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MX2011012040A - Compuestos de haloalquil heteroaril benzamida. - Google Patents

Compuestos de haloalquil heteroaril benzamida.

Info

Publication number
MX2011012040A
MX2011012040A MX2011012040A MX2011012040A MX2011012040A MX 2011012040 A MX2011012040 A MX 2011012040A MX 2011012040 A MX2011012040 A MX 2011012040A MX 2011012040 A MX2011012040 A MX 2011012040A MX 2011012040 A MX2011012040 A MX 2011012040A
Authority
MX
Mexico
Prior art keywords
benzamide compounds
haloalkyl heteroaryl
heteroaryl benzamide
haloalkyl
compounds
Prior art date
Application number
MX2011012040A
Other languages
English (en)
Other versions
MX337460B (es
Inventor
J Edward Semple
Jean-Francois Rossignol
Original Assignee
Romark Lab Lc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43069021&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2011012040(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Romark Lab Lc filed Critical Romark Lab Lc
Publication of MX2011012040A publication Critical patent/MX2011012040A/es
Publication of MX337460B publication Critical patent/MX337460B/es

Links

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    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/426—1,3-Thiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
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    • A61K31/445—Non condensed piperidines, e.g. piperocaine
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    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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Abstract

Se describe una nueva clase de haloalquil heteroaril benzamidas. Estos compuestos muestran una fuerte actividad contra los virus de la hepatitis.
MX2011012040A 2009-05-12 2010-05-11 Compuestos de haloalquil heteroaril benzamida. MX337460B (es)

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US17762609P 2009-05-12 2009-05-12
PCT/US2010/034319 WO2010132404A1 (en) 2009-05-12 2010-05-11 Haloalkyl heteroaryl benzamide compounds

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PE20121118A1 (es) 2012-09-05
US8846727B2 (en) 2014-09-30
US9126992B2 (en) 2015-09-08
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CN102803203B (zh) 2016-05-11
NZ596538A (en) 2014-04-30
CA2761876A1 (en) 2010-11-18
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JP5918124B2 (ja) 2016-05-18
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DOP2011000353A (es) 2012-07-31
US20140341850A1 (en) 2014-11-20
CA2940954A1 (en) 2010-11-18
HK1178512A1 (zh) 2013-09-13
KR101760956B1 (ko) 2017-07-24
AP3074A (en) 2014-12-31
EP2429986A1 (en) 2012-03-21
NI201100199A (es) 2012-03-28
IL216331B (en) 2018-06-28
JP2012526820A (ja) 2012-11-01
EA201171378A1 (ru) 2012-05-30
AU2016202439B2 (en) 2017-06-15
JP6193922B2 (ja) 2017-09-06
CN105853415A (zh) 2016-08-17
ECSP11011511A (es) 2012-03-30
HK1223819A1 (zh) 2017-08-11
EP2429986A4 (en) 2012-11-14
USRE46724E1 (en) 2018-02-20
AU2010247816B2 (en) 2015-12-17
CR20110607A (es) 2012-02-13
US20100292274A1 (en) 2010-11-18
CA2761876C (en) 2017-01-03
KR20120036827A (ko) 2012-04-18
BRPI1010547A2 (pt) 2019-04-09
SG10201402281WA (en) 2014-07-30
SG176045A1 (en) 2011-12-29
AP2011006015A0 (en) 2011-12-31
HN2011003002A (es) 2015-08-03
CL2011002830A1 (es) 2012-03-23
MX337460B (es) 2016-03-03

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