NO20015865D0 - Pyrrolidinyl-, piperidinyl- eller homopiperidinyl=substituerte (benzodioksan, benzofuran ellerbenzopyran) derivater - Google Patents

Pyrrolidinyl-, piperidinyl- eller homopiperidinyl=substituerte (benzodioksan, benzofuran ellerbenzopyran) derivater

Info

Publication number: NO20015865D0
Authority: NO; Norway
Prior art keywords: benzodioxane; homopiperidinyl; benzopyran; benzofuran; pyrrolidinyl
Prior art date: 1999-06-02

Application number

NO20015865A

Other languages

English (en)

Other versions

NO319950B1 (no

NO20015865L (no

Inventor

Marcel Frans Leopold De Bruyn

Kristof Van Emelen

Piet Tom Bert Paul Wigerinck

Wim Gaston Verschueren

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-06-02

Filing date

2001-11-30

Publication date

2001-11-30

2001-11-30 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2001-11-30 Publication of NO20015865D0 publication Critical patent/NO20015865D0/no

2002-02-01 Publication of NO20015865L publication Critical patent/NO20015865L/no

2005-10-03 Publication of NO319950B1 publication Critical patent/NO319950B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Public Health (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Nutrition Science (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

NO20015865A 1999-06-02 2001-11-30 Pyrrolidinyl- eller piperidinyl-substituerte kromanderivater, deres fremstilling og farmasoytiske sammensetninger omfattende disse samt deres anvendelse. NO319950B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP99201746		1999-06-02
PCT/EP2000/004747 WO2000075137A1 (en)	1999-06-02	2000-05-23	Pyrrolidinyl, piperidinyl or homopiperidinyl substituted (benzodioxan, benzofuran or benzopyran) derivatives

Publications (3)

Publication Number	Publication Date
NO20015865D0 true NO20015865D0 (no)	2001-11-30
NO20015865L NO20015865L (no)	2002-02-01
NO319950B1 NO319950B1 (no)	2005-10-03

Family

ID=8240259

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20015865A NO319950B1 (no)	1999-06-02	2001-11-30	Pyrrolidinyl- eller piperidinyl-substituerte kromanderivater, deres fremstilling og farmasoytiske sammensetninger omfattende disse samt deres anvendelse.

Country Status (30)

Country	Link
US (2)	US6900222B1 (no)
EP (1)	EP1187831B1 (no)
JP (1)	JP2003501428A (no)
KR (1)	KR100702526B1 (no)
CN (1)	CN1131862C (no)
AR (1)	AR033645A1 (no)
AT (1)	ATE279409T1 (no)
AU (1)	AU777601B2 (no)
BG (1)	BG65278B1 (no)
BR (1)	BR0011247A (no)
CA (1)	CA2374905C (no)
CZ (1)	CZ20014167A3 (no)
DE (1)	DE60014896T2 (no)
EA (1)	EA004648B1 (no)
EE (1)	EE04720B1 (no)
ES (1)	ES2231189T3 (no)
HR (1)	HRP20010869A2 (no)
HU (1)	HUP0201344A3 (no)
IL (1)	IL146824A0 (no)
MX (1)	MXPA01012323A (no)
MY (1)	MY120617A (no)
NO (1)	NO319950B1 (no)
NZ (1)	NZ515478A (no)
PL (1)	PL198532B1 (no)
SK (1)	SK286159B6 (no)
TR (1)	TR200103433T2 (no)
TW (1)	TW575571B (no)
UA (1)	UA73123C2 (no)
WO (1)	WO2000075137A1 (no)
ZA (1)	ZA200109863B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PL198552B1 (pl)	1999-06-02	2008-06-30	Janssen Pharmaceutica Nv	Pochodna benzopiranu podstawionego aminoalkilem i sposób jej otrzymywania oraz kompozycja farmaceutyczna i sposób jej otrzymywania
JO2352B1 (en) *	2000-06-22	2006-12-12	جانسين فارماسيوتيكا ان. في	Compounds for the treatment of non-adaptation of the bottom of the uterus
JO2654B1 (en)	2000-09-04	2012-06-17	شركة جانسين فارماسوتيكا ان. في	Multiple aryl caroxa amides are useful as lipid - lowering agents
JO2409B1 (en)	2000-11-21	2007-06-17	شركة جانسين فارماسوتيكا ان. في	Second-phenyl carboxy amides are useful as lipid-lowering agents
ATE527247T1 (de) *	2001-07-05	2011-10-15	Takeda Pharmaceutical	Benzokondensierte 5gliedrige heterocyclische verbindungen, verfahren zu deren herstellung und deren verwendung
HUE026904T2 (en)	2003-04-24	2016-08-29	Incyte Holdings Corp	Aza-spiroalkane derivatives as inhibitors of metalloproteases
CN1696115B (zh) *	2004-05-11	2010-06-09	中国科学院上海药物研究所	合成砌块4-取代基-4-氨基-哌啶衍生物、其制备方法和用途
GB201612938D0 (en)	2016-07-26	2016-09-07	Almac Discovery Ltd	Pharmaceutical compounds

