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NO20031521D0 - Assosiasjon av CB1-reseptorantagonist og et sibutramin, farmasöytiske preparater inneholdende denne samt dens anvendelse for behandling avfedme - Google Patents

Assosiasjon av CB1-reseptorantagonist og et sibutramin, farmasöytiske preparater inneholdende denne samt dens anvendelse for behandling avfedme

Info

Publication number
NO20031521D0
NO20031521D0 NO20031521A NO20031521A NO20031521D0 NO 20031521 D0 NO20031521 D0 NO 20031521D0 NO 20031521 A NO20031521 A NO 20031521A NO 20031521 A NO20031521 A NO 20031521A NO 20031521 D0 NO20031521 D0 NO 20031521D0
Authority
NO
Norway
Prior art keywords
association
receptor antagonist
obesity
sibutramine
treatment
Prior art date
Application number
NO20031521A
Other languages
English (en)
Other versions
NO20031521L (no
Inventor
Odile Piot-Grosjean
Philippe Picaut
Francois Petitet
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8854974&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20031521(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of NO20031521D0 publication Critical patent/NO20031521D0/no
Publication of NO20031521L publication Critical patent/NO20031521L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20031521A 2000-10-04 2003-04-03 Assosiasjon av CB1-reseptorantagonist og et sibutramin, farmasöytiske preparater inneholdende denne samt dens anvendelse for behandling avfedme NO20031521L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0012646A FR2814678B1 (fr) 2000-10-04 2000-10-04 Association d'un antagoniste du recepteur cb1 et de sibutramine, les compositions pharmaceutiques les contenant et leur utilisation pour la traitement de l'obesite
PCT/FR2001/003022 WO2002028346A2 (fr) 2000-10-04 2001-10-01 Association d'un antagoniste du recepteur cb1 et de sibutramine, pour le traitement de l'obesite

Publications (2)

Publication Number Publication Date
NO20031521D0 true NO20031521D0 (no) 2003-04-03
NO20031521L NO20031521L (no) 2003-04-24

Family

ID=8854974

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20031521A NO20031521L (no) 2000-10-04 2003-04-03 Assosiasjon av CB1-reseptorantagonist og et sibutramin, farmasöytiske preparater inneholdende denne samt dens anvendelse for behandling avfedme

Country Status (29)

Country Link
EP (1) EP1328269B2 (no)
JP (1) JP4221221B2 (no)
KR (1) KR20030036885A (no)
CN (1) CN100409845C (no)
AT (1) ATE267595T1 (no)
AU (2) AU9393601A (no)
BG (1) BG107739A (no)
BR (1) BR0114410A (no)
CA (1) CA2424934A1 (no)
DE (1) DE60103556T3 (no)
DK (1) DK1328269T5 (no)
EA (1) EA005924B1 (no)
EE (1) EE200300121A (no)
ES (1) ES2217191T5 (no)
FR (1) FR2814678B1 (no)
HR (1) HRP20030249A2 (no)
HU (1) HUP0302044A3 (no)
IL (1) IL155236A0 (no)
MX (1) MXPA03002845A (no)
NO (1) NO20031521L (no)
NZ (1) NZ524904A (no)
PL (1) PL362833A1 (no)
PT (1) PT1328269E (no)
SI (1) SI1328269T2 (no)
SK (1) SK4032003A3 (no)
TR (1) TR200401264T4 (no)
WO (1) WO2002028346A2 (no)
YU (1) YU26103A (no)
ZA (1) ZA200303015B (no)

