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NO20010964L - Alkynyl-substituerte quinolin-2-onderivater nyttige som anticancer midler - Google Patents

Alkynyl-substituerte quinolin-2-onderivater nyttige som anticancer midler

Info

Publication number
NO20010964L
NO20010964L NO20010964A NO20010964A NO20010964L NO 20010964 L NO20010964 L NO 20010964L NO 20010964 A NO20010964 A NO 20010964A NO 20010964 A NO20010964 A NO 20010964A NO 20010964 L NO20010964 L NO 20010964L
Authority
NO
Norway
Prior art keywords
alkynyl
anticancer agents
derivatives useful
substituted quinoline
quinoline
Prior art date
Application number
NO20010964A
Other languages
English (en)
Norwegian (no)
Other versions
NO20010964D0 (no
Inventor
Susan Deborah La Greca
Joseph Peter Lyssikatos
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO20010964D0 publication Critical patent/NO20010964D0/no
Publication of NO20010964L publication Critical patent/NO20010964L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20010964A 1998-08-27 2001-02-26 Alkynyl-substituerte quinolin-2-onderivater nyttige som anticancer midler NO20010964L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US9814598P 1998-08-27 1998-08-27
PCT/IB1999/001398 WO2000012499A1 (fr) 1998-08-27 1999-08-06 Derives de quinolin-2-one a substitution alcynyle, utiles en tant qu'agents anticancereux

Publications (2)

Publication Number Publication Date
NO20010964D0 NO20010964D0 (no) 2001-02-26
NO20010964L true NO20010964L (no) 2001-04-26

Family

ID=22267481

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20010964A NO20010964L (no) 1998-08-27 2001-02-26 Alkynyl-substituerte quinolin-2-onderivater nyttige som anticancer midler

Country Status (40)

Country Link
US (3) US6150377A (fr)
EP (1) EP1107963B1 (fr)
JP (1) JP3495706B2 (fr)
KR (1) KR20010072991A (fr)
CN (1) CN1314904A (fr)
AP (1) AP2001002079A0 (fr)
AT (1) ATE321037T1 (fr)
AU (1) AU4925499A (fr)
BG (1) BG105365A (fr)
BR (1) BRPI9913138B8 (fr)
CA (2) CA2578326C (fr)
CO (1) CO5130017A1 (fr)
CZ (1) CZ2001660A3 (fr)
DE (1) DE69930518T2 (fr)
DZ (1) DZ2880A1 (fr)
EA (1) EA200100135A1 (fr)
EE (1) EE200100118A (fr)
ES (1) ES2259237T3 (fr)
GE (1) GEP20033001B (fr)
GT (1) GT199900140A (fr)
HK (1) HK1039123A1 (fr)
HR (1) HRP20010142A2 (fr)
HU (1) HUP0103228A3 (fr)
ID (1) ID27562A (fr)
IL (1) IL141239A0 (fr)
IS (1) IS5818A (fr)
MA (1) MA26680A1 (fr)
NO (1) NO20010964L (fr)
NZ (1) NZ509372A (fr)
OA (1) OA11645A (fr)
PA (1) PA8480101A1 (fr)
PE (1) PE20000986A1 (fr)
PL (1) PL346426A1 (fr)
SK (1) SK2442001A3 (fr)
SV (1) SV1999000141A (fr)
TN (1) TNSN99162A1 (fr)
TR (1) TR200101343T2 (fr)
UY (1) UY25682A1 (fr)
WO (1) WO2000012499A1 (fr)
ZA (1) ZA200101173B (fr)

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Also Published As

Publication number Publication date
US6294552B1 (en) 2001-09-25
TR200101343T2 (tr) 2001-09-21
JP3495706B2 (ja) 2004-02-09
PE20000986A1 (es) 2000-09-30
AU4925499A (en) 2000-03-21
BRPI9913138B8 (pt) 2016-05-17
WO2000012499A1 (fr) 2000-03-09
BR9913138B1 (pt) 2013-11-05
NO20010964D0 (no) 2001-02-26
KR20010072991A (ko) 2001-07-31
HK1039123A1 (zh) 2002-04-12
SV1999000141A (es) 2000-07-06
ZA200101173B (en) 2002-04-12
CN1314904A (zh) 2001-09-26
IS5818A (is) 2001-01-19
GT199900140A (es) 2001-02-14
UY25682A1 (es) 2000-03-31
CZ2001660A3 (cs) 2002-05-15
US20020128287A1 (en) 2002-09-12
US6579887B2 (en) 2003-06-17
IL141239A0 (en) 2002-03-10
EP1107963B1 (fr) 2006-03-22
EE200100118A (et) 2002-06-17
MA26680A1 (fr) 2004-12-20
EA200100135A1 (ru) 2001-08-27
JP2002523504A (ja) 2002-07-30
GEP20033001B (en) 2003-06-25
OA11645A (en) 2004-11-16
CO5130017A1 (es) 2002-02-27
DE69930518T2 (de) 2006-09-21
BR9913138A (pt) 2001-05-08
BG105365A (en) 2001-11-30
ES2259237T3 (es) 2006-09-16
PL346426A1 (en) 2002-02-11
AP2001002079A0 (en) 2001-03-31
PA8480101A1 (es) 2003-06-30
HUP0103228A2 (hu) 2002-02-28
ATE321037T1 (de) 2006-04-15
ID27562A (id) 2001-04-12
HUP0103228A3 (en) 2003-01-28
DZ2880A1 (fr) 2003-12-15
SK2442001A3 (en) 2002-10-08
CA2578326C (fr) 2009-11-24
CA2341690C (fr) 2007-04-17
US6150377A (en) 2000-11-21
CA2578326A1 (fr) 2000-03-09
NZ509372A (en) 2003-08-29
HRP20010142A2 (en) 2002-02-28
TNSN99162A1 (fr) 2005-11-10
CA2341690A1 (fr) 2000-03-09
EP1107963A1 (fr) 2001-06-20
DE69930518D1 (de) 2006-05-11

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