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US19051A (en) *		1858-01-05		sloan
US3910930A (en)	1973-01-04	1975-10-07	Janssen Pharmaceutica Nv	1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones
US3929801A (en)	1973-11-20	1975-12-30	Janssen Pharmaceutica Nv	2-Benzimidazolinones
GR71865B (no)	1978-03-20	1983-07-07	Ciba Geigy
ES469096A1 (es)	1978-04-24	1978-11-16	Antibioticos Sa	Un procedimiento para la preparacion dos sustancialmente insolubles en agua.
DE2852945A1 (de)	1978-12-07	1980-06-26	Boehringer Sohn Ingelheim	Benzodioxanyl-hydroxyaethylpiperidyl- imidazolidinone, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
US4329348A (en)	1979-02-26	1982-05-11	Ciba-Geigy Corporation	N-Oxacyclic-alkylpiperidines as psychostimulants
DE3124366A1 (de)	1981-06-20	1982-12-30	Hoechst Ag, 6000 Frankfurt	N-oxacyclyl-alkylpiperidin-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und deren verwendung
FR2533584B1 (fr)	1982-09-28	1986-03-21	Pasteur Institut	Procede de detection du pouvoir mutagene de substances, susceptibles d'induire la deterioration d'adn cellulaires, mettant en jeu la production d'une reponse sos
DE3901814A1 (de)	1988-07-28	1990-02-01	Bayer Ag	Substituierte aminomethylzetraline sowie ihre heterocyclischen analoga
DE4140540A1 (de) *	1991-12-09	1993-06-17	Bayer Ag	Neue azaheterocyclylmethyl-chromane
SI9300097B (en)	1992-02-27	2001-12-31	Janssen Pharmaceutica Nv	(benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines
DE4319038A1 (de)	1993-06-08	1994-12-15	Bayer Ag	Verwendung von teilweise bekannten substituierten Chromanen als Arzneimittel, neue Wirkstoffe und Verfahren zu ihrer Herstellung
WO1995005383A1 (en)	1993-08-19	1995-02-23	Janssen Pharmaceutica N.V.	Vasocontrictive dihydrobenzopyran derivatives
US5541199A (en)	1995-06-02	1996-07-30	American Home Products Corporation	Chroman-2-ylmethylamino derivatives
FR2744451B1 (fr)	1996-02-01	1998-04-24	Pf Medicament	Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique
US6133277A (en)	1997-12-05	2000-10-17	Janssen Pharmaceutica N.V.	(Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
PL198552B1 (pl)	1999-06-02	2008-06-30	Janssen Pharmaceutica Nv	Pochodna benzopiranu podstawionego aminoalkilem i sposób jej otrzymywania oraz kompozycja farmaceutyczna i sposób jej otrzymywania
JO2352B1 (en)	2000-06-22	2006-12-12	جانسين فارماسيوتيكا ان. في	Compounds for the treatment of non-adaptation of the bottom of the uterus

