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NO20090173L - Kondensert spiroketalderivat og anvendelse derav som legemiddel for a behandle diabetes - Google Patents

Kondensert spiroketalderivat og anvendelse derav som legemiddel for a behandle diabetes

Info

Publication number
NO20090173L
NO20090173L NO20090173A NO20090173A NO20090173L NO 20090173 L NO20090173 L NO 20090173L NO 20090173 A NO20090173 A NO 20090173A NO 20090173 A NO20090173 A NO 20090173A NO 20090173 L NO20090173 L NO 20090173L
Authority
NO
Norway
Prior art keywords
condensed
drug
treating diabetes
spiroketal derivative
spiroketal
Prior art date
Application number
NO20090173A
Other languages
English (en)
Inventor
Takashi Emura
Tsutomu Sato
Masahiro Nishimoto
Takamitsu Kobayashi
Yoshihito Ohtake
Marina Yamaguchi
Kyouko Takami
Original Assignee
Chugai Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38981587&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20090173(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Chugai Pharmaceutical Co Ltd filed Critical Chugai Pharmaceutical Co Ltd
Publication of NO20090173L publication Critical patent/NO20090173L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)

Abstract

Foreliggende oppfinnelse angår forbindelser som har formelen (I) hvori X, Y, U, A, B, W, Z, RI og R2 er som definert i beskrivelsen. Fremgangsmåte for fremstilling og anvendelse i terapeutiske midler.
NO20090173A 2006-07-27 2009-01-12 Kondensert spiroketalderivat og anvendelse derav som legemiddel for a behandle diabetes NO20090173L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006205242 2006-07-27
PCT/JP2007/064802 WO2008013277A1 (en) 2006-07-27 2007-07-27 Fused ring spiroketal derivative and use thereof as drug for treating diabetes

Publications (1)

Publication Number Publication Date
NO20090173L true NO20090173L (no) 2009-04-27

Family

ID=38981587

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20090173A NO20090173L (no) 2006-07-27 2009-01-12 Kondensert spiroketalderivat og anvendelse derav som legemiddel for a behandle diabetes

Country Status (18)

Country Link
US (1) US8207134B2 (no)
EP (1) EP2048152A4 (no)
JP (1) JP5165565B2 (no)
KR (1) KR20090033911A (no)
CN (1) CN101495494A (no)
AR (1) AR062110A1 (no)
AU (1) AU2007277704A1 (no)
BR (1) BRPI0715248A2 (no)
CA (1) CA2658921A1 (no)
CL (1) CL2007002186A1 (no)
IL (1) IL196585A0 (no)
MX (1) MX2009000579A (no)
NO (1) NO20090173L (no)
PE (1) PE20080521A1 (no)
RU (1) RU2009106866A (no)
TW (1) TWI432446B (no)
WO (1) WO2008013277A1 (no)
ZA (1) ZA200900706B (no)

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BRPI0918841B8 (pt) 2008-08-28 2021-05-25 Pfizer derivados de dioxa-biciclo[3.2.1]octano-2,3,4-triol, seus cristais, composições farmacêuticas e usos
SI2496583T1 (sl) 2009-11-02 2015-02-27 Pfizer Inc. Derivati dioksa-biciklo(3.2.1)oktan-2,3,4-triola
AR079438A1 (es) 2009-12-09 2012-01-25 Panacea Biotec Ltd Derivados de azucar, composiciones farmaceuticas y sus usos
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2582709B1 (de) 2010-06-18 2018-01-24 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
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WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
CN104987314A (zh) * 2015-07-14 2015-10-21 佛山市赛维斯医药科技有限公司 含苯并异恶唑和末端硝基苄基类结构的化合物及其用途
CN105001174A (zh) * 2015-07-14 2015-10-28 佛山市赛维斯医药科技有限公司 含苯并异恶唑和末端腈基苄基类结构的化合物及其用途
CN110483476B (zh) * 2019-08-15 2020-11-27 绍兴文理学院 一种催化法制备苯并硒吩类化合物的工艺
CN110483475B (zh) * 2019-08-15 2020-11-27 绍兴文理学院 一种氧化银催化法制备苯并噻吩类化合物的方法
CN112574226A (zh) * 2020-12-15 2021-03-30 海门华祥医药科技有限公司 5,6-亚甲基二氧基吲哚的制备方法
CN116178143B (zh) * 2021-11-26 2024-10-01 中国科学院大连化学物理研究所 一种1,4-萘二甲酸/酯、1,4-萘二甲酸衍生物及其制备方法和应用
CN117050126A (zh) * 2023-08-15 2023-11-14 南京华威医药科技集团有限公司 一种新的托格列净关键异构体制备方法

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Also Published As

Publication number Publication date
WO2008013277A1 (en) 2008-01-31
CL2007002186A1 (es) 2008-02-01
IL196585A0 (en) 2009-11-18
KR20090033911A (ko) 2009-04-06
RU2009106866A (ru) 2010-09-10
AR062110A1 (es) 2008-10-15
PE20080521A1 (es) 2008-06-13
JPWO2008013277A1 (ja) 2009-12-17
US20100234609A1 (en) 2010-09-16
US8207134B2 (en) 2012-06-26
EP2048152A1 (en) 2009-04-15
TWI432446B (zh) 2014-04-01
AU2007277704A1 (en) 2008-01-31
ZA200900706B (en) 2010-05-26
JP5165565B2 (ja) 2013-03-21
TW200821323A (en) 2008-05-16
CN101495494A (zh) 2009-07-29
EP2048152A4 (en) 2013-01-23
MX2009000579A (es) 2009-01-27
CA2658921A1 (en) 2008-01-31
BRPI0715248A2 (pt) 2013-06-04

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