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NO20012465L - N-(4-(3-klor-4-fluor-fenylamino)-7-(3-morfolin-4-yl-propoksy)- kinazolin-6-yl)-akrylamid, en irreversibel inhibitor av tyrosin-kinaser - Google Patents

N-(4-(3-klor-4-fluor-fenylamino)-7-(3-morfolin-4-yl-propoksy)- kinazolin-6-yl)-akrylamid, en irreversibel inhibitor av tyrosin-kinaser

Info

Publication number
NO20012465L
NO20012465L NO20012465A NO20012465A NO20012465L NO 20012465 L NO20012465 L NO 20012465L NO 20012465 A NO20012465 A NO 20012465A NO 20012465 A NO20012465 A NO 20012465A NO 20012465 L NO20012465 L NO 20012465L
Authority
NO
Norway
Prior art keywords
quinazolin
morpholin
phenylamino
propoxy
acrylamide
Prior art date
Application number
NO20012465A
Other languages
English (en)
Other versions
NO319357B1 (no
NO20012465D0 (no
Inventor
Alexander James Bridges
Denise Driscoll
Wayne Daniel Klohs
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of NO20012465D0 publication Critical patent/NO20012465D0/no
Publication of NO20012465L publication Critical patent/NO20012465L/no
Publication of NO319357B1 publication Critical patent/NO319357B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20012465A 1998-11-19 2001-05-18 N-(4-(3-klor-4-fluor-fenylamino)-7-(3-morfolin-4-yl-propoksy)-kinazolin-6-yl)-akrylamid, en irreversibel inhibitor av tyrosin-kinaser NO319357B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10906598P 1998-11-19 1998-11-19
PCT/US1999/022116 WO2000031048A1 (en) 1998-11-19 1999-09-23 N-[4-(3-chloro-4-fluoro-phenylamino)-7-(3-morpholin-4-yl-propoxy)-quinazolin-6-yl]-acrylamide, an irreversible inhibitor of tyrosine kinases

Publications (3)

Publication Number Publication Date
NO20012465D0 NO20012465D0 (no) 2001-05-18
NO20012465L true NO20012465L (no) 2001-07-13
NO319357B1 NO319357B1 (no) 2005-07-18

Family

ID=22325607

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20012465A NO319357B1 (no) 1998-11-19 2001-05-18 N-(4-(3-klor-4-fluor-fenylamino)-7-(3-morfolin-4-yl-propoksy)-kinazolin-6-yl)-akrylamid, en irreversibel inhibitor av tyrosin-kinaser

Country Status (30)

Country Link
US (1) US6344455B1 (no)
EP (1) EP1131304B1 (no)
JP (1) JP3687900B2 (no)
KR (1) KR20010080491A (no)
CN (1) CN1160338C (no)
AR (1) AR023706A1 (no)
AT (1) ATE229008T1 (no)
AU (1) AU763626B2 (no)
BG (1) BG105608A (no)
BR (1) BR9915487A (no)
CA (1) CA2349721A1 (no)
CO (1) CO5150185A1 (no)
CZ (1) CZ20011759A3 (no)
DE (1) DE69904358T2 (no)
DK (1) DK1131304T3 (no)
EA (1) EA003786B1 (no)
EE (1) EE200100271A (no)
ES (1) ES2188254T3 (no)
GE (1) GEP20032997B (no)
HU (1) HUP0104211A3 (no)
IL (1) IL143089A0 (no)
NO (1) NO319357B1 (no)
NZ (2) NZ527718A (no)
PE (1) PE20001242A1 (no)
PL (1) PL347717A1 (no)
PT (1) PT1131304E (no)
SK (1) SK283688B6 (no)
UY (1) UY25809A1 (no)
WO (1) WO2000031048A1 (no)
ZA (1) ZA200103535B (no)

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