ZA9136B - 3-aminopiperidine derivatives and related nitrogen containing heterocycles - Google Patents

3-aminopiperidine derivatives and related nitrogen containing heterocycles

Info

Publication number: ZA9136B
Authority: ZA; South Africa
Prior art keywords: nitrogen containing; containing heterocycles; related nitrogen; aminopiperidine derivatives; aminopiperidine
Prior art date: 1990-01-04

Application number

ZA9136A

Other languages

English (en)

Inventor

Manoj C Desai

C Desai Manoj

Terry J Rosen

J Rosen Terry

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-01-04

Filing date

1991-01-03

Publication date

1992-08-26

1991-01-03 Application filed by Pfizer filed Critical Pfizer

1992-08-26 Publication of ZA9136B publication Critical patent/ZA9136B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/20—Spiro-condensed ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/74—Oxygen atoms
- C07D211/76—Oxygen atoms attached in position 2 or 6
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Immunology (AREA)
Psychiatry (AREA)
Pulmonology (AREA)
Pain & Pain Management (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Anesthesiology (AREA)
Rheumatology (AREA)
Hospice & Palliative Care (AREA)
Dermatology (AREA)
Addiction (AREA)
Hydrogenated Pyridines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Other In-Based Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)

ZA9136A 1990-01-04 1991-01-03 3-aminopiperidine derivatives and related nitrogen containing heterocycles ZA9136B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/US1990/000116 WO1991009844A1 (en)	1990-01-04	1990-01-04	Substance p antagonists

Publications (1)

Publication Number	Publication Date
ZA9136B true ZA9136B (en)	1992-08-26

Family

ID=22220614

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA9136A ZA9136B (en)	1990-01-04	1991-01-03	3-aminopiperidine derivatives and related nitrogen containing heterocycles

Country Status (27)

Country	Link
EP (2)	EP0558156A3 (de)
JP (1)	JPH0757748B2 (de)
KR (1)	KR930009441B1 (de)
CN (2)	CN1035944C (de)
AT (1)	ATE115127T1 (de)
AU (1)	AU625511B2 (de)
BR (1)	BR9100016A (de)
CA (1)	CA2033497C (de)
CZ (1)	CZ289485B6 (de)
DE (1)	DE69014848T2 (de)
DK (1)	DK0436334T3 (de)
ES (1)	ES2064667T3 (de)
FI (2)	FI114096B (de)
GR (1)	GR3014940T3 (de)
HU (5)	HU222724B1 (de)
IE (1)	IE63770B1 (de)
IL (3)	IL96821A (de)
MY (1)	MY105438A (de)
NO (1)	NO178187C (de)
NZ (1)	NZ236581A (de)
PL (5)	PL164244B1 (de)
PT (1)	PT96405B (de)
RU (1)	RU2105758C1 (de)
UA (1)	UA41251C2 (de)
WO (1)	WO1991009844A1 (de)
YU (1)	YU48026B (de)
ZA (1)	ZA9136B (de)