2000
- 2000-05-23 HU HU0201344A patent/HUP0201344A3/hu unknown
- 2000-05-23 US US09/980,451 patent/US6900222B1/en not_active Expired - Lifetime
- 2000-05-23 KR KR1020017014585A patent/KR100702526B1/ko not_active Expired - Fee Related
- 2000-05-23 AT AT00927243T patent/ATE279409T1/de not_active IP Right Cessation
- 2000-05-23 AU AU45685/00A patent/AU777601B2/en not_active Ceased
- 2000-05-23 CZ CZ20014167A patent/CZ20014167A3/cs unknown
- 2000-05-23 EA EA200101237A patent/EA004648B1/ru not_active IP Right Cessation
- 2000-05-23 EE EEP200100640A patent/EE04720B1/xx not_active IP Right Cessation
- 2000-05-23 TR TR2001/03433T patent/TR200103433T2/xx unknown
- 2000-05-23 MX MXPA01012323A patent/MXPA01012323A/es active IP Right Grant
- 2000-05-23 IL IL14682400A patent/IL146824A0/xx not_active IP Right Cessation
- 2000-05-23 WO PCT/EP2000/004747 patent/WO2000075137A1/en not_active Ceased
- 2000-05-23 CN CN008083177A patent/CN1131862C/zh not_active Expired - Fee Related
- 2000-05-23 UA UA2001128826A patent/UA73123C2/uk unknown
- 2000-05-23 HR HR20010869A patent/HRP20010869A2/hr not_active Application Discontinuation
- 2000-05-23 JP JP2001502420A patent/JP2003501428A/ja not_active Withdrawn
- 2000-05-23 NZ NZ515478A patent/NZ515478A/xx unknown
- 2000-05-23 EP EP00927243A patent/EP1187831B1/en not_active Expired - Lifetime
- 2000-05-23 SK SK1692-2001A patent/SK286159B6/sk not_active IP Right Cessation
- 2000-05-23 BR BR0011247-0A patent/BR0011247A/pt not_active Application Discontinuation
- 2000-05-23 DE DE60014896T patent/DE60014896T2/de not_active Expired - Lifetime
- 2000-05-23 ES ES00927243T patent/ES2231189T3/es not_active Expired - Lifetime
- 2000-05-23 PL PL352063A patent/PL198532B1/pl not_active IP Right Cessation
- 2000-05-23 CA CA2374905A patent/CA2374905C/en not_active Expired - Lifetime
- 2000-05-24 TW TW89109976A patent/TW575571B/zh not_active IP Right Cessation
- 2000-05-30 MY MYPI20002410A patent/MY120617A/en unknown
- 2000-06-01 AR ARP000102715A patent/AR033645A1/es active IP Right Grant
2001
- 2001-11-28 BG BG106157A patent/BG65278B1/bg unknown
- 2001-11-29 ZA ZA200109863A patent/ZA200109863B/xx unknown
- 2001-11-30 NO NO20015865A patent/NO319950B1/no not_active IP Right Cessation
2005
- 2005-03-14 US US11/079,606 patent/US7358239B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
PL352063A1 (en)	2003-07-28
ZA200109863B (en)	2003-05-28
US20050159406A1 (en)	2005-07-21
DE60014896D1 (de)	2004-11-18
EP1187831A1 (en)	2002-03-20
KR100702526B1 (ko)	2007-04-04
WO2000075137A1 (en)	2000-12-14
TR200103433T2 (tr)	2002-06-21
HUP0201344A2 (en)	2002-08-28
HUP0201344A3 (en)	2005-09-28
SK16922001A3 (sk)	2002-07-02
EE04720B1 (et)	2006-10-16
PL198532B1 (pl)	2008-06-30
TW575571B (en)	2004-02-11
CN1353708A (zh)	2002-06-12
EA004648B1 (ru)	2004-06-24
ATE279409T1 (de)	2004-10-15
CN1131862C (zh)	2003-12-24
CA2374905C (en)	2010-02-23
CZ20014167A3 (cs)	2002-06-12
NO319950B1 (no)	2005-10-03
BG65278B1 (bg)	2007-11-30
MXPA01012323A (es)	2002-07-22
US6900222B1 (en)	2005-05-31
MY120617A (en)	2005-11-30
UA73123C2 (en)	2005-06-15
NO20015865L (no)	2002-02-01
EA200101237A1 (ru)	2002-04-25
EP1187831B1 (en)	2004-10-13
CA2374905A1 (en)	2000-12-14
AR033645A1 (es)	2004-01-07
SK286159B6 (sk)	2008-04-07
US7358239B2 (en)	2008-04-15
BG106157A (en)	2002-06-28
DE60014896T2 (de)	2006-02-02
EE200100640A (et)	2003-02-17
HRP20010869A2 (en)	2003-08-31
ES2231189T3 (es)	2005-05-16
BR0011247A (pt)	2002-03-05
AU4568500A (en)	2000-12-28
KR20010113951A (ko)	2001-12-28
IL146824A0 (en)	2002-07-25
NZ515478A (en)	2003-03-28
JP2003501428A (ja)	2003-01-14
AU777601B2 (en)	2004-10-21

