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NO20010319D0 - Fremgangsmåte for fremstilling av Citalopram - Google Patents

Fremgangsmåte for fremstilling av Citalopram

Info

Publication number
NO20010319D0
NO20010319D0 NO20010319A NO20010319A NO20010319D0 NO 20010319 D0 NO20010319 D0 NO 20010319D0 NO 20010319 A NO20010319 A NO 20010319A NO 20010319 A NO20010319 A NO 20010319A NO 20010319 D0 NO20010319 D0 NO 20010319D0
Authority
NO
Norway
Prior art keywords
citalopram
preparation
Prior art date
Application number
NO20010319A
Other languages
English (en)
Other versions
NO20010319L (no
NO328542B1 (no
Inventor
Hans Peterson
Michael Harold Rock
Henrik Svane
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of NO20010319D0 publication Critical patent/NO20010319D0/no
Publication of NO20010319L publication Critical patent/NO20010319L/no
Publication of NO328542B1 publication Critical patent/NO328542B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J23/00—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00
    • B01J23/38—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals
    • B01J23/40—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals of the platinum group metals
    • B01J23/44—Palladium
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/81—Radicals substituted by nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Materials Engineering (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Steroid Compounds (AREA)
NO20010319A 1999-06-25 2001-01-19 Fremgangsmate og forbindelse for fremstillingen av Citalopram NO328542B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA199900920 1999-06-25
PCT/DK1999/000640 WO2000013648A2 (en) 1999-06-25 1999-11-22 Method for the preparation of citalopram

Publications (3)

Publication Number Publication Date
NO20010319D0 true NO20010319D0 (no) 2001-01-19
NO20010319L NO20010319L (no) 2001-02-23
NO328542B1 NO328542B1 (no) 2010-03-15

Family

ID=8099035

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20010319A NO328542B1 (no) 1999-06-25 2001-01-19 Fremgangsmate og forbindelse for fremstillingen av Citalopram

Country Status (36)