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1990
- 1990-01-04 UA UA5010406A patent/UA41251C2/uk unknown
- 1990-01-04 WO PCT/US1990/000116 patent/WO1991009844A1/en not_active Ceased
- 1990-12-14 AT AT90313680T patent/ATE115127T1/de not_active IP Right Cessation
- 1990-12-14 DE DE69014848T patent/DE69014848T2/de not_active Expired - Fee Related
- 1990-12-14 ES ES90313680T patent/ES2064667T3/es not_active Expired - Lifetime
- 1990-12-14 EP EP19930201034 patent/EP0558156A3/de not_active Ceased
- 1990-12-14 EP EP90313680A patent/EP0436334B1/de not_active Expired - Lifetime
- 1990-12-14 DK DK90313680.2T patent/DK0436334T3/da active
- 1990-12-20 NZ NZ236581A patent/NZ236581A/xx unknown
- 1990-12-28 IL IL96821A patent/IL96821A/xx not_active IP Right Cessation
- 1990-12-28 JP JP2409476A patent/JPH0757748B2/ja not_active Expired - Fee Related
- 1990-12-28 IL IL112348A patent/IL112348A/en not_active IP Right Cessation
1991
- 1991-01-02 PT PT96405A patent/PT96405B/pt active IP Right Grant
- 1991-01-02 PL PL91293389A patent/PL164244B1/pl unknown
- 1991-01-02 PL PL91293392A patent/PL164205B1/pl not_active IP Right Cessation
- 1991-01-02 PL PL91288592A patent/PL163967B1/pl not_active IP Right Cessation
- 1991-01-02 PL PL91293390A patent/PL164203B1/pl not_active IP Right Cessation
- 1991-01-02 HU HU9203403A patent/HU222724B1/hu not_active IP Right Cessation
- 1991-01-02 HU HU916A patent/HUT60719A/hu unknown
- 1991-01-02 CA CA002033497A patent/CA2033497C/en not_active Expired - Fee Related
- 1991-01-02 PL PL91293391A patent/PL164204B1/pl not_active IP Right Cessation
- 1991-01-02 MY MYPI91000002A patent/MY105438A/en unknown
- 1991-01-02 HU HU9203403A patent/HUT68130A/hu unknown
- 1991-01-02 HU HU9203405A patent/HUT68179A/hu unknown
- 1991-01-02 AU AU68621/91A patent/AU625511B2/en not_active Ceased
- 1991-01-02 HU HU9203404A patent/HU220602B1/hu unknown
- 1991-01-03 ZA ZA9136A patent/ZA9136B/xx unknown
- 1991-01-03 YU YU491A patent/YU48026B/sh unknown
- 1991-01-03 CN CN91100039A patent/CN1035944C/zh not_active Expired - Fee Related
- 1991-01-03 KR KR1019910000001A patent/KR930009441B1/ko not_active Expired - Fee Related
- 1991-01-03 FI FI910034A patent/FI114096B/fi active
- 1991-01-03 IE IE791A patent/IE63770B1/en not_active IP Right Cessation
- 1991-01-03 BR BR919100016A patent/BR9100016A/pt not_active Application Discontinuation
- 1991-01-03 NO NO910016A patent/NO178187C/no unknown
- 1991-01-04 CZ CS199110A patent/CZ289485B6/cs not_active IP Right Cessation
- 1991-12-23 RU SU5010406A patent/RU2105758C1/ru not_active IP Right Cessation
1993
- 1993-08-20 CN CN93116286A patent/CN1045595C/zh not_active Expired - Fee Related
1995
- 1995-01-16 IL IL11234895A patent/IL112348A0/xx unknown
- 1995-02-01 GR GR950400206T patent/GR3014940T3/el unknown
2004
- 2004-04-01 FI FI20040479A patent/FI20040479A7/fi not_active Application Discontinuation

Also Published As

Publication number	Publication date
PL163967B1 (pl)	1994-06-30
HUT68180A (en)	1995-05-29
HUT68179A (en)	1995-05-29
FI910034A0 (fi)	1991-01-03
AU6862191A (en)	1991-07-18
CA2033497A1 (en)	1991-07-05
EP0436334B1 (de)	1994-12-07
KR930009441B1 (ko)	1993-10-04
HU222724B1 (hu)	2003-09-29
IL96821A (en)	1997-03-18
CS1091A3 (en)	1991-08-13
BR9100016A (pt)	1991-10-22
PL293390A1 (en)	1992-07-13
IL112348A0 (en)	1995-03-30
YU48026B (sh)	1996-10-09
NO910016D0 (no)	1991-01-03
PL293391A1 (en)	1992-07-13
HUT60719A (en)	1992-10-28
FI20040479A7 (fi)	2004-04-01
PL164204B1 (pl)	1994-06-30
IL112348A (en)	1998-06-15
MY105438A (en)	1994-10-31
UA41251C2 (uk)	2001-09-17
NZ236581A (en)	1992-10-28
FI910034L (fi)	1991-07-05
CN1053060A (zh)	1991-07-17
EP0436334A2 (de)	1991-07-10
WO1991009844A1 (en)	1991-07-11
NO910016L (no)	1991-07-05
DK0436334T3 (da)	1995-02-13
HUT68130A (en)	1995-05-29
YU491A (sh)	1994-01-20
JPH04103570A (ja)	1992-04-06
CN1035944C (zh)	1997-09-24
RU2105758C1 (ru)	1998-02-27
ES2064667T3 (es)	1995-02-01
IL96821A0 (en)	1991-09-16
GR3014940T3 (en)	1995-05-31
FI114096B (fi)	2004-08-13
PL164203B1 (pl)	1994-06-30
HU220602B1 (hu)	2002-03-28
PL164244B1 (en)	1994-07-29
EP0436334A3 (en)	1992-05-27
CA2033497C (en)	1997-01-07
CN1087083A (zh)	1994-05-25
CN1045595C (zh)	1999-10-13
PL293389A1 (en)	1992-07-13
CZ289485B6 (cs)	2002-02-13
PT96405B (pt)	1998-06-30
NO178187B (no)	1995-10-30
HU910006D0 (en)	1991-08-28
IE910007A1 (en)	1991-07-17
PL164205B1 (en)	1994-06-30
KR910014350A (ko)	1991-08-31
PL288592A1 (en)	1992-06-15
EP0558156A3 (de)	1993-10-06
PT96405A (pt)	1991-10-15
AU625511B2 (en)	1992-07-16
IE63770B1 (en)	1995-06-14
ATE115127T1 (de)	1994-12-15
EP0558156A2 (de)	1993-09-01
DE69014848T2 (de)	1995-05-04
JPH0757748B2 (ja)	1995-06-21
DE69014848D1 (de)	1995-01-19
NO178187C (no)	1996-02-07
PL293392A1 (en)	1992-07-13

