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NO20072854L - Acylerte nonadepsipeptider anvendt som lysobaktinderivater - Google Patents

Acylerte nonadepsipeptider anvendt som lysobaktinderivater

Info

Publication number
NO20072854L
NO20072854L NO20072854A NO20072854A NO20072854L NO 20072854 L NO20072854 L NO 20072854L NO 20072854 A NO20072854 A NO 20072854A NO 20072854 A NO20072854 A NO 20072854A NO 20072854 L NO20072854 L NO 20072854L
Authority
NO
Norway
Prior art keywords
nonadepsipeptides
acylated
derivatives
lysobactin
lysobactin derivatives
Prior art date
Application number
NO20072854A
Other languages
English (en)
Inventor
Rainer Endermann
Franz Von Nussbaum
Guido Schiffer
Nina Brunner
Chantal Fuerstner
Elke Hartmann
Holger Paulsen
Jacques Ragot
Joachim Schumacher
Niels Svenstrup
Joachim Telser
Sonja Anlauf
Michael-Alexander Bruening
Original Assignee
Aicuris Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aicuris Gmbh & Co Kg filed Critical Aicuris Gmbh & Co Kg
Publication of NO20072854L publication Critical patent/NO20072854L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

Det beskrives nonadepsipeptider (lysobaktinderivater) og fremgangsmåter for deres fremstilling samt deres anvendelse for fremstilling av legemidler for terapi og/eller profylakse av sykdommer og særlig bakterie- eller infeksjonssykdommer. De nye lysobaktinderivater skiller seg fra naturstoffer ved den N-terminale peptidkjede som omfatter en 3-(3-pyridyl)-alanyl-rest.
NO20072854A 2004-11-05 2007-06-05 Acylerte nonadepsipeptider anvendt som lysobaktinderivater NO20072854L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004053407A DE102004053407A1 (de) 2004-11-05 2004-11-05 Acylierte Nonadepsipeptide II
PCT/EP2005/011363 WO2006048139A1 (de) 2004-11-05 2005-10-22 Acylierte nonadepsipeptide als lysobactinderivate

Publications (1)

Publication Number Publication Date
NO20072854L true NO20072854L (no) 2007-08-01

Family

ID=35462537

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20072854A NO20072854L (no) 2004-11-05 2007-06-05 Acylerte nonadepsipeptider anvendt som lysobaktinderivater

Country Status (27)

Country Link
US (1) US7531507B2 (no)
EP (1) EP1807443A1 (no)
JP (1) JP4843614B2 (no)
KR (1) KR20070083984A (no)
CN (1) CN101056887A (no)
AR (1) AR053775A1 (no)
AU (1) AU2005300815B2 (no)
BR (1) BRPI0516677A (no)
CA (1) CA2586704A1 (no)
CR (1) CR9079A (no)
DE (1) DE102004053407A1 (no)
GT (1) GT200500308A (no)
HN (1) HN2005030779A (no)
IL (1) IL182739A (no)
MA (1) MA29218B1 (no)
MX (1) MX2007005382A (no)
MY (1) MY145448A (no)
NO (1) NO20072854L (no)
NZ (1) NZ554813A (no)
PE (1) PE20060942A1 (no)
RU (1) RU2414477C2 (no)
SV (1) SV2006002290A (no)
TW (1) TW200621799A (no)
UA (1) UA89800C2 (no)
UY (1) UY29189A1 (no)
WO (1) WO2006048139A1 (no)
ZA (1) ZA200703674B (no)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004051025A1 (de) * 2004-10-20 2006-04-27 Bayer Healthcare Ag Substituierte Nonadepsipeptide
DE102004051024A1 (de) * 2004-10-20 2006-04-27 Bayer Healthcare Ag Heterocyclyl-substituierte Nonadepsipeptide
DE102004051023A1 (de) * 2004-10-20 2006-05-04 Bayer Healthcare Ag Desoxo-Nonadepsipeptide
DE102004053410A1 (de) * 2004-11-05 2006-05-11 Bayer Healthcare Ag Cyclische Nonadepsipeptidamide
DE102006003443A1 (de) * 2006-01-25 2007-07-26 Aicuris Gmbh & Co. Kg Asparagin-10-substituierte Nonadepsipeptide
DE102006018080A1 (de) * 2006-04-13 2007-10-18 Aicuris Gmbh & Co. Kg Lysobactinamide
DE102006018250A1 (de) * 2006-04-13 2007-10-18 Aicuris Gmbh & Co. Kg Verfahren zum Herstellen von cyclischen Depsipeptiden
TW201717991A (zh) * 2015-08-17 2017-06-01 拜耳動物保健有限公司 用於治療牛乳房炎之溶桿菌素
US10100066B2 (en) * 2015-10-23 2018-10-16 Navitor Pharmaceuticals, Inc. Modulators of sestrin-GATOR2 interaction and uses thereof
EP3363452A1 (en) * 2017-02-17 2018-08-22 Bayer Animal Health GmbH Combinations of lysobactin and aminogylcosides against diseases caused by gram-positive and gram-negative bacteria in non-human animals
AU2018258355B2 (en) 2017-04-26 2024-05-30 Navitor Pharmaceuticals, Inc. Modulators of sestrin-gator2 interaction and uses thereof
WO2021087432A1 (en) 2019-11-01 2021-05-06 Navitor Pharmaceuticals, Inc. Methods of treatment using an mtorc1 modulator

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1266247C (en) 1985-03-25 1990-02-27 ANTIBIOTIC PREPARED BY LYSOBACTER SP. SC14.067
JPH01132600A (ja) 1987-11-17 1989-05-25 Shionogi & Co Ltd カタノシンａおよびｂならびにその製造法
DE10320781A1 (de) * 2003-05-09 2004-11-25 Bayer Healthcare Ag Acylierte Nonadepsipeptide

Also Published As

Publication number Publication date
US7531507B2 (en) 2009-05-12
AU2005300815B2 (en) 2011-05-19
ZA200703674B (en) 2008-09-25
GT200500308A (es) 2006-06-02
PE20060942A1 (es) 2006-10-20
JP4843614B2 (ja) 2011-12-21
UA89800C2 (en) 2010-03-10
HN2005030779A (es) 2010-08-19
MA29218B1 (fr) 2008-02-01
MY145448A (en) 2012-02-15
MX2007005382A (es) 2007-08-14
DE102004053407A1 (de) 2006-05-11
WO2006048139A1 (de) 2006-05-11
CA2586704A1 (en) 2006-05-11
CN101056887A (zh) 2007-10-17
CR9079A (es) 2007-08-28
RU2007120686A (ru) 2008-12-10
IL182739A0 (en) 2007-07-24
EP1807443A1 (de) 2007-07-18
JP2008518982A (ja) 2008-06-05
BRPI0516677A (pt) 2008-09-16
TW200621799A (en) 2006-07-01
US20060264358A1 (en) 2006-11-23
AU2005300815A1 (en) 2006-05-11
IL182739A (en) 2013-03-24
SV2006002290A (es) 2006-10-13
UY29189A1 (es) 2006-06-30
AR053775A1 (es) 2007-05-23
KR20070083984A (ko) 2007-08-24
RU2414477C2 (ru) 2011-03-20
NZ554813A (en) 2009-11-27

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