[go: up one dir, main page]

MX2013012187A - Formulaciones topicas de tipo suspension que comprenden depsipeptido ciclico. - Google Patents

Formulaciones topicas de tipo suspension que comprenden depsipeptido ciclico.

Info

Publication number
MX2013012187A
MX2013012187A MX2013012187A MX2013012187A MX2013012187A MX 2013012187 A MX2013012187 A MX 2013012187A MX 2013012187 A MX2013012187 A MX 2013012187A MX 2013012187 A MX2013012187 A MX 2013012187A MX 2013012187 A MX2013012187 A MX 2013012187A
Authority
MX
Mexico
Prior art keywords
cyclic depsipeptide
suspension type
topical formulations
type topical
compositions
Prior art date
Application number
MX2013012187A
Other languages
English (en)
Other versions
MX338156B (es
Inventor
Claire Haug
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46148908&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2013012187(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX2013012187A publication Critical patent/MX2013012187A/es
Publication of MX338156B publication Critical patent/MX338156B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/10—Anti-acne agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La invención se refiere a novedosas composiciones farmacéuticas tópicas en donde el agente activo es un depsipéptido cíclico de la fórmula (II): (ver Fórmula) y a métodos para la elaboración de estas composiciones. La solicitud da a conocer en particular ungüentos hidrofóbicos que comprenden una base hidrofóbica y un agente de consistencia, de preferencia miristato de isopropilo.
MX2013012187A 2011-04-20 2012-04-18 Formulaciones topicas de tipo suspension que comprenden depsipeptido ciclico. MX338156B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161477297P 2011-04-20 2011-04-20
PCT/IB2012/051946 WO2012143868A1 (en) 2011-04-20 2012-04-18 Suspension type topical formulations comprising cyclic depsipeptide

Publications (2)

Publication Number Publication Date
MX2013012187A true MX2013012187A (es) 2013-11-04
MX338156B MX338156B (es) 2016-04-05

Family

ID=46148908

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013012187A MX338156B (es) 2011-04-20 2012-04-18 Formulaciones topicas de tipo suspension que comprenden depsipeptido ciclico.

Country Status (22)

Country Link
US (2) US8680054B2 (es)
EP (1) EP2699231B1 (es)
JP (1) JP5906304B2 (es)
KR (1) KR101612170B1 (es)
CN (1) CN103476396B (es)
AR (1) AR086109A1 (es)
AU (1) AU2012245960B2 (es)
BR (1) BR112013026698A2 (es)
CA (1) CA2833326A1 (es)
CL (1) CL2013003036A1 (es)
EA (1) EA201391555A1 (es)
ES (1) ES2651639T3 (es)
GT (1) GT201300257A (es)
IL (1) IL228863A0 (es)
MA (1) MA35158B1 (es)
MX (1) MX338156B (es)
PE (1) PE20141068A1 (es)
PH (1) PH12013502054A1 (es)
SG (1) SG11201402441WA (es)
TN (1) TN2013000386A1 (es)
TW (1) TW201247218A (es)
WO (1) WO2012143868A1 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20120123579A (ko) 2007-08-17 2012-11-08 노파르티스 아게 시클릭 뎁시펩티드
US8680054B2 (en) 2011-04-20 2014-03-25 Novartis Ag Suspension type topical formulations comprising cyclic depsipeptide
US8614289B2 (en) 2011-04-20 2013-12-24 Novartis Ag Processes for the manufacture of macrocyclic depsipeptides and new intermediates
US9067978B2 (en) 2012-10-09 2015-06-30 Novartis Ag Solution phase processes for the manufacture of macrocyclic depsipeptides and new intermediates
US8987413B2 (en) 2012-10-09 2015-03-24 Novartis Ag Aldehyde acetal based processes for the manufacture of macrocyclic depsipeptides and new intermediates
US9226890B1 (en) 2013-12-10 2016-01-05 Englewood Lab, Llc Polysilicone base for scar treatment
CN108888590A (zh) * 2018-08-06 2018-11-27 江苏知原药业有限公司 包含他克莫司的混悬类型的局部制剂
CN115397398A (zh) * 2020-03-06 2022-11-25 生脉药业股份有限公司 环状酯肽的局部药物制剂