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AU2003223510B2 (en) 2002-04-12 2008-05-08 Merck Sharp & Dohme Corp. Bicyclic amides
ES2301833T3 (es) 2002-07-29 2008-07-01 Hoffmann La Roche Derivados de benzodioxol.
ATE450505T1 (de) 2003-01-02 2009-12-15 Hoffmann La Roche Cb 1 rezeptor inversagonisten
ATE400571T1 (de) 2003-01-02 2008-07-15 Hoffmann La Roche Pyrrolyl-thiazole und ihre verwendung als inverse agonisten des cb 1 rezeptors
US7329658B2 (en) * 2003-02-06 2008-02-12 Pfizer Inc Cannabinoid receptor ligands and uses thereof
US20040224962A1 (en) * 2003-05-09 2004-11-11 Pfizer Inc Pharmaceutical composition for the treatment of obesity or to facilitate or promote weight loss
KR20060019587A (ko) 2003-06-11 2006-03-03 머크 앤드 캄파니 인코포레이티드 치환된 3-알킬 및 3-알케닐 아제티딘 유도체
ATE390922T1 (de) 2003-06-20 2008-04-15 Hoffmann La Roche 2-aminobenzothiazole als cb1 rezeptor inverse agonisten
EP1498122A1 (en) * 2003-07-18 2005-01-19 Aventis Pharma S.A. Semi-solid systems containing azetidine derivatives
EP1498123A1 (en) * 2003-07-18 2005-01-19 Aventis Pharma S.A. Emulsifying systems containing azetidine derivatives
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FR2861303A1 (fr) * 2003-10-24 2005-04-29 Sanofi Synthelabo Utilisation d'un derive de pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement du syndrome metabolique
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CN100509808C (zh) 2003-12-08 2009-07-08 霍夫曼-拉罗奇有限公司 新型噻唑衍生物
BRPI0507120A (pt) 2004-01-28 2007-06-19 Hoffmann La Roche compostos, processo para a manufatura dos mesmos, composições farmacêuticas que os compreendem, método para o tratamento e/ou profilaxia de enfermidades que estão associadas com a modulação de receptores de cb1 e sua utilização
ATE432275T1 (de) 2004-05-10 2009-06-15 Hoffmann La Roche Pyrrol- bzw. imidazolamide zur behandlung von obesitas
US20060025448A1 (en) 2004-07-22 2006-02-02 Cadila Healthcare Limited Hair growth stimulators
CA2581596A1 (en) * 2004-09-29 2006-04-13 Schering Corporation Combinations of substituted azetidonones and cb1 antagonists
FR2876689B1 (fr) 2004-10-14 2008-02-22 Aventis Pharma Sa Nouveau procede et intermediaires de preparation de derives de n-(1-benzhydryl-azetidin-3-yl)-n-phenyl-methylsulfonamide
WO2006045799A2 (en) 2004-10-25 2006-05-04 Solvay Pharmaceuticals Gmbh Pharmaceutical compositions comprising cb1 cannabinoid receptor antagonists and potassium channel openers for the treatment of diabetes mellitus type i, obesity and related conditions
JP2008517959A (ja) 2004-10-27 2008-05-29 エフ．ホフマン−ラ ロシュ アーゲー 新規なインドール又はベンゾイミダゾール誘導体
JP4675969B2 (ja) 2004-11-09 2011-04-27 エフ．ホフマン−ラ ロシュ アーゲー ジベンゾスベロン誘導体
ES2326280T3 (es) 2005-04-06 2009-10-06 F. Hoffmann-La Roche Ag Derivados de piridin-3-carboxamida como agonistas inversos de cb1.
US7906652B2 (en) 2005-11-28 2011-03-15 Merck Sharp & Dohme Corp. Heterocycle-substituted 3-alkyl azetidine derivatives
JP2009528999A (ja) * 2006-02-21 2009-08-13 アンプラ ファーマシューティカルズ インコーポレイテッド Ｃｂ１アンタゴニストおよび逆アゴニスト
WO2007110449A1 (en) * 2006-03-29 2007-10-04 Euro-Celtique S.A. Benzenesulfonamide compounds and their use
WO2007118853A1 (en) 2006-04-13 2007-10-25 Euro-Celtique S.A. Benzenesulfonamide compounds and their use as blockers of calcium channels
TW200812963A (en) 2006-04-13 2008-03-16 Euro Celtique Sa Benzenesulfonamide compounds and the use thereof
US7629346B2 (en) 2006-06-19 2009-12-08 Hoffmann-La Roche Inc. Pyrazinecarboxamide derivatives as CB1 antagonists
WO2008038143A2 (en) * 2006-06-22 2008-04-03 Medichem, S.A. Novel solid forms of rimonabant and synthetic processes for their preparation
WO2008026219A2 (en) * 2006-09-01 2008-03-06 Hetero Drugs Limited Novel polymorphs of rimonabant
US7781593B2 (en) 2006-09-14 2010-08-24 Hoffmann-La Roche Inc. 5-phenyl-nicotinamide derivatives
MX2009002888A (es) * 2006-09-25 2009-03-31 Boehringer Ingelheim Int Compuestos que modulan el receptor cb2.
DE102007002260A1 (de) 2007-01-16 2008-07-31 Sanofi-Aventis Verwendung von substituierten Pyranonsäurederivaten zur Herstellung von Medikamenten zur Behandlung des Metabolischen Syndroms
EP1953144A1 (en) * 2007-01-30 2008-08-06 Sandoz AG Novel polymorphic forms of N-piperidino-5-(4-chlorophenyl)-1-(2, 4-dichlorphenyl)-4-methyl-3-pyrazolecarboxamide
WO2008124118A1 (en) 2007-04-09 2008-10-16 Purdue Pharma L.P. Benzenesulfonyl compounds and the use therof
US8765736B2 (en) 2007-09-28 2014-07-01 Purdue Pharma L.P. Benzenesulfonamide compounds and the use thereof
PE20091270A1 (es) * 2007-12-18 2009-09-23 Sanofi Aventis Derivados de azetidinas con actividad sobre receptores cb1 y su preparacion
WO2010079241A1 (es) 2009-01-12 2010-07-15 Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion Uso de antagonistas y/o agonistas inversos de los receptores cb1 para la preparación de medicamentos que incrementen la excitabilidad de las motoneuronas
BRPI0902481B8 (pt) 2009-07-31 2021-05-25 Soc Beneficente De Senhoras Hospital Sirio Libanes composição farmacêutica compreendendo hemopressina e seu uso.
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Also Published As

