MX2020003667A - Sistema terapeutico transdermico para la administracion transdermica de guanfacina que comprende un polimero de silicona. - Google Patents
Sistema terapeutico transdermico para la administracion transdermica de guanfacina que comprende un polimero de silicona.Info
- Publication number
- MX2020003667A MX2020003667A MX2020003667A MX2020003667A MX2020003667A MX 2020003667 A MX2020003667 A MX 2020003667A MX 2020003667 A MX2020003667 A MX 2020003667A MX 2020003667 A MX2020003667 A MX 2020003667A MX 2020003667 A MX2020003667 A MX 2020003667A
- Authority
- MX
- Mexico
- Prior art keywords
- guanfacine
- transdermal
- therapeutic system
- silicone polymer
- transdermal therapeutic
- Prior art date
Links
- INJOMKTZOLKMBF-UHFFFAOYSA-N Guanfacine Chemical compound NC(=N)NC(=O)CC1=C(Cl)C=CC=C1Cl INJOMKTZOLKMBF-UHFFFAOYSA-N 0.000 title abstract 5
- 229960002048 guanfacine Drugs 0.000 title abstract 5
- 230000001225 therapeutic effect Effects 0.000 title abstract 3
- 229920005573 silicon-containing polymer Polymers 0.000 title abstract 2
- 230000003014 reinforcing effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7069—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained otherwise than by reactions only involving carbon to carbon unsaturated bonds, e.g. polysiloxane, polyesters, polyurethane, polyethylene oxide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención se refiere a un sistema terapéutico transdérmico para la administración transdérmica de guanfacina, que comprende una estructura de capa que contiene guanfacina, dicha estructura de capa que contiene guanfacina comprende: A) una capa de refuerzo; y B) una capa que contiene guanfacina en donde el sistema terapéutico transdérmico comprende al menos un polímero de silicona.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762570746P | 2017-10-11 | 2017-10-11 | |
| EP17205543 | 2017-12-05 | ||
| PCT/EP2018/077791 WO2019072997A1 (en) | 2017-10-11 | 2018-10-11 | TRANSDERMAL THERAPEUTIC SYSTEM FOR TRANSDERMAL GUANFACIN ADMINISTRATION COMPRISING A SILICONE POLYMER |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2020003667A true MX2020003667A (es) | 2020-10-01 |
Family
ID=63794520
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2020003667A MX2020003667A (es) | 2017-10-11 | 2018-10-11 | Sistema terapeutico transdermico para la administracion transdermica de guanfacina que comprende un polimero de silicona. |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US11576874B2 (es) |
| EP (1) | EP3694496A1 (es) |
| JP (2) | JP2020536877A (es) |
| KR (1) | KR20200070305A (es) |
| CN (1) | CN111465392B (es) |
| AU (1) | AU2018348801B2 (es) |
| BR (1) | BR112020007091A2 (es) |
| CA (1) | CA3079696A1 (es) |
| MX (1) | MX2020003667A (es) |
| TW (1) | TWI882948B (es) |
| WO (1) | WO2019072997A1 (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2018348801B2 (en) * | 2017-10-11 | 2024-06-27 | Lts Lohmann Therapie-Systeme Ag | Transdermal therapeutic system for the transdermal administration of guanfacine comprising a silicone polymer |
| BR112020007011A2 (pt) | 2017-10-11 | 2020-10-06 | Lts Lohmann Therapie-Systeme Ag | sistema terapêutico transdérmico para a administração transdérmica de guanfacina compreendendo pelo menos um aditivo |
| AU2018348769A1 (en) | 2017-10-11 | 2020-04-16 | Ddp Specialty Electronic Materials Us 9, Llc | Transdermal therapeutic system for the transdermal administration of guanfacine comprising a silicone acrylic hybrid polymer |
| CN114522155B (zh) * | 2020-10-30 | 2024-02-20 | 江苏恒瑞医药股份有限公司 | 一种利多卡因经皮吸收的药物组合物及其制备方法 |
| JP2024517376A (ja) * | 2021-04-06 | 2024-04-22 | ディディピー スペシャルティ エレクトロニック マテリアルズ ユーエス 9 エルエルシー | フィルム形成組成物 |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US4537776A (en) | 1983-06-21 | 1985-08-27 | The Procter & Gamble Company | Penetrating topical pharmaceutical compositions containing N-(2-hydroxyethyl) pyrrolidone |
| US4655767A (en) | 1984-10-29 | 1987-04-07 | Dow Corning Corporation | Transdermal drug delivery devices with amine-resistant silicone adhesives |
| JPS62289514A (ja) * | 1986-04-03 | 1987-12-16 | ハ−コン ラボラトリ−ズ コ−ポレ−シヨン | 薬理活性物質を経皮、経口又は皮下移植により投与する為の製品 |
| JPH01265021A (ja) * | 1987-10-29 | 1989-10-23 | Hercon Lab Corp | 薬理学的活性物質を含有する組成物を動物組織に制御放出および供給するための物品 |
| US5028431A (en) | 1987-10-29 | 1991-07-02 | Hercon Laboratories Corporation | Article for the delivery to animal tissue of a pharmacologically active agent |
| US5656286A (en) * | 1988-03-04 | 1997-08-12 | Noven Pharmaceuticals, Inc. | Solubility parameter based drug delivery system and method for altering drug saturation concentration |
