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ZA200803894B - Imidazopyrazines as protein kinase inhibitors - Google Patents

Imidazopyrazines as protein kinase inhibitors

Info

Publication number
ZA200803894B
ZA200803894B ZA200803894A ZA200803894A ZA200803894B ZA 200803894 B ZA200803894 B ZA 200803894B ZA 200803894 A ZA200803894 A ZA 200803894A ZA 200803894 A ZA200803894 A ZA 200803894A ZA 200803894 B ZA200803894 B ZA 200803894B
Authority
ZA
South Africa
Prior art keywords
imidazopyrazines
protein kinase
kinase inhibitors
inhibitors
protein
Prior art date
Application number
ZA200803894A
Other languages
English (en)
Inventor
Zhao Lianyun
David B Belanger
Panduranga A Reddy
Timothy J Guzi
Siddiqui M Arshad
Patrick J Curran
Hamann Blake
Paruch Kamil
Michael P Dwyer
Praveen K Tadikonda
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of ZA200803894B publication Critical patent/ZA200803894B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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ZA200803894A 2005-11-10 2008-05-07 Imidazopyrazines as protein kinase inhibitors ZA200803894B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73598205P 2005-11-10 2005-11-10

Publications (1)

Publication Number Publication Date
ZA200803894B true ZA200803894B (en) 2009-03-25

Family

ID=38008330

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200803894A ZA200803894B (en) 2005-11-10 2008-05-07 Imidazopyrazines as protein kinase inhibitors

Country Status (17)

Country Link
US (1) US20070117804A1 (no)
EP (1) EP1945644A2 (no)
JP (1) JP5031760B2 (no)
KR (1) KR20080074963A (no)
CN (1) CN101370811A (no)
AR (1) AR056785A1 (no)
AU (1) AU2006315718B2 (no)
BR (1) BRPI0618520A2 (no)
CA (1) CA2628455A1 (no)
EC (1) ECSP088440A (no)
IL (1) IL191294A0 (no)
NO (1) NO20082530L (no)
PE (1) PE20070805A1 (no)
RU (1) RU2008122967A (no)
TW (1) TW200804386A (no)
WO (1) WO2007058942A2 (no)
ZA (1) ZA200803894B (no)

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