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3043252C2 (de) 1980-11-15 1982-12-02 Degussa Ag, 6000 Frankfurt Cyclische Acetale von N-Acylglutaminsäure -γ- semialdehyden, Verfahren zu deren Herstellung und ihre Verwendung
US5595756A (en) 1993-12-22 1997-01-21 Inex Pharmaceuticals Corporation Liposomal compositions for enhanced retention of bioactive agents
DE4421113A1 (de) 1994-06-16 1995-12-21 Biotechnolog Forschung Gmbh Chondramide, Gewinnungsverfahren, Mittel mit Chondramiden und Mischkultur zur Chondramid-Gewinnung
DE19828043A1 (de) 1998-06-24 1999-12-30 Bayer Ag Ektoparasitizide Mittel
JP2000154198A (ja) 1998-11-20 2000-06-06 Nisshin Flour Milling Co Ltd 環状デプシペプチドの固相合成方法及びその中間体
JP2001131085A (ja) * 1999-08-25 2001-05-15 Saitama Daiichi Seiyaku Kk 経皮・経粘膜吸収用の医薬組成物
GB0108234D0 (en) 2001-04-02 2001-05-23 Pharma Mar Sa Process for producing trunkamide A compounds
US20040110228A1 (en) 2002-04-01 2004-06-10 Mcalpine Shelli R. Combinatorial organic synthesis of unique biologically active compounds
CA2525383C (en) 2003-06-06 2012-03-06 Arexis Ab Use of heterocyclic compounds as scce inhibitors
GB0322140D0 (en) * 2003-09-22 2003-10-22 Pfizer Ltd Combinations
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
EP1716248A1 (en) 2004-02-03 2006-11-02 Bayer HealthCare AG Diagnostics and therapeutics for diseases associated with kallikrein 7 (klk7)
CA2651796A1 (en) 2006-02-27 2007-09-07 Arizona Board Of Regents For And On Behalf Of Arizona State University Identification and use of novopeptides for the treatment of cancer
EP2183270B1 (en) 2007-08-17 2014-12-17 Novartis AG Use of cyclic depsipeptides to inhibit kallikrein 7
KR20120123579A (ko) * 2007-08-17 2012-11-08 노파르티스 아게 시클릭 뎁시펩티드
DE102007052391A1 (de) 2007-10-31 2009-05-07 Henkel Ag & Co. Kgaa Mattwachs
JP2010241784A (ja) * 2008-06-19 2010-10-28 Mitsubishi Tanabe Pharma Corp 経皮投与製剤
US20110112121A1 (en) 2009-07-06 2011-05-12 Joerg Berghausen Pharmaceutical Compositions and Solid Forms
KR101004362B1 (ko) 2010-03-19 2010-12-28 가톨릭대학교 산학협력단 자가 면역 질환 예방 및 치료용 ＴＮＦ－α와 ＴＷＥＡＫ 이중 길항제
US20120064136A1 (en) 2010-09-10 2012-03-15 Nanobio Corporation Anti-aging and wrinkle treatment methods using nanoemulsion compositions
WO2012035468A2 (en) 2010-09-14 2012-03-22 Trima - Israel Pharmaceutical Products Maabarot Ltd. Foamable topical composition
KR20140003572A (ko) 2011-01-24 2014-01-09 안테리오스, 인코퍼레이티드 나노입자 조성물
IL293156A (en) 2011-01-24 2022-07-01 Anterios Inc Nanoparticle compounds, their formulations, and their use
US8680054B2 (en) 2011-04-20 2014-03-25 Novartis Ag Suspension type topical formulations comprising cyclic depsipeptide
US8614289B2 (en) 2011-04-20 2013-12-24 Novartis Ag Processes for the manufacture of macrocyclic depsipeptides and new intermediates
US8987413B2 (en) 2012-10-09 2015-03-24 Novartis Ag Aldehyde acetal based processes for the manufacture of macrocyclic depsipeptides and new intermediates
US9067978B2 (en) 2012-10-09 2015-06-30 Novartis Ag Solution phase processes for the manufacture of macrocyclic depsipeptides and new intermediates

