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NO20070742L - Progesteron reseptormodulatorer inneholdende pyrrol-oksindolderivater og deres anvendelse. - Google Patents

Progesteron reseptormodulatorer inneholdende pyrrol-oksindolderivater og deres anvendelse.

Info

Publication number
NO20070742L
NO20070742L NO20070742A NO20070742A NO20070742L NO 20070742 L NO20070742 L NO 20070742L NO 20070742 A NO20070742 A NO 20070742A NO 20070742 A NO20070742 A NO 20070742A NO 20070742 L NO20070742 L NO 20070742L
Authority
NO
Norway
Prior art keywords
progesterone receptor
receptor modulators
oxindole derivatives
containing pyrrole
modulators containing
Prior art date
Application number
NO20070742A
Other languages
English (en)
Inventor
Andrew Fensome
Jay E Wrobel
Casey Cameron Mccomas
Michael Anthony Marella
Edward George Melenski
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34979790&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20070742(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of NO20070742L publication Critical patent/NO20070742L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Pregnancy & Childbirth (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Det er tilveiebrakt pyrroloksindol-derivater som er anvendelige som progesteronreseptor-antagonister, og metoder for fremstilling av disse. Det er beskrevet farmasøytiske preparater som inneholder disse derivatene, samt anvendelsen av disse som prevensjon og mot hormonrelaterte lidelser.
NO20070742A 2004-08-09 2007-02-08 Progesteron reseptormodulatorer inneholdende pyrrol-oksindolderivater og deres anvendelse. NO20070742L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US60003104P 2004-08-09 2004-08-09
US67168405P 2005-04-15 2005-04-15
PCT/US2005/023795 WO2006023109A1 (en) 2004-08-09 2005-07-06 Progesterone receptor modulators comprising pyrrole-oxindole derivatives and uses thereof

Publications (1)

Publication Number Publication Date
NO20070742L true NO20070742L (no) 2007-05-07

Family

ID=34979790

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20070742A NO20070742L (no) 2004-08-09 2007-02-08 Progesteron reseptormodulatorer inneholdende pyrrol-oksindolderivater og deres anvendelse.

Country Status (20)

Country Link
US (2) US7317037B2 (no)
EP (1) EP1776107A1 (no)
JP (1) JP2008509217A (no)
KR (1) KR20070039567A (no)
AR (1) AR049706A1 (no)
AU (1) AU2005277881A1 (no)
BR (1) BRPI0514180A (no)
CA (1) CA2573314A1 (no)
CR (1) CR8847A (no)
EC (1) ECSP077233A (no)
GT (1) GT200500185A (no)
IL (1) IL181043A0 (no)
MX (1) MX2007001608A (no)
NO (1) NO20070742L (no)
PA (1) PA8638801A1 (no)
PE (1) PE20060486A1 (no)
RU (1) RU2007101303A (no)
SV (1) SV2006002167A (no)
TW (1) TW200607798A (no)
WO (1) WO2006023109A1 (no)

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Also Published As

Publication number Publication date
MX2007001608A (es) 2007-04-10
AR049706A1 (es) 2006-08-30
US7317037B2 (en) 2008-01-08
JP2008509217A (ja) 2008-03-27
CA2573314A1 (en) 2006-03-02
IL181043A0 (en) 2007-07-04
KR20070039567A (ko) 2007-04-12
ECSP077233A (es) 2007-03-29
US20060030717A1 (en) 2006-02-09
TW200607798A (en) 2006-03-01
BRPI0514180A (pt) 2008-06-03
US20080114050A1 (en) 2008-05-15
PA8638801A1 (es) 2006-06-02
SV2006002167A (es) 2006-03-15
PE20060486A1 (es) 2006-07-06
CR8847A (es) 2007-08-28
EP1776107A1 (en) 2007-04-25
WO2006023109A1 (en) 2006-03-02
RU2007101303A (ru) 2008-09-20
AU2005277881A1 (en) 2006-03-02
GT200500185A (es) 2006-04-10

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