ZA200406332B - ACC inhibitors. - Google Patents

ACC inhibitors. Download PDF

Info

Publication number: ZA200406332B
Authority: ZA; South Africa
Prior art keywords: insulin; moiety; human; patient; conjugate
Prior art date: 2002-02-27

Application number

ZA200406332A

Other languages

English (en)

Inventor

David Austen Perry

Harwood Harold James Jr

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-02-27

Filing date

2004-08-10

Publication date

2005-09-28

2004-08-10 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2005-09-28 Publication of ZA200406332B publication Critical patent/ZA200406332B/en

Links

229940121373 acetyl-coa carboxylase inhibitor Drugs 0.000 title 1
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Diabetes (AREA)
Hematology (AREA)
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Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
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ZA200406332A 2002-02-27 2004-08-10 ACC inhibitors. ZA200406332B (en)

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KR (1)	KR20040095239A (is)
CN (1)	CN1642599A (is)
AT (1)	ATE303178T1 (is)
AU (1)	AU2003248354A1 (is)
CO (1)	CO5601002A2 (is)
DE (1)	DE60301491T2 (is)
EA (1)	EA200400980A1 (is)
ES (1)	ES2246481T3 (is)
HR (1)	HRP20040716A2 (is)
IL (1)	IL163659A0 (is)
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PL (1)	PL372887A1 (is)
TN (1)	TNSN04164A1 (is)
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US7884189B2 (en) *	2003-01-10	2011-02-08	The Trustees Of Columbia University In The City Of New York	Carboxyltransferase domain of acetyl-CoA carboxylase
AU2004212004B2 (en)	2003-02-13	2008-01-10	Albert Einstein College Of Medicine Of Yeshiva University	Regulation of food intake and glucose production by modulation of long-chain fatty acyl-coa levels in the hypothalamus
US20040242566A1 (en)	2003-03-25	2004-12-02	Syrrx, Inc.	Dipeptidyl peptidase inhibitors
EP1625122A1 (en)	2003-05-14	2006-02-15	Takeda San Diego, Inc.	Dipeptidyl peptidase inhibitors
US7169926B1 (en)	2003-08-13	2007-01-30	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
CA2535619A1 (en)	2003-08-13	2005-02-24	Takeda Pharmaceutical Company Limited	4-pyrimidone derivatives and their use as peptidyl peptidase inhibitors
JP2007505121A (ja)	2003-09-08	2007-03-08	武田薬品工業株式会社	ジペプチジルぺプチダーゼ阻害剤
US7371759B2 (en)	2003-09-25	2008-05-13	Bristol-Myers Squibb Company	HMG-CoA reductase inhibitors and method
WO2005044814A1 (en) *	2003-11-07	2005-05-19	F. Hoffmann-La Roche Ag	BENZO [b][1,4] DIOXEPINE DERIVATIVES
GB0326029D0 (en) *	2003-11-07	2003-12-10	Astrazeneca Ab	Chemical compounds
US7420059B2 (en)	2003-11-20	2008-09-02	Bristol-Myers Squibb Company	HMG-CoA reductase inhibitors and method
US7732446B1 (en)	2004-03-11	2010-06-08	Takeda Pharmaceutical Company Limited	Dipeptidyl peptidase inhibitors
GEP20094679B (en)	2004-03-15	2009-05-10	Takeda Pharmaceuticals Co	Dipeptidyl peptidase inhibitors
WO2005113069A2 (en) *	2004-05-14	2005-12-01	Research Development Foundation	Use of circumin and analogues as inhibitors of acc2
US7687638B2 (en)	2004-06-04	2010-03-30	Takeda San Diego, Inc.	Dipeptidyl peptidase inhibitors
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2003
- 2003-02-17 PL PL03372887A patent/PL372887A1/xx not_active Application Discontinuation
- 2003-02-17 DE DE60301491T patent/DE60301491T2/de not_active Expired - Fee Related
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PL372887A1 (en)	2005-08-08
IS7391A (is)	2004-08-09
CN1642599A (zh)	2005-07-20
US6979741B2 (en)	2005-12-27
NZ534582A (en)	2006-03-31
NO20044034L (no)	2004-11-24
AU2003248354A1 (en)	2003-09-09
DE60301491T2 (de)	2006-05-18
DE60301491D1 (en)	2005-10-06
EP1478437A1 (en)	2004-11-24
KR20040095239A (ko)	2004-11-12
HRP20040716A2 (en)	2005-02-28
EA200400980A1 (ru)	2005-02-24
ES2246481T3 (es)	2006-02-16
TNSN04164A1 (fr)	2007-03-12
MA27178A1 (fr)	2005-01-03
CO5601002A2 (es)	2006-01-31
IL163659A0 (en)	2005-12-18
WO2003072197A1 (en)	2003-09-04
EP1478437B1 (en)	2005-08-31
US20030187254A1 (en)	2003-10-02
ATE303178T1 (de)	2005-09-15

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