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MX2007011453A - Inhibidores de la dipeptidil peptidasa-iv. - Google Patents

Inhibidores de la dipeptidil peptidasa-iv.

Info

Publication number
MX2007011453A
MX2007011453A MX2007011453A MX2007011453A MX2007011453A MX 2007011453 A MX2007011453 A MX 2007011453A MX 2007011453 A MX2007011453 A MX 2007011453A MX 2007011453 A MX2007011453 A MX 2007011453A MX 2007011453 A MX2007011453 A MX 2007011453A
Authority
MX
Mexico
Prior art keywords
dpp
inhibitors
compounds
dipeptidyl peptidase
present
Prior art date
Application number
MX2007011453A
Other languages
English (en)
Inventor
Matthias Schneider
Christoph Steeneck
Frank Richter
Heiko Kroth
Tim Feuerstein
Jurgen Boer
Michael Essers
Bert Nolte
Matthias Hochguertel
Fritz-Frieder Frickel
Arthur Taveras
Original Assignee
Alantos Pharmaceuticals Holding Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36694223&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2007011453(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alantos Pharmaceuticals Holding Inc filed Critical Alantos Pharmaceuticals Holding Inc
Publication of MX2007011453A publication Critical patent/MX2007011453A/es

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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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  • Health & Medical Sciences (AREA)
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  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
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  • Obesity (AREA)
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Abstract

La presente invencion se refiere en general a compuestos inhibidores de la DPP-IV de pirrolidina y tiazolidina. La presente invencion tambien provee metodos de sintesis para la preparacion de tales compuestos, metodos para inhibir la DPP-IV usando tales compuestos y formulaciones farmaceuticas que los contienen para el tratamiento de enfermedades mediadas por DPP-IV, en particular, la diabetes tipo 2.
MX2007011453A 2005-04-22 2006-04-21 Inhibidores de la dipeptidil peptidasa-iv. MX2007011453A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67415105P 2005-04-22 2005-04-22
PCT/US2006/015200 WO2006116157A2 (en) 2005-04-22 2006-04-21 Dipeptidyl peptidase-iv inhibitors

Publications (1)

Publication Number Publication Date
MX2007011453A true MX2007011453A (es) 2008-02-12

Family

ID=36694223

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2007011453A MX2007011453A (es) 2005-04-22 2006-04-21 Inhibidores de la dipeptidil peptidasa-iv.

Country Status (19)

Country Link
US (3) US7553861B2 (es)
EP (1) EP1888562B1 (es)
JP (2) JP4568361B2 (es)
KR (1) KR20080000665A (es)
CN (1) CN101277949A (es)
AP (1) AP2007004234A0 (es)
AU (2) AU2006239929B2 (es)
BR (1) BRPI0608469A2 (es)
CA (1) CA2599419A1 (es)
CR (1) CR9462A (es)
EA (1) EA200702208A1 (es)
ES (1) ES2477868T3 (es)
IL (1) IL186607A0 (es)
MA (1) MA29387B1 (es)
MX (1) MX2007011453A (es)
NO (1) NO20075973L (es)
TN (1) TNSN07244A1 (es)
WO (1) WO2006116157A2 (es)
ZA (1) ZA200708179B (es)

Families Citing this family (73)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
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