Publication number Publication date
DE60103556T2 (de) 2005-06-30
BG107739A (bg) 2004-01-30
DK1328269T5 (da) 2009-03-16
NO20031521L (no) 2003-04-24
MXPA03002845A (es) 2004-09-10
CN1473040A (zh) 2004-02-04
FR2814678B1 (fr) 2002-12-20
AU2001293936B2 (en) 2007-01-25
JP4221221B2 (ja) 2009-02-12
HUP0302044A3 (en) 2005-05-30
WO2002028346A2 (fr) 2002-04-11
ATE267595T1 (de) 2004-06-15
YU26103A (sh) 2006-08-17
HRP20030249A2 (en) 2005-02-28
EP1328269B2 (fr) 2008-07-30
DK1328269T4 (da) 2008-11-24
EA200300441A1 (ru) 2003-08-28
SI1328269T2 (sl) 2008-12-31
JP2004512279A (ja) 2004-04-22
PT1328269E (pt) 2004-08-31
EP1328269B1 (fr) 2004-05-26
ES2217191T5 (es) 2009-02-16
FR2814678A1 (fr) 2002-04-05
CN100409845C (zh) 2008-08-13
EP1328269A2 (fr) 2003-07-23
HUP0302044A2 (hu) 2003-11-28
DE60103556T3 (de) 2009-04-09
AU9393601A (en) 2002-04-15
ES2217191T3 (es) 2004-11-01
SK4032003A3 (en) 2003-09-11
BR0114410A (pt) 2004-02-17
DE60103556D1 (de) 2004-07-01
ZA200303015B (en) 2004-02-26
NZ524904A (en) 2004-11-26
SI1328269T1 (en) 2004-10-31
CA2424934A1 (fr) 2002-04-11
EE200300121A (et) 2005-04-15
TR200401264T4 (tr) 2004-07-21
KR20030036885A (ko) 2003-05-09
WO2002028346A3 (fr) 2002-08-29
EA005924B1 (ru) 2005-08-25
IL155236A0 (en) 2003-11-23
DK1328269T3 (da) 2004-09-20
PL362833A1 (en) 2004-11-02

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