| US5762952A (en) | 1993-04-27 | 1998-06-09 | Hercon Laboratories Corporation | Transdermal delivery of active drugs |
| JPH07145048A (ja) | 1993-11-25 | 1995-06-06 | Sekisui Chem Co Ltd | 医療用貼付剤 |
| US5843472A (en) | 1997-02-28 | 1998-12-01 | Cygnus, Inc. | Transdermal drug delivery sytem for the administration of tamsulosin, and related compositions and methods of use |
| CN100411692C (zh) | 2004-01-13 | 2008-08-20 | 北京康倍得医药技术开发有限公司 | 丙烯酸基粘合剂组合物及其药物组合物和透皮治疗系统 |
| GT200600396A (es) | 2005-09-07 | 2007-04-23 | Dispositivos para la aplicacion de medicamentos transdermicos conteniendo o-desmetil venlafaxina (odv) o sus sales | |
| JP2007284370A (ja) * | 2006-04-14 | 2007-11-01 | Alcare Co Ltd | 体表面用貼付材 |
| US8569416B2 (en) | 2006-06-06 | 2013-10-29 | Dow Corning Corporation | Single phase silicone acrylate formulation |
| US8124689B2 (en) | 2006-06-06 | 2012-02-28 | Dow Corning Corporation | Silicone acrylate hybride composition and method of making same |
| WO2010124187A2 (en) | 2009-04-24 | 2010-10-28 | Henkel Corporation | Silicone acrylic hybrid polymer-based adhesives |
| JP5711743B2 (ja) | 2010-07-29 | 2015-05-07 | 久光製薬株式会社 | 医療用貼付剤 |
| US9080030B2 (en) * | 2010-09-14 | 2015-07-14 | Lorama Group International Inc. | Low VOC and APE free universal paint colourant compositions |
| EP2584016A1 (en) | 2011-10-21 | 2013-04-24 | Dow Corning Corporation | Single phase silicone acrylate formulation |
| JP2013139554A (ja) | 2011-11-29 | 2013-07-18 | Dow Corning Corp | シリコーンアクリレートハイブリッド組成物及び該組成物の製造方法 |
| US20150342899A1 (en) * | 2012-12-28 | 2015-12-03 | Noven Pharmaceuticals, Inc. | Compositions and methods for transdermal delivery of amphetamine and clonidine |
| AU2015296807A1 (en) | 2014-07-31 | 2017-03-09 | Noven Pharmaceuticals, Inc. | Silicone-containing acrylic polymers for transdermal drug delivery compositions |
| WO2016130408A1 (en) | 2015-02-09 | 2016-08-18 | Dow Corning Corporation | Multi-phase silicone acrylic hybrid visco-elastic compositions and methods of making same |
| JP2018526415A (ja) * | 2015-09-14 | 2018-09-13 | アムニール ファーマシューティカルズ エルエルシー | 経皮送達システム |
| AU2018348801B2 (en) * | 2017-10-11 | 2024-06-27 | Lts Lohmann Therapie-Systeme Ag | Transdermal therapeutic system for the transdermal administration of guanfacine comprising a silicone polymer |
| BR112020007011A2 (pt) | 2017-10-11 | 2020-10-06 | Lts Lohmann Therapie-Systeme Ag | sistema terapêutico transdérmico para a administração transdérmica de guanfacina compreendendo pelo menos um aditivo |
| AU2018348769A1 (en) | 2017-10-11 | 2020-04-16 | Ddp Specialty Electronic Materials Us 9, Llc | Transdermal therapeutic system for the transdermal administration of guanfacine comprising a silicone acrylic hybrid polymer |
-
2018
- 2018-10-11 AU AU2018348801A patent/AU2018348801B2/en active Active
- 2018-10-11 KR KR1020207013346A patent/KR20200070305A/ko not_active Ceased
- 2018-10-11 CA CA3079696A patent/CA3079696A1/en active Pending
- 2018-10-11 BR BR112020007091-2A patent/BR112020007091A2/pt not_active IP Right Cessation
- 2018-10-11 JP JP2020519713A patent/JP2020536877A/ja active Pending
- 2018-10-11 EP EP18783027.8A patent/EP3694496A1/en active Pending
- 2018-10-11 TW TW107135783A patent/TWI882948B/zh active
- 2018-10-11 CN CN201880066612.7A patent/CN111465392B/zh active Active
- 2018-10-11 US US16/755,043 patent/US11576874B2/en active Active
- 2018-10-11 WO PCT/EP2018/077791 patent/WO2019072997A1/en not_active Ceased
- 2018-10-11 MX MX2020003667A patent/MX2020003667A/es unknown
-
2023
- 2023-01-11 US US18/152,965 patent/US12168074B2/en active Active
- 2023-06-14 JP JP2023097636A patent/JP7660162B2/ja active Active
Also Published As
| Publication number | Publication date |
|---|---|
| RU2020115503A3 (es) | 2021-12-22 |
| JP2023116687A (ja) | 2023-08-22 |
| US11576874B2 (en) | 2023-02-14 |
| KR20200070305A (ko) | 2020-06-17 |
| US12168074B2 (en) | 2024-12-17 |
| TW201927296A (zh) | 2019-07-16 |
| TWI882948B (zh) | 2025-05-11 |
| AU2018348801A1 (en) | 2020-04-16 |
| AU2018348801B2 (en) | 2024-06-27 |
| JP2020536877A (ja) | 2020-12-17 |
| US20200315987A1 (en) | 2020-10-08 |
| CA3079696A1 (en) | 2019-04-18 |
| EP3694496A1 (en) | 2020-08-19 |
| JP7660162B2 (ja) | 2025-04-10 |
| CN111465392A (zh) | 2020-07-28 |
| WO2019072997A1 (en) | 2019-04-18 |
| US20230241004A1 (en) | 2023-08-03 |
| BR112020007091A2 (pt) | 2020-09-24 |
| RU2020115503A (ru) | 2021-11-12 |
| CN111465392B (zh) | 2024-12-17 |
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