Publication	Publication Date	Title
DE60019577D1 (de)	2005-05-25	4, 5, 6, 7-tetrahydroindazolderivate als antitumormittel
FI20010154L (fi)	2001-02-09	Menetelmä citalopramin valmistamiseksi
ZA9811081B (en)	2000-06-22	(Benzodioxan, Benzofuran or Benzopyran) Derivatives having fundic relaxation properties.
FI20010155L (fi)	2001-02-09	Menetelmä citalopramin valmistamiseksi
DK1085976T3 (da)	2007-03-05	Ark dannet ud fra polyester, der indbefatter isosorbid
NO20006293L (no)	2001-02-13	Nye benzopyran eller tiobenzopyranderivater
FI20011621A7 (fi)	2002-02-19	Menetelmä sitalopraamin valmistamiseksi
KR950700288A (ko)	1995-01-16	5-에이취티4 길항제로서의 벤조피란, 벤조티오피란 및 벤조푸란 유도체(Benzopyran, benzothiopyran and benzofuran derivatives as 5-HT4 antagonists)
EP1078926A4 (en)	2002-02-04	Pyran derivatives
NO20015865D0 (no)	2001-11-30	Pyrrolidinyl-, piperidinyl- eller homopiperidinyl=substituerte (benzodioksan, benzofuran ellerbenzopyran) derivater
IL152893A0 (en)	2003-06-24	Novel benzofuran derivatives
ATE296818T1 (de)	2005-06-15	Substituierte 6h-dibenzo(c,h)chromene als oestrogene agentien
PT1140890E (pt)	2003-07-31	Derivados de cromano
NO20015903L (no)	2001-12-03	Aminoalkylsubstituerte (benzodioksan-, benzofuran eller benzopyran) derivater
DE50100383D1 (de)	2003-08-21	H-annellierte benzo [f]chromene
TR199802200A3 (tr)	1999-05-21	Sülfonamid sübstitüe edilmis benzopiran türevleri, üretilme yöntemi.
BR9706239B1 (pt)	2010-10-19	3-(1-hidroxifenil-1-alcoxiiminometil) dioxazinas bem como processos de preparação dos mesmos.
ATE273973T1 (de)	2004-09-15	Benzofuranderivate
NO20015652L (no)	2002-01-14	1-trifluorometyl-4-hydroksy-7-piperidinyl- aminometylkromanderivater
FI970833L (fi)	1997-02-27	Dihydro-2,3-bentsodiatsepiinijohdannaiset
PT1115708E (pt)	2004-08-31	Derivados aminoalquil-3,4-di-hidroquinolina como inibidores da sintetase do no
MA25693A1 (fr)	2003-04-01	Procede de stabilisation de compositions de blanchiment colorees.
IT1311346B1 (it)	2002-03-12	Macchina per spaccare legna da ardere.

Legal Events

Date	Code	Title	Description
2010-12-27	MM1K	Lapsed by not paying the annual fees