Also Published As

Publication number Publication date
NZ615551A (en) 2015-08-28
EP2699231B1 (en) 2017-09-13
TN2013000386A1 (en) 2015-01-20
CL2013003036A1 (es) 2014-04-04
US20120270796A1 (en) 2012-10-25
PE20141068A1 (es) 2014-09-04
EP2699231A1 (en) 2014-02-26
CA2833326A1 (en) 2012-10-26
AU2012245960A1 (en) 2013-10-17
WO2012143868A1 (en) 2012-10-26
KR101612170B1 (ko) 2016-04-12
ES2651639T3 (es) 2018-01-29
AR086109A1 (es) 2013-11-20
SG11201402441WA (en) 2014-09-26
TW201247218A (en) 2012-12-01
JP5906304B2 (ja) 2016-04-20
MA35158B1 (fr) 2014-06-02
CN103476396A (zh) 2013-12-25
GT201300257A (es) 2015-02-19
KR20130133295A (ko) 2013-12-06
JP2014512377A (ja) 2014-05-22
MX338156B (es) 2016-04-05
AU2012245960B2 (en) 2014-09-25
US9114110B2 (en) 2015-08-25
BR112013026698A2 (pt) 2016-12-27
PH12013502054A1 (en) 2013-12-16
US8680054B2 (en) 2014-03-25
EA201391555A1 (ru) 2014-11-28
US20140162959A1 (en) 2014-06-12
CN103476396B (zh) 2015-08-05
IL228863A0 (en) 2013-12-31

Similar Documents

Publication Publication Date Title
TN2013000386A1 (en) Suspension type topical formulations comprising cyclic depsipeptide
MX2013001677A (es) Formulaciones estables de linaclotida.
MY198204A (en) Cyclic Boronic Acid Ester Derivatives And Therapeutic Uses Thereof
MX2015000813A (es) Composiciones liposómicas de inhibidores de proteasoma basadas en epoxicetona.
MX341324B (es) Polipeptidos.
UA109661C2 (uk) Фармацевтична композиція співкристалів трамадолу і коксибів
MX2019012939A (es) Formulaciones que contienen linaclotida para administracion oral.
NZ708821A (en) Lfa-1 inhibitor formulations
LT2012092A (lt) Fluorinti benzensulfonamidai kaip karboanhidrazės inhibitoriai
IN2012DN00239A (es)
MX2016001422A (es) Composicion farmaceutica de fingolimod.
TR201009167A2 (tr) Sefalosporin içeren farmasötik granüller.
MX2012013607A (es) Polisacarido de las semillas de tamarindo para usarse en el tatamiento de enfermedades inflamatorias.
TR201009394A2 (tr) Geliştirilmiş montelukast formülasyonları.
MX357704B (es) Composiciones farmaceuticas topicas de tipo emulsion aceite en agua que contienen un retinoide.
EA201490573A1 (ru) Соединение бензотиазолона
EA201492280A1 (ru) Стабильный состав пексиганана
TR200909785A1 (tr) Aktif ajan olarak sefdinir içeren farmasötik kompozisyonlar.
WO2011093831A3 (en) Effervescent formulations comprising cefprozil as active agent
IN2014DN10134A (es)
WO2012007758A3 (en) Pharmaceutical formulations
TR201010859A2 (tr) Sefdinir içeren tablet formları.
TR201009166A2 (tr) Sefdinir içeren farmasötik bileşim için üretim yöntemi
TR201009165A2 (tr) Sefdinir içeren tabletler
EA201190243A1 (ru) Стабильная фармацевтическая композиция флударабина фосфата

Legal Events

Date Code Title Description
FG Grant or registration