Publication	Publication Date	Title
EP0436334A3 (en)	1992-05-27	3-aminopiperidine derivatives and related nitrogen containing heterocycles
HU896032D0 (en)	1990-02-28	Process for the preparation of novel quinuc lidine derivatives and pharmaceutical compositions containing them
PH24326A (en)	1990-05-29	Substituted 3,4-dihydro-2h-benzopyrans,pharmaceutical compositions containing same and method of use thereof
ZA913445B (en)	1992-07-29	Process for preparation of 1,5-(alkylimino)-1,5-dideoxy-d-glucitol and derivatives thereof
FI894546A7 (fi)	1990-03-28	Menetelmä uusien 2'-halogeenimetylideeni-, 2'-etenylideeni- ja 2'-etynyyliadenosiinijohdannaisten valmistamiseksi
EG18544A (en)	1994-01-30	Six - membred heterocyclic derivatives of n', - substituted - n, n'-diacylhydrazines
EP0434827A4 (en)	1992-01-08	Quinolinyl-benzopyran derivatives as antagonists of leukotriene d 4?
AP8800109A0 (en)	1989-01-31	"Heterocyclic insecticides".
GB2247237B (en)	1994-05-18	1-(N'-Cyanoguanyl) derivatives of N-containing five-membered ring heterocycles
HU9202510D0 (en)	1992-10-28	Method for producing new 1-benzo-pyrano(4,3)pyrazole derivatives and those of 1-benzo-thiopyrano(4,3)pyrazole and pharmaceutical preparatives containing said compounds
NZ227880A (en)	1991-10-25	Pyridyl substituted 1,3 dioxane alkenoic acid derivatives and pharmaceutical compositions
HU8902302D0 (en)	1990-05-28	Process for preparation of 1,2-hydroxy-phosphonates and derivatives thereof
NZ224812A (en)	1991-06-25	Derivatives of 2',3'-dideoxycytidine and pharmaceutical compositions
IL92759A0 (en)	1990-09-17	Pharmaceutical compositions containing 1,2,3,4-tetrahydroacridine derivatives and certain such novel compounds
GB8903437D0 (en)	1989-04-05	Imidazolyl derivatives of 3,4-dihydro-2h-1-benzothiopyran
NZ223761A (en)	1990-10-26	Preparation of benzo(chalcogeno)(4,3,2-cd)indazole derivatives and certain such compounds
IE862566L (en)	1987-05-12	"new conjugates of vinblastine and its derivatives, a¹process for their preparation and pharmaceutical¹compositions containing the same"
IE861924L (en)	1987-01-22	"new derivatives of diphenoxyethylamine, a process for their¹production and the pharmaceutical compositions containing¹the same"
NZ230987A (en)	1993-03-26	Pyridyl-substituted 1,3 dioxane derivatives and pharmaceutical compositions
HU9802779D0 (en)	1999-02-01	Azol-derivatives of cycloalkylenes and pharmaceutical compositions containing the same
CS8805285A1 (en)	1990-10-12	Connection of grafic table's circuits
IL87498A (en)	1993-08-18	Process for the preparation of 3,3(-disubstituted n-substituted b-lactams, and novel compounds obtained thereby
PL284232A1 (en)	1991-09-23	Method of obtaining novel derivatives of 3,3'/4,6-dihydroxy-m-phenyl/bis(3-phenylphtalide)