A1 (en) | 2008-03-06 |
| PE20080923A1 (es) | 2008-07-11 |
| US20100010039A1 (en) | 2010-01-14 |
| MX2009002301A (es) | 2009-03-20 |
| EP2066639A1 (en) | 2009-06-10 |
| AR063698A1 (es) | 2009-02-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |