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NO20083003L - Anvendelse av benzofuserte heterocykliske sulfamidderivater for a senke lipider og blodglykosenivaer - Google Patents

Anvendelse av benzofuserte heterocykliske sulfamidderivater for a senke lipider og blodglykosenivaer

Info

Publication number
NO20083003L
NO20083003L NO20083003A NO20083003A NO20083003L NO 20083003 L NO20083003 L NO 20083003L NO 20083003 A NO20083003 A NO 20083003A NO 20083003 A NO20083003 A NO 20083003A NO 20083003 L NO20083003 L NO 20083003L
Authority
NO
Norway
Prior art keywords
blood glucose
glucose levels
sulfamide derivatives
benzofused heterocyclic
lowering lipids
Prior art date
Application number
NO20083003A
Other languages
English (en)
Inventor
Allen B Reitz
Virginia L Smith-Swintosky
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NO20083003L publication Critical patent/NO20083003L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

Foreliggende oppfinnelse er en fremgangsmåte for glukoserelaterte forstyrrelser og lipidrelaterte forstyrrelser som innbefatter administrering til et subjekt som trenger det av en terapeutisk effektiv mengde av ett eller flere nye benzosammensmeltede hererosyklussulfamidderivater med formel (I) eller formel (II) som definert heri. Foreliggende oppfinnelse angår videre fremgangsmåter for behandling som innbefatter samtidig behandling med et anti-diabetisk middel og anti-lipidmiddel og/eller en anti-fedmemiddel.
NO20083003A 2005-12-19 2008-07-03 Anvendelse av benzofuserte heterocykliske sulfamidderivater for a senke lipider og blodglykosenivaer NO20083003L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US75167705P 2005-12-19 2005-12-19
US11/611,961 US8497298B2 (en) 2005-12-19 2006-12-18 Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
PCT/US2006/048477 WO2007092086A2 (en) 2005-12-19 2006-12-19 Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels

Publications (1)

Publication Number Publication Date
NO20083003L true NO20083003L (no) 2008-09-18

Family

ID=38225368

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20083003A NO20083003L (no) 2005-12-19 2008-07-03 Anvendelse av benzofuserte heterocykliske sulfamidderivater for a senke lipider og blodglykosenivaer

Country Status (24)

Country Link
US (1) US8497298B2 (no)
EP (1) EP1973541B1 (no)
JP (1) JP5190374B2 (no)
KR (1) KR101363332B1 (no)
CN (1) CN101365441B (no)
AT (1) ATE486595T1 (no)
AU (1) AU2006337617B8 (no)
BR (1) BRPI0620011A2 (no)
CA (1) CA2634419C (no)
CR (1) CR10169A (no)
CY (1) CY1111161T1 (no)
DE (1) DE602006018066D1 (no)
DK (1) DK1973541T3 (no)
EA (2) EA016892B1 (no)
HR (1) HRP20110008T1 (no)
IL (1) IL192101A (no)
MY (1) MY148866A (no)
NO (1) NO20083003L (no)
NZ (1) NZ569043A (no)
PL (1) PL1973541T3 (no)
PT (1) PT1973541E (no)
RS (1) RS51521B (no)
SI (1) SI1973541T1 (no)
WO (1) WO2007092086A2 (no)

Families Citing this family (16)

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MY147767A (en) 2004-06-16 2013-01-31 Janssen Pharmaceutica Nv Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders
AU2006249577A1 (en) * 2005-05-20 2006-11-30 Janssen Pharmaceutica N.V. Process for preparation of sulfamide derivatives
US8691867B2 (en) 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
US8937096B2 (en) 2005-12-19 2015-01-20 Janssen Pharmaceutica Nv Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder
US20070155827A1 (en) * 2005-12-19 2007-07-05 Smith-Swintosky Virginia L Use of benzo-fused heterocycle sulfamide derivatives for the treatment of depression
US8497298B2 (en) 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
AU2007253814A1 (en) 2006-05-19 2007-11-29 Janssen Pharmaceutica N.V. Co-therapy for the treatment of epilepsy
US20090247616A1 (en) * 2008-03-26 2009-10-01 Smith-Swintosky Virginia L Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety
US20090247617A1 (en) * 2008-03-26 2009-10-01 Abdel-Magid Ahmed F Process for the preparation of benzo-fused heteroaryl sulfamates
EA018567B1 (ru) 2008-06-23 2013-08-30 Янссен Фармацевтика Нв Кристаллическая форма (2s)-(-)-n-(6-хлор-2,3-дигидробензо[1,4]диоксин-2-илметил)сульфамида
US8815939B2 (en) * 2008-07-22 2014-08-26 Janssen Pharmaceutica Nv Substituted sulfamide derivatives
WO2013045681A1 (en) 2011-09-29 2013-04-04 Janssen Pharmaceutica Nv Improved process for the preparation of sulfamide derivatives
JP2014528953A (ja) 2011-09-29 2014-10-30 ヤンセン ファーマシューティカ エヌ．ベー． スルファミド誘導体の調製プロセス
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CN105232543A (zh) * 2015-11-11 2016-01-13 朱忠良 一种抗糖尿病的口服药物组合物
CN105232544A (zh) * 2015-11-11 2016-01-13 朱忠良 一种抗糖尿病的口服药物组合物

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DK1973541T3 (da) 2011-02-14
EA016892B1 (ru) 2012-08-30
ATE486595T1 (de) 2010-11-15
IL192101A0 (en) 2009-08-03
RS51521B (sr) 2011-06-30
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EP1973541B1 (en) 2010-11-03
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SI1973541T1 (sl) 2011-02-28
AU2006337617A1 (en) 2007-08-16
EA015606B1 (ru) 2011-10-31
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EA200870088A1 (ru) 2009-02-27
IL192101A (en) 2013-03-24
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US8497298B2 (en) 2013-07-30
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CR10169A (es) 2009-01-14
JP2009520032A (ja) 2009-05-21
BRPI0620011A2 (pt) 2011-10-25
EA201000630A1 (ru) 2010-10-29
WO2007092086A3 (en) 2007-09-27
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