Country Link
US (2) US20020077353A1 (no)
EP (1) EP1159274B1 (no)
JP (1) JP3447267B2 (no)
KR (1) KR100491368B1 (no)
CN (2) CN1140521C (no)
AR (1) AR020863A1 (no)
AT (3) ATE235478T1 (no)
AU (2) AU2001100440B4 (no)
BG (1) BG65574B1 (no)
BR (1) BR9917368B1 (no)
CA (2) CA2290127C (no)
CH (1) CH691305A5 (no)
CZ (1) CZ292198B6 (no)
DE (2) DE69906389T2 (no)
DK (2) DK1159274T3 (no)
EA (1) EA002560B1 (no)
ES (2) ES2194545T3 (no)
FI (1) FI108641B (no)
GB (2) GB2354239B (no)
HK (1) HK1049002B (no)
HU (1) HUP0103235A3 (no)
IL (2) IL145959A0 (no)
IS (1) IS2343B (no)
IT (1) ITMI991581A1 (no)
MX (1) MXPA01010989A (no)
NO (1) NO328542B1 (no)
NZ (1) NZ514979A (no)
PL (1) PL205579B1 (no)
PT (1) PT1159274E (no)
SE (1) SE516690C2 (no)
SI (1) SI1159274T1 (no)
SK (1) SK285813B6 (no)
TR (1) TR200103702T2 (no)
UA (1) UA63034C2 (no)
WO (1) WO2000013648A2 (no)
ZA (1) ZA200108854B (no)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200101796T2 (tr) 1998-12-23 2001-11-21 H. Lundbeck A/S 5-Siyanofitalitin preparasyonuna yönelik metot
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
AU759716B2 (en) 1999-04-14 2003-04-17 H. Lundbeck A/S Method for the preparation of citalopram
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
EP1228056B1 (en) 1999-10-25 2004-09-22 H. Lundbeck A/S Method for the preparation of citalopram
DE69920526T2 (de) 1999-10-25 2006-02-23 H. Lundbeck A/S Verfahren zur herstellung von citalopram
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
PT1246812E (pt) 1999-12-28 2004-08-31 Lundbeck & Co As H Metodo para a preparacao de citalopram
UA73336C2 (en) 1999-12-30 2005-07-15 Lundbeck & Co As H A method for the preparation of 5-cyano-phtalid
ES2206177T3 (es) 2000-01-14 2004-05-16 H. Lundbeck A/S Metodo para la preparacion de 5-cianoftalida.
FR2805812A1 (fr) 2000-02-24 2001-09-07 Lundbeck & Co As H Procede de preparation du citalopram
IES20010157A2 (en) 2000-03-03 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
GB2357762B (en) 2000-03-13 2002-01-30 Lundbeck & Co As H Crystalline base of citalopram
IL151490A0 (en) 2000-03-13 2003-04-10 Lundbeck & Co As H Method for the preparation of citalopram
NL1017500C1 (nl) 2000-03-13 2001-04-26 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
WO2001068629A1 (en) 2000-03-13 2001-09-20 H. Lundbeck A/S Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
DE60101786T2 (de) 2000-03-14 2004-07-15 H. Lundbeck A/S, Valby Verfahren zur herstellung von citalopram
PL360115A1 (en) * 2000-03-16 2004-09-06 H.Lundbeck A/S Method for the preparation of 5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
WO2002004435A1 (en) * 2000-07-06 2002-01-17 H. Lundbeck A/S Method for the preparation of citalopram
IL144816A (en) * 2000-08-18 2005-09-25 Lundbeck & Co As H Method for the preparation of citalopram
IL147226A (en) 2000-12-22 2006-04-10 Lundbeck & Co As H Process for the preparation of pure citalopram
PL353369A1 (en) * 2000-12-28 2003-11-17 H.Lundbeck A/S Process for the preparation of pure citalopram
WO2002060886A1 (en) 2001-01-30 2002-08-08 Orion Corporation, Fermion Process for the preparation of 1-(3-dimethylaminopropyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-carbonitrile
GB0105627D0 (en) * 2001-03-07 2001-04-25 Cipla Ltd Preparation of phthalanes
HUP0400095A3 (en) * 2001-03-09 2005-10-28 Ranbaxy Lab Ltd Process for the preparation of citalopram
US6967259B2 (en) * 2001-09-24 2005-11-22 Pharmachem Technologies Limited Process for the preparation of Citalopram intermediate
US7148364B2 (en) * 2002-01-07 2006-12-12 Sun Pharmaceutical Industries Process for the preparation of 1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3-dihydro-5-isobenzofuran carbonitrile
PE20040991A1 (es) 2002-08-12 2004-12-27 Lundbeck & Co As H Separacion de intermediarios para la preparacion de escitalopram
AU2003223105A1 (en) * 2003-03-24 2004-10-18 Hetero Drugs Limited Novel crystalline forms of (s)-citalopram oxalate
EP1486492A3 (en) 2003-06-10 2005-02-23 Sun Pharmaceuticals Industries Ltd. A process for hydrogenolysis of [1-(3-dimethylamino)propyl)]-1-(4-fluorophenyl)-1,3-dihydro-5-halo-isobenzofuran.
TWI339651B (en) 2004-02-12 2011-04-01 Lundbeck & Co As H Method for the separation of intermediates which may be used for the preparation of escitalopram
EP2141156A1 (en) 2004-08-23 2010-01-06 Sun Pharma Global FZE Process for Preparation of Citalopram and Enantiomers
US7834201B2 (en) 2005-06-22 2010-11-16 H. Lundbeck A/S Crystalline base of escitalopram and orodispersible tablets comprising escitalopram base
TWI347942B (en) 2005-06-22 2011-09-01 Lundbeck & Co As H Crystalline base of escitalopram and orodispersible tablets comprising escitalopram base
EP2017271A1 (en) 2007-07-06 2009-01-21 Aurobindo Pharma Limited Process for the preparation of escitalopram

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1143702A (no) * 1965-03-18
GB1526331A (en) * 1976-01-14 1978-09-27 Kefalas As Phthalanes
GB8419963D0 (en) * 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) * 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
US5296507A (en) * 1990-09-06 1994-03-22 H.Lundbeck A/S Treatment of cerbrovascular disorders
DK213290D0 (da) * 1990-09-06 1990-09-06 Lundbeck & Co As H Treatment of cerebrovascular disorders
DE19626659A1 (de) * 1996-07-03 1998-01-08 Basf Ag Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de) * 1996-07-10 1998-01-15 Basf Ag Verfahren zur Herstellung von Phthaliden
EA001728B1 (ru) * 1997-07-08 2001-08-27 Х.Лундбекк А/С Способ получения циталопрама
UA62985C2 (en) * 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
CZ292911B6 (cs) * 1997-11-11 2004-01-14 H. Lundbeck A/S Způsob výroby citalopramu
NZ510858A (en) * 1998-10-20 2003-11-28 H Method for the preparation of citalopram
TR200101796T2 (tr) * 1998-12-23 2001-11-21 H. Lundbeck A/S 5-Siyanofitalitin preparasyonuna yönelik metot
AR022329A1 (es) * 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
AU759716B2 (en) * 1999-04-14 2003-04-17 H. Lundbeck A/S Method for the preparation of citalopram
ITMI991579A1 (it) * 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
EP1228056B1 (en) * 1999-10-25 2004-09-22 H. Lundbeck A/S Method for the preparation of citalopram
AR026063A1 (es) * 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
FR2805812A1 (fr) * 2000-02-24 2001-09-07 Lundbeck & Co As H Procede de preparation du citalopram
IES20010143A2 (en) * 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
IL144816A (en) * 2000-08-18 2005-09-25 Lundbeck & Co As H Method for the preparation of citalopram
IL147226A (en) * 2000-12-22 2006-04-10 Lundbeck & Co As H Process for the preparation of pure citalopram
PL353369A1 (en) * 2000-12-28 2003-11-17 H.Lundbeck A/S Process for the preparation of pure citalopram

