MX9300409A - HEXAHIDROAZEPINONAS AND TETRAHIDROBENZOAZEPINONAS SUBSTITUTED. - Google Patents
HEXAHIDROAZEPINONAS AND TETRAHIDROBENZOAZEPINONAS SUBSTITUTED.Info
- Publication number
- MX9300409A MX9300409A MX9300409A MX9300409A MX9300409A MX 9300409 A MX9300409 A MX 9300409A MX 9300409 A MX9300409 A MX 9300409A MX 9300409 A MX9300409 A MX 9300409A MX 9300409 A MX9300409 A MX 9300409A
- Authority
- MX
- Mexico
- Prior art keywords
- substituted
- tetrahidrobenzoazepinonas
- hexahidroazepinonas
- tetrahydrobenzoazepinones
- haxahydroazepinones
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D223/16—Benzazepines; Hydrogenated benzazepines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Esta invención se refiere a nuevas haxahidroazepinonas y tetrahidrobenzoazepinonas sustituidas estos compuestos son útiles en el tratamiento y preparación de los trastornos gastrointestinales, el dolor y los trastornos de ansiedad.This invention relates to novel substituted haxahydroazepinones and tetrahydrobenzoazepinones these compounds are useful in the treatment and preparation of gastrointestinal disorders, pain and anxiety disorders.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US82567792A | 1992-01-27 | 1992-01-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9300409A true MX9300409A (en) | 1993-07-01 |
Family
ID=25244657
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9300409A MX9300409A (en) | 1992-01-27 | 1993-01-26 | HEXAHIDROAZEPINONAS AND TETRAHIDROBENZOAZEPINONAS SUBSTITUTED. |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP0625145A1 (en) |
| JP (1) | JPH07503465A (en) |
| KR (1) | KR950700257A (en) |
| CN (1) | CN1074903A (en) |
| AU (1) | AU3276193A (en) |
| BR (1) | BR9207071A (en) |
| CA (1) | CA2117367A1 (en) |
| CZ (1) | CZ391092A3 (en) |
| FI (1) | FI943513A0 (en) |
| HU (1) | HUT70496A (en) |
| IL (1) | IL104472A0 (en) |
| MX (1) | MX9300409A (en) |
| NO (1) | NO942775L (en) |
| NZ (1) | NZ245759A (en) |
| RU (1) | RU94038063A (en) |
| TW (1) | TW213901B (en) |
| WO (1) | WO1993015059A1 (en) |
| YU (1) | YU4393A (en) |
| ZA (1) | ZA93582B (en) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2097688A1 (en) * | 1993-07-14 | 1997-04-01 | Pfizer | HEXAHIDROAZEPINONAS AND TETRAHIDROBENZAZEPINONAS SUBSTITUTED. |
| AU6686694A (en) * | 1993-07-26 | 1995-02-20 | Pfizer Inc. | Tetrahydro-1h-benzazepinones and hexahydroazepinones as selective cholecystokinin-b receptor antagonists |
| AU681924B2 (en) * | 1993-11-22 | 1997-09-11 | Merck & Co., Inc. | 3-acylaminobenzazepines |
| US5453424A (en) * | 1993-11-22 | 1995-09-26 | Merck & Co., Inc. | Furanodiazepines |
| CA2200336C (en) * | 1994-10-04 | 2001-12-11 | Pfizer Limited | Processes and intermediates for preparing 3-amino-benzo(b)azepinones |
| ATE210447T1 (en) * | 1994-10-14 | 2001-12-15 | Glaxo Wellcome Spa | USE OF CCK-B RECEPTOR ANTAGONISTS TO TREAT SLEEP DISORDERS |
| DE10153348A1 (en) | 2001-10-29 | 2003-05-08 | Gruenenthal Gmbh | Substituted benzo (b) azepin-2-one compounds |
| MX2007016064A (en) * | 2005-06-16 | 2008-03-10 | Novartis Ag | Compositions and methods for viral inhibition. |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0166357A3 (en) * | 1984-06-26 | 1988-10-26 | Merck & Co. Inc. | Benzofused lactams and pharmaceutical compositions containing them |
| US4767756A (en) * | 1987-07-17 | 1988-08-30 | E. R. Squibb & Sons, Inc. | 3-substituted benzazepines |
| EP0322779A3 (en) * | 1987-12-29 | 1991-05-08 | Yoshitomi Pharmaceutical Industries, Ltd. | Benzolactam compounds and pharmaceutical uses thereof |
| US5206234A (en) * | 1990-10-22 | 1993-04-27 | Merck & Co., Inc. | Benzolactam analogs as antagonists of cck |
-
1992
- 1992-12-15 TW TW081110044A patent/TW213901B/zh active
- 1992-12-16 FI FI943513A patent/FI943513A0/en unknown
- 1992-12-16 BR BR9207071A patent/BR9207071A/en not_active Application Discontinuation
- 1992-12-16 WO PCT/US1992/010720 patent/WO1993015059A1/en not_active Ceased
- 1992-12-16 CA CA002117367A patent/CA2117367A1/en not_active Abandoned
- 1992-12-16 RU RU94038063/04A patent/RU94038063A/en unknown
- 1992-12-16 KR KR1019940702565A patent/KR950700257A/en not_active Ceased
- 1992-12-16 HU HU9402195A patent/HUT70496A/en unknown
- 1992-12-16 AU AU32761/93A patent/AU3276193A/en not_active Abandoned
- 1992-12-16 EP EP93901470A patent/EP0625145A1/en not_active Withdrawn
- 1992-12-16 JP JP5513196A patent/JPH07503465A/en active Pending
- 1992-12-28 CZ CS923910A patent/CZ391092A3/en unknown
-
1993
- 1993-01-21 CN CN93101158A patent/CN1074903A/en active Pending
- 1993-01-21 IL IL104472A patent/IL104472A0/en unknown
- 1993-01-26 MX MX9300409A patent/MX9300409A/en unknown
- 1993-01-26 NZ NZ245759A patent/NZ245759A/en unknown
- 1993-01-26 YU YU4393A patent/YU4393A/en unknown
- 1993-01-27 ZA ZA93582A patent/ZA93582B/en unknown
-
1994
- 1994-07-26 NO NO942775A patent/NO942775L/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2117367A1 (en) | 1993-08-05 |
| WO1993015059A1 (en) | 1993-08-05 |
| NZ245759A (en) | 1997-06-24 |
| BR9207071A (en) | 1995-12-05 |
| EP0625145A1 (en) | 1994-11-23 |
| HU9402195D0 (en) | 1994-09-28 |
| KR950700257A (en) | 1995-01-16 |
| ZA93582B (en) | 1994-07-27 |
| AU3276193A (en) | 1993-09-01 |
| CZ391092A3 (en) | 1994-01-19 |
| JPH07503465A (en) | 1995-04-13 |
| FI943513A7 (en) | 1994-07-26 |
| IL104472A0 (en) | 1993-05-13 |
| TW213901B (en) | 1993-10-01 |
| FI943513L (en) | 1994-07-26 |
| FI943513A0 (en) | 1994-07-26 |
| HUT70496A (en) | 1995-10-30 |
| CN1074903A (en) | 1993-08-04 |
| NO942775D0 (en) | 1994-07-26 |
| YU4393A (en) | 1996-01-09 |
| RU94038063A (en) | 1996-05-27 |
| NO942775L (en) | 1994-09-20 |
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