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MX2022011203A - Compuestos de 9-aminometil minociclina y usos de los mismos. - Google Patents

Compuestos de 9-aminometil minociclina y usos de los mismos.

Info

Publication number
MX2022011203A
MX2022011203A MX2022011203A MX2022011203A MX2022011203A MX 2022011203 A MX2022011203 A MX 2022011203A MX 2022011203 A MX2022011203 A MX 2022011203A MX 2022011203 A MX2022011203 A MX 2022011203A MX 2022011203 A MX2022011203 A MX 2022011203A
Authority
MX
Mexico
Prior art keywords
subject
minocycline
dose
dimethyl
methyl
Prior art date
Application number
MX2022011203A
Other languages
English (en)
Inventor
S Ken Tanaka
Lynne Garrity-Ryan
Evangelos L Tzanis
Amy Manley
Original Assignee
Paratek Pharm Innc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Paratek Pharm Innc filed Critical Paratek Pharm Innc
Publication of MX2022011203A publication Critical patent/MX2022011203A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/65Tetracyclines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/24Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton
    • C07C237/26Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton of a ring being part of a condensed ring system formed by at least four rings, e.g. tetracycline
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se describen métodos y composiciones para usar un compuesto de tetraciclina para tratar infecciones bacterianas. En una modalidad, por ejemplo, la invención proporciona un método para tratar a un sujeto por una infección, que comprende administrar a dicho sujeto una cantidad eficaz de 9-[(2,2-dimetil-propilamino)-m etil]-minociclina o una sal de la misma, de modo que dicho sujeto sea tratado, en donde la 9-[(2,2-dimetil-propilamino)-metil]-minoc iclina se administra por vía oral a una dosis de aproximadamente 450 mg por día durante dos días consecutivos, luego a una dosis de aproximadamente 300 mg por día durante 5 o más días.
MX2022011203A 2016-08-03 2019-02-01 Compuestos de 9-aminometil minociclina y usos de los mismos. MX2022011203A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662370527P 2016-08-03 2016-08-03
US201762514479P 2017-06-02 2017-06-02
US201762532454P 2017-07-14 2017-07-14

Publications (1)

Publication Number Publication Date
MX2022011203A true MX2022011203A (es) 2022-09-19

Family

ID=61074001

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2019001412A MX395671B (es) 2016-08-03 2017-08-03 Compuestos de 9-aminometil minociclina y usos de los mismos.
MX2022011203A MX2022011203A (es) 2016-08-03 2019-02-01 Compuestos de 9-aminometil minociclina y usos de los mismos.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MX2019001412A MX395671B (es) 2016-08-03 2017-08-03 Compuestos de 9-aminometil minociclina y usos de los mismos.

Country Status (14)

Country Link
US (3) US10111890B2 (es)
EP (1) EP3493813A4 (es)
JP (3) JP7225088B2 (es)
CN (1) CN109789153A (es)
AU (3) AU2017305409C1 (es)
BR (1) BR112019001948A2 (es)
CA (1) CA3031790A1 (es)
MX (2) MX395671B (es)
MY (1) MY197146A (es)
PH (1) PH12019500242A1 (es)
RU (1) RU2760186C2 (es)
SG (2) SG11201900379RA (es)
TW (2) TW202206081A (es)
WO (1) WO2018026987A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2010140682A (ru) * 2008-03-05 2012-04-10 Пэрэтек Фамэсьютикэлс, Инк. (US) Способ лечения пациента от инфекции, фармацевтическая композиция (варианты) и лекарственное средство
BR112019008897A2 (pt) 2016-11-01 2019-08-13 Paratek Pharm Innc método para tratar pneumonia bacteriana adquirida na comunidade.
CA3111447A1 (en) * 2018-09-04 2020-03-12 Paratek Pharmaceuticals, Inc. Methods of treating mycobacterial infections using tetracycline compounds
PT117254B (pt) 2021-05-26 2024-04-18 Hovione Farm S A Método de síntese de compostos 9-aminometil tetraciclinas
WO2023238143A1 (en) * 2022-06-11 2023-12-14 Gufic Biosciences Limited A freeze dried parenteral composition of omadacycline tosylate with improved stability

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1434704A (zh) * 1999-12-16 2003-08-06 三叉技术有限责任公司 延长其受体负荷剂量的治疗剂释放的系统和方法
CN101307017A (zh) * 2002-03-08 2008-11-19 帕拉特克药品公司 氨基-甲基取代的四环素类化合物
US7981930B2 (en) * 2007-03-13 2011-07-19 Adamas Pharmaceuticals, Inc. Compositions and kits for treating influenza
RU2010140682A (ru) * 2008-03-05 2012-04-10 Пэрэтек Фамэсьютикэлс, Инк. (US) Способ лечения пациента от инфекции, фармацевтическая композиция (варианты) и лекарственное средство
TW202332671A (zh) * 2008-05-19 2023-08-16 美商Prtk Spv2公司 四環素化合物之甲苯磺酸鹽及同素異形體
KR20240051297A (ko) * 2015-03-24 2024-04-19 파라테크 파마슈티컬스, 인크. 생물방어를 위한 미노시클린 화합물
US20170319603A1 (en) * 2016-03-24 2017-11-09 Paratek Pharmaceuticals, Inc. Methods for treating and preventing c. difficile infection
EP3452048A4 (en) * 2016-05-02 2019-11-13 Paratek Pharmaceuticals, Inc. 9-AMINOMETHYL MINOCYCLINE COMPOUNDS AND METHOD FOR USE THEREOF IN THE TREATMENT OF HARNWEG INFECTIONS (UTI)

Also Published As

Publication number Publication date
TW201808307A (zh) 2018-03-16
US20250275989A1 (en) 2025-09-04
RU2019101842A3 (es) 2020-09-04
US10111890B2 (en) 2018-10-30
AU2017305409B2 (en) 2022-03-17
AU2024205530A1 (en) 2024-08-22
JP2019524767A (ja) 2019-09-05
BR112019001948A2 (pt) 2019-05-07
EP3493813A4 (en) 2020-04-08
TW202206081A (zh) 2022-02-16
CA3031790A1 (en) 2018-02-08
TWI746610B (zh) 2021-11-21
JP2023058586A (ja) 2023-04-25
EP3493813A1 (en) 2019-06-12
MX2019001412A (es) 2019-06-24
WO2018026987A1 (en) 2018-02-08
JP2025041903A (ja) 2025-03-26
MX395671B (es) 2025-03-25
US20180055859A1 (en) 2018-03-01
MY197146A (en) 2023-05-26
PH12019500242A1 (en) 2019-07-29
AU2017305409A1 (en) 2019-03-21
SG10201913574SA (en) 2020-02-27
RU2760186C2 (ru) 2021-11-22
CN109789153A (zh) 2019-05-21
US20190125767A1 (en) 2019-05-02
JP7225088B2 (ja) 2023-02-20
AU2022203977A1 (en) 2022-06-30
RU2019101842A (ru) 2020-09-04
SG11201900379RA (en) 2019-02-27
AU2017305409C1 (en) 2022-06-23

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