Also Published As

Publication number Publication date
HUP0103235A2 (hu) 2002-01-28
WO2000013648A3 (en) 2000-07-13
IS2343B (is) 2008-02-15
IL145959A0 (en) 2002-07-25
EA002560B1 (ru) 2002-06-27
AU1374500A (en) 2000-03-27
KR100491368B1 (ko) 2005-05-24
HK1049002A1 (en) 2003-04-25
US20090088469A1 (en) 2009-04-02
JP2002526386A (ja) 2002-08-20
AU2001100440A4 (en) 2001-11-01
ATA904199A (de) 2002-05-15
DK1159274T3 (da) 2003-07-21
ES2189699A1 (es) 2003-07-01
CZ292198B6 (cs) 2003-08-13
IL145959A (en) 2007-07-24
US20020077353A1 (en) 2002-06-20
NO20010319L (no) 2001-02-23
JP3447267B2 (ja) 2003-09-16
FI108641B (fi) 2002-02-28
SK18402001A3 (sk) 2002-06-04
FI20010155L (fi) 2001-02-09
SK285813B6 (sk) 2007-08-02
CZ2001320A3 (en) 2001-05-16
BG65574B1 (bg) 2009-01-30
CH691305A5 (de) 2001-06-29
AU2001100440B4 (en) 2002-01-24
SE516690C2 (sv) 2002-02-12
GB2357761B (en) 2001-09-05
WO2000013648A2 (en) 2000-03-16
UA63034C2 (en) 2004-01-15
AR020863A1 (es) 2002-05-29
PL346237A1 (en) 2002-01-28
WO2000013648B1 (en) 2001-03-15
MXPA01010989A (es) 2002-06-04
PT1159274E (pt) 2003-08-29
GB2354239A (en) 2001-03-21
BR9917368B1 (pt) 2010-02-09
GB0105182D0 (en) 2001-04-18
TR200103702T2 (tr) 2002-06-21
DE69906389T2 (de) 2003-10-30
GB2354239B (en) 2001-06-06
DE69906389D1 (de) 2003-04-30
NZ514979A (en) 2004-01-30
ITMI991581A0 (it) 1999-07-15
DK200100060A (da) 2001-04-10
KR20020012204A (ko) 2002-02-15
SE0100193L (sv) 2001-04-25
DE19983487C1 (de) 2002-07-25
NO328542B1 (no) 2010-03-15
ZA200108854B (en) 2002-08-28
ES2194545T3 (es) 2003-11-16
GB2357761A (en) 2001-07-04
GB0101504D0 (en) 2001-03-07
CA2475401A1 (en) 2000-12-25
HK1049002B (zh) 2004-12-31
ITMI991581A1 (it) 2001-01-15
CN1502616A (zh) 2004-06-09
CN1367786A (zh) 2002-09-04
ATE235478T1 (de) 2003-04-15
SE0100193D0 (sv) 2001-01-24
WO2000013648A8 (en) 2000-05-11
HUP0103235A3 (en) 2003-01-28
IS5861A (is) 2001-02-23
AT4365U1 (de) 2001-06-25
CA2290127C (en) 2005-01-25
CN1140521C (zh) 2004-03-03
PL205579B1 (pl) 2010-05-31
EP1159274B1 (en) 2003-03-26
BG106191A (en) 2002-08-30
EA200101072A1 (ru) 2002-02-28
BR9917368A (pt) 2002-03-05
CA2290127A1 (en) 2000-12-25
SI1159274T1 (en) 2003-10-31
AT409961B (de) 2002-12-27
EP1159274A2 (en) 2001-12-05

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Representative=s name: PLOUGMANN & VINGTOFT, POSTBOKS 1003 SENTRUM, 0104

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