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NO20011351D0 - FremgangsmÕte for behandling av diabetes ved anvendelse av en AP2 inhibitor og kombinasjon derav - Google Patents

FremgangsmÕte for behandling av diabetes ved anvendelse av en AP2 inhibitor og kombinasjon derav

Info

Publication number
NO20011351D0
NO20011351D0 NO20011351A NO20011351A NO20011351D0 NO 20011351 D0 NO20011351 D0 NO 20011351D0 NO 20011351 A NO20011351 A NO 20011351A NO 20011351 A NO20011351 A NO 20011351A NO 20011351 D0 NO20011351 D0 NO 20011351D0
Authority
NO
Norway
Prior art keywords
inhibitor
combination
treating diabetes
pravastatin
employing
Prior art date
Application number
NO20011351A
Other languages
English (en)
Other versions
NO20011351L (no
Inventor
Jeffrey A Robl
Rex A Parker
Scott A Biller
Haris Amil
Bruce L Acobson
Krishna Odukula
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22280975&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20011351(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20011351D0 publication Critical patent/NO20011351D0/no
Publication of NO20011351L publication Critical patent/NO20011351L/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/4211,3-Oxazoles, e.g. pemoline, trimethadione
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Steroid Compounds (AREA)
  • Electrical Discharge Machining, Electrochemical Machining, And Combined Machining (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20011351A 1998-09-17 2001-03-16 Fremgangsmåte for behandling av diabetes ved anvendelse av en AP2 inhibitor og kombinasjon derav NO20011351L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10067798P 1998-09-17 1998-09-17
PCT/US1999/020946 WO2000015229A1 (en) 1998-09-17 1999-09-13 METHOD FOR TREATING DIABETES EMPLOYING AN aP2 INHIBITOR AND COMBINATION

Publications (2)

Publication Number Publication Date
NO20011351D0 true NO20011351D0 (no) 2001-03-16
NO20011351L NO20011351L (no) 2001-05-11

Family

ID=22280975

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20011352A NO20011352L (no) 1998-09-17 2001-03-16 Fremgangsmåte for behandling av aterosklerose ved anvendelse av en AP2 inhibitor og kombinasjon derav
NO20011351A NO20011351L (no) 1998-09-17 2001-03-16 Fremgangsmåte for behandling av diabetes ved anvendelse av en AP2 inhibitor og kombinasjon derav

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO20011352A NO20011352L (no) 1998-09-17 2001-03-16 Fremgangsmåte for behandling av aterosklerose ved anvendelse av en AP2 inhibitor og kombinasjon derav

Country Status (30)

Country Link
US (1) US20020035064A1 (no)
EP (2) EP1113801A4 (no)
JP (2) JP2002524517A (no)
KR (2) KR20010075150A (no)
CN (2) CN1319012A (no)
AT (1) ATE406898T1 (no)
AU (2) AU755563B2 (no)
BG (2) BG105431A (no)
BR (2) BR9913833A (no)
CA (2) CA2344309A1 (no)
CO (2) CO5130026A1 (no)
CZ (2) CZ2001965A3 (no)
DE (1) DE69939481D1 (no)
EE (2) EE200100155A (no)
ES (1) ES2311306T3 (no)
GE (2) GEP20033044B (no)
HU (2) HUP0104108A2 (no)
ID (2) ID27833A (no)
IL (2) IL141786A0 (no)
LT (2) LT4870B (no)
LV (2) LV12687B (no)
NO (2) NO20011352L (no)
NZ (2) NZ510207A (no)
PE (2) PE20001056A1 (no)
PL (2) PL346660A1 (no)
SK (1) SK3202001A3 (no)
TR (2) TR200100774T2 (no)
UY (2) UY25713A1 (no)
WO (2) WO2000015229A1 (no)
ZA (2) ZA200207430B (no)

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JP6514282B2 (ja) * 2014-03-24 2019-05-15 花王株式会社 Gip上昇抑制剤の評価又は選択方法
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WO2018005551A1 (en) * 2016-06-27 2018-01-04 President And Fellows Of Harvard College Compounds useful to treat metabolic disorders
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Also Published As

Publication number Publication date
LV12687B (lv) 2001-10-20
AU6143799A (en) 2000-04-03
LT2001022A (en) 2001-08-27
CZ2001965A3 (cs) 2002-02-13
PE20001047A1 (es) 2000-12-24
SK3202001A3 (en) 2002-04-04
BG105432A (en) 2001-12-29
DE69939481D1 (de) 2008-10-16
TR200100774T2 (tr) 2001-12-21
EP1121129A1 (en) 2001-08-08
UY25714A1 (es) 2001-08-27
WO2000015230A1 (en) 2000-03-23
EE04356B1 (et) 2004-10-15
HUP0104240A2 (hu) 2002-03-28
CN1319012A (zh) 2001-10-24
ID27833A (id) 2001-04-26
EP1113801A1 (en) 2001-07-11
BG105431A (en) 2001-12-29
LT2001023A (en) 2001-08-27
GEP20033044B (en) 2003-08-25
LV12686A (en) 2001-07-20
EP1113801A4 (en) 2002-10-02
NZ510207A (en) 2003-08-29
PE20001056A1 (es) 2000-12-24
CA2344300A1 (en) 2000-03-23
LT4871B (lt) 2001-12-27
LV12686B (lv) 2001-10-20
CZ2001964A3 (cs) 2002-01-16
AU6387799A (en) 2000-04-03
CN1317970A (zh) 2001-10-17
ID28450A (id) 2001-05-24
NO20011352D0 (no) 2001-03-16
LT4870B (lt) 2001-12-27
PL346661A1 (en) 2002-02-25
ES2311306T3 (es) 2009-02-01
NO20011352L (no) 2001-05-11
CO5130026A1 (es) 2002-02-27
JP2002524517A (ja) 2002-08-06
CA2344309A1 (en) 2000-03-23
CO5130025A1 (es) 2002-02-27
IL141786A0 (en) 2002-03-10
PL346660A1 (en) 2002-02-25
ATE406898T1 (de) 2008-09-15
KR20010079842A (ko) 2001-08-22
NO20011351L (no) 2001-05-11
US20020035064A1 (en) 2002-03-21
ZA200207433B (en) 2003-10-27
AU755563B2 (en) 2002-12-12
HUP0104108A2 (hu) 2002-03-28
NZ510209A (en) 2003-07-25
EE200100155A (et) 2002-08-15
WO2000015229A1 (en) 2000-03-23
BR9913833A (pt) 2001-05-29
KR20010075150A (ko) 2001-08-09
BR9913831A (pt) 2001-05-29
IL141785A0 (en) 2002-03-10
EP1121129A4 (en) 2002-10-16
UY25713A1 (es) 2001-08-27
ZA200207430B (en) 2003-09-16
GEP20033045B (en) 2003-08-25
JP2002524518A (ja) 2002-08-06
LV12687A (en) 2001-07-20
EE200100154A (et) 2002-12-16
AU754488B2 (en) 2002-11-14
EP1121129B1 (en) 2008-09-03
TR200100773T2 (tr) 2001-07-23

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